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Azaphen

Catalog No. T7521 CAS 24853-80-3

Synonyms: Pipofezine hydrochloride, Pipofezin hydrochloride, Azafen

Azaphen is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Azaphen, CAS 24853-80-3

Pack Size	Availability	Price/USD
100 mg	In stock	$ 135.00
500 mg	In stock	$ 324.00
1 mL * 10 mM (in Water)	In stock	Inquiry

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Purity: 97.12%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Azaphen is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.

Synonyms	Pipofezine hydrochloride, Pipofezin hydrochloride, Azafen
Molecular Weight	370.28
Formula	C16H21Cl2N5O
CAS No.	24853-80-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 2 years

Solubility Information

DMSO: Insoluble

H2O: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Aleeva G N , Molodavkin G M , Voronina T A . Comparison of Antidepressant Effects of Azafan, Tianeptine, and Paroxetine[J]. Bull Exp Biol Med, 2009, 148(1):54-56.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Parkinson's Disease Compound Library Anti-Neurodegenerative Disease Compound Library Bioactive Compounds Library Max Antidepressant Compound Library GPCR Compound Library Neurotransmitter Receptor Compound Library Inhibitor Library Bioactive Compound Library Neuronal Signaling Compound Library Anti-Cancer Compound Library

Related Products

Related compounds with same targets

Dapoxetine Mesoridazine Besylate F 14679 Piclozotan Syk Inhibitor II SKF-83566 Pardoprunox Auraptenol

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Azaphen 24853-80-3 GPCR/G Protein Neuroscience 5-HT Receptor Serotonin Transporter Pipofezine hydrochloride Pipofezin hydrochloride Pipofezin inhibit Inhibitor Pipofezine SERT 5-HTT SLC6A4 Azafen inhibitor

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