Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment of seasonal allergic rhinitis, asthma, allergic conjunctivitis, and chronic idiopathic urticaria.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 42.00 | |
10 mg | In stock | $ 58.00 | |
25 mg | In stock | $ 94.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 46.00 |
Description | Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment of seasonal allergic rhinitis, asthma, allergic conjunctivitis, and chronic idiopathic urticaria. |
Synonyms | Laridal, Histaminos, Paralergin |
Molecular Weight | 458.57 |
Formula | C28H31FN4O |
CAS No. | 68844-77-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (119.94 mM)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Astemizole 68844-77-9 GPCR/G Protein Immunology/Inflammation Membrane transporter/Ion channel Neuroscience Potassium Channel Histamine Receptor antipruritic hERG K+ Laridal R43512 histamine H1-receptor R 43512 R-43512 KcsA antihistamine drug inhibit Histaminos Inhibitor Paralergin inhibitor