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Metarrestin

Metarrestin
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Purity:99.04%
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Metarrestin

Catalog No. T12006Cas No. 1443414-10-5
Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis. Metarrestin disrupts the nucleolar structure and inhibits RNA polymerase (Pol) I transcription, at least in part by interacting with the translation elongation factor eEF1A2.
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Pack SizePriceAvailabilityQuantity
1 mg$34In Stock
2 mg$48In Stock
5 mg$80In Stock
10 mg$147In Stock
25 mg$313In Stock
50 mg$538In Stock
100 mg$778In Stock
500 mg$1,620In Stock
1 mL x 10 mM (in DMSO)$84In Stock
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Product Introduction

Bioactivity
Description
Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis. Metarrestin disrupts the nucleolar structure and inhibits RNA polymerase (Pol) I transcription, at least in part by interacting with the translation elongation factor eEF1A2.
AliasML246
Chemical Properties
Molecular Weight474.6
FormulaC31H30N4O
Cas No.1443414-10-5
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 4.75 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.1070 mL10.5352 mL21.0704 mL105.3519 mL
5 mM0.4214 mL2.1070 mL4.2141 mL21.0704 mL

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