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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T20637 | Diatrizoate meglumine | Reno,Renografin,Renovist,Hypaque,Renocal,Sinografin | Others |
Diatrizoate meglumine (Renocal) is the meglumine salt of diatrizoate, it is an organic, iodinated, radiopaque X-ray contrast medium used in diagnostic radiography. | |||
T2519 | Lercanidipine | Masnidipine | Calcium Channel |
Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class. | |||
T6874 | Lercanidipine hydrochloride | Corifeo,Carmen,Cardiovasc | Calcium Channel |
Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class. | |||
T0354 | Canrenone | 6,7-Dehydro-7α-desthioacetylspironolactone,SC9376,Aldadiene,RP-11614,SC14266 | Glucocorticoid Receptor , Endogenous Metabolite |
Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity. | |||
T8231 | Adrenocorticotropic Hormone (ACTH) (1-39), human | ACTH (1-39), human | Others |
Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor. | |||
T5A2455 | Arenobufagin | Others | |
Arenobufagin is a natural bufadienolide from toad venom with potent antineoplastic activity against HCC HepG2 cells and corresponding multidrug-resistant HepG2/ADM cells. | |||
T7974 | Lynestrenol | Progesterone Receptor | |
Lynestrenol is a synthetic progestational hormone, is the progesterone receptor agonist | |||
T10233 | Acetylarenobufagin | HIF | |
Acetylarenobufagin is a steroidal hypoxia-inducible factor-1 (HIF-1) modulator. | |||
T0870 | Altrenogest | R2267,RU2267,Allyltrenbolone,A35957 | Estrogen/progestogen Receptor , Progesterone Receptor |
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone. | |||
TN6795 | 5-Methoxysuberenone | Others | |
5-Methoxysuberenone is a chemical constituent of the root bark of Toddalia asiatica (L.) Lam. (T. aculeata Pers.), Rutaceae. | |||
T7804 | Garenoxacin mesylate hydrate | Garenoxacin mesylate [USAN],BMS284756 (Mesylate hydrate) | Antibacterial |
Garenoxacin mesylate hydrate (Garenoxacin mesylate [USAN]) with potent antimicrobial activity, against common respiratory pathogens, including resistant strains. | |||
T7567L | Adrenorphin 3TFA(88377-68-8(free base)) | Metorphamide | Opioid Receptor |
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM). | |||
T22236 | Alprenolol hydrochloride | 5-HT Receptor | |
Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor. | |||
T3096 | Canrenoate potassium | Potassium aldadiene,Canrenoic acid potassium salt,Potassium canrenoate,Soldactone | Glucocorticoid Receptor |
Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity. | |||
T13881 | Dicirenone | SC26304 | ATPase , Glucocorticoid Receptor |
Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal cytoplasmic and nuclear receptors. | |||
T3929 | Kaurenoic acid | Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid | Others |
Kaurenoic acid (kaurenoate) has anti-inflammatory potential in acetic acid-induced colitis, decreases in MDA level. Kaurenoic acid exerts a uterine relaxant effect acting principally through calcium blockade and in part,... | |||
TN1459 | Bufarenogin | 3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide | ERK , MEK , PI3K |
Bufarenogin (3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide) is a bufadienolide isolated from parotoid gland secretions of the Cuban endemic toad Peltophryne fustiger. Bufarenogin shows anti-tumor activity. | |||
T15246 | Esaxerenone | XL-550,CS-3150 | Glucocorticoid Receptor |
Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor. | |||
T2677 | Crenolanib | ARO 002,CP-868596 | FLT , PDGFR , Autophagy |
Crenolanib (ARO 002) is an orally bioavailable type III tyrosine kinases inhibitor of PDGFRα/β and FLT3 (IC50s: 11, 3.2, and 4 nM). | |||
T14301 | Apararenone | MT-3995 | Glucocorticoid Receptor |
Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy. |