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20

Compounds

Cat No. Product Name Synonyms Targets
T20637 Diatrizoate meglumine Reno,Renografin,Renovist,Hypaque,Renocal,Sinografin Others
Diatrizoate meglumine (Renocal) is the meglumine salt of diatrizoate, it is an organic, iodinated, radiopaque X-ray contrast medium used in diagnostic radiography.
T2519 Lercanidipine Masnidipine Calcium Channel
Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.
T6874 Lercanidipine hydrochloride Corifeo,Carmen,Cardiovasc Calcium Channel
Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.
T0354 Canrenone 6,7-Dehydro-7α-desthioacetylspironolactone,SC9376,Aldadiene,RP-11614,SC14266 Glucocorticoid Receptor , Endogenous Metabolite
Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.
T8231 Adrenocorticotropic Hormone (ACTH) (1-39), human ACTH (1-39), human Others
Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.
T5A2455 Arenobufagin Others
Arenobufagin is a natural bufadienolide from toad venom with potent antineoplastic activity against HCC HepG2 cells and corresponding multidrug-resistant HepG2/ADM cells.
T7974 Lynestrenol Progesterone Receptor
Lynestrenol is a synthetic progestational hormone, is the progesterone receptor agonist
T10233 Acetylarenobufagin HIF
Acetylarenobufagin is a steroidal hypoxia-inducible factor-1 (HIF-1) modulator.
T0870 Altrenogest R2267,RU2267,Allyltrenbolone,A35957 Estrogen/progestogen Receptor , Progesterone Receptor
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.
TN6795 5-Methoxysuberenone Others
5-Methoxysuberenone is a chemical constituent of the root bark of Toddalia asiatica (L.) Lam. (T. aculeata Pers.), Rutaceae.
T7804 Garenoxacin mesylate hydrate Garenoxacin mesylate [USAN],BMS284756 (Mesylate hydrate) Antibacterial
Garenoxacin mesylate hydrate (Garenoxacin mesylate [USAN]) with potent antimicrobial activity, against common respiratory pathogens, including resistant strains.
T7567L Adrenorphin 3TFA(88377-68-8(free base)) Metorphamide Opioid Receptor
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
T22236 Alprenolol hydrochloride 5-HT Receptor
Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.
T3096 Canrenoate potassium Potassium aldadiene,Canrenoic acid potassium salt,Potassium canrenoate,Soldactone Glucocorticoid Receptor
Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.
T13881 Dicirenone SC26304 ATPase , Glucocorticoid Receptor
Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal cytoplasmic and nuclear receptors.
T3929 Kaurenoic acid Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid Others
Kaurenoic acid (kaurenoate) has anti-inflammatory potential in acetic acid-induced colitis, decreases in MDA level. Kaurenoic acid exerts a uterine relaxant effect acting principally through calcium blockade and in part,...
TN1459 Bufarenogin 3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide ERK , MEK , PI3K
Bufarenogin (3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide) is a bufadienolide isolated from parotoid gland secretions of the Cuban endemic toad Peltophryne fustiger. Bufarenogin shows anti-tumor activity.
T15246 Esaxerenone XL-550,CS-3150 Glucocorticoid Receptor
Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.
T2677 Crenolanib ARO 002,CP-868596 FLT , PDGFR , Autophagy
Crenolanib (ARO 002) is an orally bioavailable type III tyrosine kinases inhibitor of PDGFRα/β and FLT3 (IC50s: 11, 3.2, and 4 nM).
T14301 Apararenone MT-3995 Glucocorticoid Receptor
Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.

Compounds

Diatrizoate meglumine
T20637
Synonym: Reno,Renografin,Renovist,Hypaque,Renocal,Sinografin
Target: Others
Lercanidipine
T2519
Synonym: Masnidipine
Target: Calcium Channel
Lercanidipine hydrochloride
T6874
Synonym: Corifeo,Carmen,Cardiovasc
Target: Calcium Channel
Canrenone
T0354
Synonym: 6,7-Dehydro-7α-desthioacetylspironolactone,SC9376,Aldadiene,RP-11614,SC14266
Target: Glucocorticoid Receptor, Endogenous Metabolite
Adrenocorticotropic Hormone (ACTH) (1-39), human
T8231
Synonym: ACTH (1-39), human
Target: Others
Arenobufagin
T5A2455
Synonym:
Target: Others
Lynestrenol
T7974
Synonym:
Target: Progesterone Receptor
Acetylarenobufagin
T10233
Synonym:
Target: HIF
Altrenogest
T0870
Synonym: R2267,RU2267,Allyltrenbolone,A35957
Target: Estrogen/progestogen Receptor, Progesterone Receptor
5-Methoxysuberenone
TN6795
Synonym:
Target: Others
Garenoxacin mesylate hydrate
T7804
Synonym: Garenoxacin mesylate [USAN],BMS284756 (Mesylate hydrate)
Target: Antibacterial
Adrenorphin 3TFA(88377-68-8(free base))
T7567L
Synonym: Metorphamide
Target: Opioid Receptor
Alprenolol hydrochloride
T22236
Synonym:
Target: 5-HT Receptor
Canrenoate potassium
T3096
Synonym: Potassium aldadiene,Canrenoic acid potassium salt,Potassium canrenoate,Soldactone
Target: Glucocorticoid Receptor
Dicirenone
T13881
Synonym: SC26304
Target: ATPase, Glucocorticoid Receptor
Kaurenoic acid
T3929
Synonym: Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid
Target: Others
Bufarenogin
TN1459
Synonym: 3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide
Target: ERK, MEK, PI3K
Esaxerenone
T15246
Synonym: XL-550,CS-3150
Target: Glucocorticoid Receptor
Crenolanib
T2677
Synonym: ARO 002,CP-868596
Target: FLT, PDGFR, Autophagy
Apararenone
T14301
Synonym: MT-3995
Target: Glucocorticoid Receptor
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TargetMol