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Search Results for " antihistamine "

20

Compounds

Cat No. Product Name Synonyms Targets
T10335 Antihistamine-1 P450
Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).
T25180 Bromodiphenhydramine hydrochloride Others
Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T0211 Azelastine Azelastina,Astelin,Azelastinum SARS-CoV , Histamine Receptor
Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
T1278 Astemizole Laridal,Histaminos,Paralergin Potassium Channel , Histamine Receptor
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re...
T0118 Mizolastine SL 850324 Histamine Receptor
Mizolastine (SL 850324) (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergic rhinitis), hives.
T0211L Azelastine hydrochloride Optivar,Azelastine HCl,Allergodil,Astelin SARS-CoV , Histamine Receptor
Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.
T1030 Triprolidine hydrochloride monohydrate Triprolidine hydrochloride Histamine Receptor
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
T6488 Epinastine hydrochloride Alesion,Epinastine HCl,WAL-801CL HCl,Elestat 5-HT Receptor , Histamine Receptor
Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
T6426 Buclizine dihydrochloride Longifene,Buclina,Buclizine HCl,UCB-4445 5-HT Receptor , AChR , Histamine Receptor
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ...
T6814 Cyproheptadine hydrochloride Periactin hydrochloride,Anarexol,Cyproheptadine HCl,Nuran 5-HT Receptor
Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
T1110 Meclizine dihydrochloride Meclozine dihydrochloride,NSC28728,Meclizine 2HCl Apoptosis , Histamine Receptor
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T2335 Ebastine Ebastel,LAS-W 090,Ebastin,Kestine,RP64305 Histamine Receptor
Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine. It does not penetrate the blood-brain barrier and thus allows an effective block of the H1 receptor in peripheral tiss...
T0205 Brompheniramine maleate Dimotane,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane 5-HT Receptor , Histamine Receptor
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
T0147 Clemastine fumarate HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate) Autophagy , Histamine Receptor
Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T3609 Dioxopromethazine Prothanon,Dioxoprothazine Others
Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.
T0174 Cyproheptadine hydrochloride sesquihydrate Peritol,Periactin hydrochloride,Cyproheptadine hydrochloride 5-HT Receptor , Histone Methyltransferase , Histamine Receptor
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
T7521 Azaphen Pipofezin hydrochloride,Pipofezine hydrochloride,Azafen 5-HT Receptor , Serotonin Transporter
Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.
T4526 Piperoxan hydrochloride dl-Piperoxan hydrochloride,Benodaine hydrochloride Adrenergic Receptor
Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
T25875 Noberastine R64947,T25875,R-64947,R 64947 Histamine Receptor
Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.

Compounds

Antihistamine-1
T10335
Synonym:
Target: P450
Bromodiphenhydramine hydrochloride
T25180
Synonym:
Target: Others
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Azelastine
T0211
Synonym: Azelastina,Astelin,Azelastinum
Target: SARS-CoV, Histamine Receptor
Astemizole
T1278
Synonym: Laridal,Histaminos,Paralergin
Target: Potassium Channel, Histamine Receptor
Mizolastine
T0118
Synonym: SL 850324
Target: Histamine Receptor
Azelastine hydrochloride
T0211L
Synonym: Optivar,Azelastine HCl,Allergodil,Astelin
Target: SARS-CoV, Histamine Receptor
Triprolidine hydrochloride monohydrate
T1030
Synonym: Triprolidine hydrochloride
Target: Histamine Receptor
Epinastine hydrochloride
T6488
Synonym: Alesion,Epinastine HCl,WAL-801CL HCl,Elestat
Target: 5-HT Receptor, Histamine Receptor
Buclizine dihydrochloride
T6426
Synonym: Longifene,Buclina,Buclizine HCl,UCB-4445
Target: 5-HT Receptor, AChR, Histamine Receptor
Cyproheptadine hydrochloride
T6814
Synonym: Periactin hydrochloride,Anarexol,Cyproheptadine HCl,Nuran
Target: 5-HT Receptor
Meclizine dihydrochloride
T1110
Synonym: Meclozine dihydrochloride,NSC28728,Meclizine 2HCl
Target: Apoptosis, Histamine Receptor
Ebastine
T2335
Synonym: Ebastel,LAS-W 090,Ebastin,Kestine,RP64305
Target: Histamine Receptor
Brompheniramine maleate
T0205
Synonym: Dimotane,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
Clemastine fumarate
T0147
Synonym: HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate)
Target: Autophagy, Histamine Receptor
Dioxopromethazine
T3609
Synonym: Prothanon,Dioxoprothazine
Target: Others
Cyproheptadine hydrochloride sesquihydrate
T0174
Synonym: Peritol,Periactin hydrochloride,Cyproheptadine hydrochloride
Target: 5-HT Receptor, Histone Methyltransferase, Histamine Receptor
Azaphen
T7521
Synonym: Pipofezin hydrochloride,Pipofezine hydrochloride,Azafen
Target: 5-HT Receptor, Serotonin Transporter
Piperoxan hydrochloride
T4526
Synonym: dl-Piperoxan hydrochloride,Benodaine hydrochloride
Target: Adrenergic Receptor
Noberastine
T25875
Synonym: R64947,T25875,R-64947,R 64947
Target: Histamine Receptor
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TargetMol