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Cat No. | Product Name | Synonyms | Targets |
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T21831 | UCM05 | G28UCM | Fatty Acid Synthase |
UCM05 (G28UCM) is a potent inhibitor of fatty acid synthase (FASN) with efficacy against HER2+ breast cancer xenografts, including in cell lines resistant to anti-HER2 drugs [1]. Additionally, it functions as an inhibito... | |||
T80290 | PP102 | ||
PP102, an antimicrobial peptide, exhibits activity against gram-positive bacteria, including B. subtilis (MIC: 25 µM), S. aureus (MIC: 13.3 µM), S. lutea (MIC: 63 µM), and B. pumilus (MIC: 23 µM) [1]. | |||
T64054 | Antibacterial agent 88 | ||
Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus. | |||
T80288 | PP13 | ||
PP13 is an antimicrobial peptide with efficacy against both Gram-negative and Gram-positive bacteria, displaying minimum inhibitory concentrations (MIC) of 16.7 µM for E. coli, 13.3 µM for B. subtilis, 23.3 µM for S. aur... | |||
T80379 | Cyclopetide 1 | ||
Cyclopeptide 1 (Compound 1) is an antimicrobial peptide exhibiting moderate efficacy in inhibiting B. subtilis, presenting a minimum inhibitory concentration (MIC) of 25 μg/mL [1]. | |||
T80386 | Gageotetrin B | ||
Gageotetrin B exhibits antimicrobial properties, demonstrating higher potency against fungi than bacteria, as evidenced by its MIC (Minimum Inhibitory Concentration) values ranging from 0.01 to 0.04 μM [1]. | |||
T80380 | Cyclopetide 2 | ||
Cyclopeptide 2 (Compound 2) is a moderately active antimicrobial peptide against B. subtilis, exhibiting a minimum inhibitory concentration (MIC) of 50 μg/mL [1]. | |||
T80291 | PP113 | ||
PP113 is an antimicrobial peptide with activity against both Gram-negative and Gram-positive bacteria, exhibiting minimum inhibitory concentrations (MICs) of 73.3 µM for E. coli, 23.3 µM for B. subtilis, 13 µM for S. aur... | |||
T23955 | Dactylfungin B | ||
Dactylfungins B is a novel antifungal antibiotic produced by Dactylaria Parvispora. The antibiotics were active against Candida pseudotropicalis and other fungi, with a MIC value of fewer than 10 micrograms/ml. | |||
T35905 | Oasomycin B | ||
Oasomycin B is a bacterial metabolite that has been found inS. baldaciiand has antiprotozoal activity.1It is active againstT. vaginalis(MIC = 62.5 μg/ml). 1.Grabley, S., Kretzschmar, G., Mayer, M., et al.Secondary metabo... | |||
T79509 | Tuberculosis inhibitor 6 | ||
Tuberculosis inhibitor 6 (compound 2c), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, is highly active against Mycobacterium tuberculosis (MIC 90 of ≤1.66 μM) and Mycobacterium marinum (MIC 90 of 2.65 μM) [1]. | |||
T74771 | Diaporthein B | ||
Diaporthein B, a highly oxidized pimarane diterpene, demonstrates significant activity against M. tuberculosis with a MIC of 3.1 μg/mL and exhibits IC50 values ranging from 1.5-3 μM/L against HCT 116 and LoVo colon cance... | |||
T63252 | Antibacterial agent 113 | ||
Antibacterial agent 113 was an effective antimicrobial agent (antibacterial) against P. aeruginosa, S. mutans, B. subtilis, E. coli, E. faecalis, S. typhimuriumand and S. aureus microorganisms exhibited antibacterial eff... | |||
T80365 | Maximin H39 | ||
Maximin H39, an antimicrobial peptide, exhibits antibacterial activity against C. albicans, S. aureus, and B. subtilis with minimum inhibitory concentrations (MIC) of 9.4, 9.4, and 18.8 μg/mL, respectively. It also demon... | |||
T61123 | Antibacterial agent 111 | ||
Antibacterial agent 111 (Compound 3) exhibits potent antibacterial activity against B. cereus and K. pneumonia, with MIC values of 3.90 μg/mL and 0.49 μg/mL, respectively. It achieves this antibacterial effect by strongl... | |||
T80301 | Aurein 3.1 | Antibiotic | |
Aurein 3.1 is an antibiotic antimicrobial peptide, whereas Aurein 2.6 demonstrates activity against Gram-positive bacteria, exhibiting minimum inhibitory concentrations (MIC) of 80 μM for M. luteus and 50 μM for S. aureu... | |||
T80300 | Aurein 2.6 | Antibiotic | |
Aurein 2.6, an antibiotic antimicrobial peptide, exhibits activity against various Gram-positive bacteria with minimum inhibitory concentrations (MIC) of 25, 25, 30, 25, and 30 μM for M. luteus, S. aureus, S. epidermis, ... | |||
T80369 | Maximin 68 | ||
Maximin 68, an antimicrobial peptide, exhibits antibacterial activity against C. albicans, S. aureus, E. coli, and B. subtilis, with MIC values of 18.8, 9.4, 37.5, and 9.4 μg/mL, respectively. It also possesses hemolytic... | |||
T14115 | Acoziborole | SCYX-7158,AN5568 | Others |
Acoziborole (SCYX-7158), a derivative of benzoxaborole, is a safe, effective and structurally novel antigen-worm agent for human African trypanosomiasis (HAT) studies. The MIC value of Acoziborole for T. b. brucei S427 w... | |||
T61772 | PknB-IN-1 | ||
PknB-IN-1 (Compound 2) is an inhibitor of protein kinase B (PknB) with a concentration causing 50% inhibition (IC50) of 14.4 μM. This compound demonstrates anti-mycobacterial activity by effectively suppressing the growt... | |||
T80364 | Maximin 45 | ||
Maximin 45, an antimicrobial peptide, exhibits antibacterial activity against S. aureus, E. coli, and B. subtilis with minimum inhibitory concentrations (MIC) of 4.7, 9.4, and 75 μg/mL, respectively. Additionally, it pos... | |||
T80368 | Im5 | ||
Im5, an antimicrobial peptide, exhibits antibacterial activity, with minimum inhibitory concentrations (MIC) of 10 μM for E. coli, 2.5-5 μM for S. aureus, and 0.5-1 μM for B. subtilis, as well as hemolytic activity with ... | |||
T35730 | Clindamycin Sulfoxide | ||
Clindamycin sulfoxide is an active metabolite of the antibiotic clindamycin . It is formed via S-oxidation of clindamycin primarily by the cytochrome P450 (CYP) isoform CYP3A4. Clindamycin sulfoxide inhibits the growth o... | |||
T35857 | Actinopyrone A | ||
Actinopyrone A is a pyrone isolated from S. pactum with diverse biological activities. It has selective and potent antimicrobial activity against H. pylori (MIC = 0.1 ng/mL) with no activity against other Gram-negative b... | |||
T75001 | Antibacterial agent 128 | ||
Antibacterial Agent 128, a siderophore analog-Ciprofloxacin (Ciprofloxacin) conjugate connected via a cleavable linker, demonstrates effective antibiotic properties. Specifically, it exhibits activity against P. aerugino... | |||
T79511 | Tuberculosis inhibitor 8 | ||
Tuberculosis inhibitor 8 (compound 3b), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, exhibits potent activity against both Mycobacterium tuberculosis and Mycobacterium marinum with an MIC 90 of 0.69 μM [1]. | |||
T36659 | Boromycin | ||
Boromycin is a boron-containing macrolide antibiotic that has been found in Streptomyces. Boromycin inhibits growth of B. subtilis (MIC = 0.05 μg/ml) and induces efflux of potassium ions from B. subtilis without affectin... | |||
T80367 | Maximin 78 | ||
Maximin 78 is an antimicrobial peptide with antibacterial activity against C. albicans, S. aureus, and B. subtilis, exhibiting minimum inhibitory concentrations (MIC) of 37.5, 4.7, and 37.5 μg/mL, respectively. Additiona... | |||
T64160 | MraY-IN-3 | ||
MraY-IN-3 (12a) is a potent inhibitor of the bacterial translocase MraY (IC50: 140 μM). 46 μg/ml). | |||
T38289 | Leucomycin A13 | Leucomycin A13 | |
Leucomycin A13 is a macrolide antibiotic and a component of the leucomycin complex originally isolated from S. kitasatoensis. It is active against B. subtilis, S. aureus, M. luteus, and E. coli with MIC values of 0.16, 0... | |||
T79510 | Tuberculosis inhibitor 7 | ||
Tuberculosis inhibitor 7 (compound 2d), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, exhibits potent activity against Mycobacterium tuberculosis and Mycobacterium marinum, with both displaying a MIC 90 of 0.6... | |||
T79512 | Tuberculosis inhibitor 9 | ||
Tuberculosis inhibitor 9 (compound 3d), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, exhibits potent activity against Mycobacterium tuberculosis and Mycobacterium marinum, with an MIC 90 of 0.64 μM for both o... | |||
T70798 | Benastatin B | ||
Benastatin B is a polyketide synthase-derived benastatin that has been found in Streptomyces and has diverse biological activities. It inhibits glutathione S-transferase (GST; Ki = 3.7 µM for the rat liver enzyme).2 Bena... | |||
T79479 | MptpB-IN-2 | Antibiotic | |
MptpB-IN-2 (compound 20), a selective inhibitor for mycobacterium tuberculosis protein tyrosine phosphatase B (MptpB), exhibits half maximal inhibitory concentrations (IC50) of 0.64 μM for MptpB, 4.06 μM for MptpA, and 4... | |||
T80277 | CaLL | ||
CaLL, an antimicrobial peptide, exhibits antibacterial activity against B. anthracis, including both its vegetative form, and B. cepacia, with minimum inhibitory concentrations (MICs) of 7.8, 31.3, and 31.3 μg/mL, respec... | |||
T35737 | Emeguisin A | ||
Emeguisin A is a depsidone fungal metabolite originally isolated fromE. unguis.1It is active against the bacteriaS. aureusand methicillin-resistantS. aureus(MRSA; MIC = 0.5 μg/ml for both), the fungusC. neoformans(MIC = ... | |||
T37723 | IT-143A | ||
IT-143A is a bacterial metabolite originally isolated fromStreptomycessp. IT-143.1It is active against the bacteriumM. luteus(MIC = 6.25 μg/ml) and the fungiA. fumigatusandT. rubrumin vitro(MICs = 12.5-25 μg/ml). 1.Uraka... | |||
T35742 | IKD-8344 | ||
IKD-8344 is a macrocyclic dilactone originally isolated from an actinomycete species and has diverse biological activities, including anticancer, antimicrobial, and anthelmintic properties.1,2,3 It is cytotoxic to L5178Y... | |||
T37536 | Carbazomycin A | ||
Carbazomycin A is a bacterial metabolite that has been found in Streptomyces and has diverse biological activities.1,2It is active againstS. aureus,T. asteroides, andT. mentagrophytes(MIC = 12.5 μg/ml for all), as well a... | |||
T79240 | DNA gyrase B-IN-2 | ||
DNA gyrase B-IN-2 (Compound E), a 2-aminobenzothiazole derivative, serves as a potent inhibitor of DNA gyrase B with substantial efficacy against ESKAPE pathogens. The compound exhibits potent nanomolar-range inhibition ... | |||
T75172 | Antibacterial agent 143 | ||
Compound 5a (Antibacterial agent 143) is an antibacterial agent exhibiting minimum inhibitory concentrations (MICs) of 25 μg/mL against B. subtilis ATCC6633 and S. aureus ATCC6538, and 50 μg/mL against P. aeruginosa ATCC... | |||
T13149 | Thiocillin I | Antibacterial | |
Thiocillin I, a thiopeptide antibiotic, demonstrates potent in vitro antibacterial effects against Gram-positive bacteria. This compound exhibits minimum inhibitory concentrations (MICs) of 2 μg/mL, 0.5 μg/mL, 4 μg/mL, a... | |||
T63552 | FtsZ-IN-1 | ||
FtsZ-IN-1 is a potent FtsZ inhibitor with a quinoline ring and has a strong inhibitory effect on Gram-positive bacteria (MIC: 0.5-8 μg/mL).FtsZ-IN-1 enhances FtsZ polymerization and significantly promotes cell elongation... | |||
T37887 | 1-Heptadecanoyl-rac-glycerol | ||
1-Heptadecanoyl-rac-glycerol is a monoacylglycerol that contains heptadecanoic acid at the sn-1 position. It is active against the bacteria E. aerogens, E. cloacae, P. mirabilis, and S. faecalis (MIC = 78 μg/ml for all).... | |||
T38009 | Kocurin | ||
Kocurin is a thiazolyl peptide originally isolated fromK. palustrisand has antibiotic activity.1It is active against methicillin-resistantS. aureus(MRSA; MIC = 0.25 μg/ml), as well asB. subtilisandE. faeciumin a solid ag... | |||
T35978 | Benastatin A | ||
Benastatin A is a polyketide synthase-derived benastatin that has been found inStreptomycesand has diverse biological activities.1,2,3It inhibits glutathione S-transferase (GST; Ki= 5 μM for the rat liver enzyme).2Benast... |
Cat No. | Product Name | Synonyms | Targets |
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T37267 | Pachybasin | Antibacterial | |
Pachybasin is an anthraquinone fungal metabolite. Pachybasin shows antimicrobial activities against E. coli, B. subtilis, M. luteus, S. cerevisiae, C. albicans, A. niger, and A. flavus, with MIC values of 64.0 μg/mL, and... | |||
T71909 | Kumbicin C | ||
Kumbicin C inhibits the growth of NS-1 mouse myeloma cells (IC50 = 0.74 μg/ml) and the growth of the Gram-positive bacteria B. subtilis (MIC = 1.6 μg/ml). | |||
TN5404 | (+)-Conocarpan | ||
Conocarpan has antinociceptive effects. Conocarpan is quite active against S. aureus and B. subtilis with MIC of 6.25 micrograms/ml, it also shows activity against M. tuberculosis (MIC=15.6 ug/ml). Conocarpan shows consi... | |||
TN4098 | Gancaonin I | GTPase , Antifection | |
Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, with a MIC value of 5 uM. | |||
T75476 | Monaschromone | ||
Monaschromone, a polyketide metabolite, effectively suppresses the growth of B. cinerea, A. solani, M. oryzae, and G. saubinettii, demonstrating minimum inhibitory concentration (MIC) values between 6.25 and 12.5 μM [1]. | |||
TN1099 | Dihydroevocarpine | MAO , P-gp , Antifection | |
Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a moderate modulator of p-glycoprotein (p-gp) activity; it s... | |||
T75468 | Asperglaucin B | ||
Asperglaucin B, an alkylated salicylaldehyde derivative isolated from the fungus Aspergillus chevalieri SQ-8, exhibits significant antibacterial properties. This compound demonstrates potent activity against the plant pa... | |||
TN4084 | Fumitremorgin B | Antifection | |
Fumitremorgen B is a mycotoxin, it exhibits a certain degree of genotoxicity, it can cause DNA damage in human lymphocytes; it shows an inhibitory activity on the cell cycle progression of mouse tsFT210 cells in the M ph... | |||
T80343 | MCF | ||
MCF, an antimicrobial peptide originating from bee venom, exhibits activity against E. coli W 160-37, S. aureus 8530, and B. subtilis, with minimum inhibitory concentration (MIC) values of 35-45 μg/ml, 25-35 μg/ml, and 1... | |||
T35761 | Carviolin | ||
Carviolin is an anthraquinone fungal metabolite that has been found inZ. longicaudatawith immunosuppressive and antitrypanosomal activities.1,2It inhibits LPS- or concanavalin A-induced proliferation of mouse splenocytes... | |||
T37442 | Aspergillin PZ | ||
Aspergillin PZ is a fungal metabolite originally isolated from A. awamori. It induces morphological deformation of P. oryzae conidia when used at a concentration of 89 nM. Aspergillin PZ is active against S. epidermidis ... | |||
T36329 | Terpendole I | ||
Terpendole I is a fungal metabolite that has been found in A. yamanashiensis.1 It is a weak inhibitor of acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 145 μM) and is active against the bacteria B. cereus and ... |
Cat No. | Product Name | Species | Expression System |
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TMPK-01243 | GDF-15 Protein, Rat, Recombinant (His) | Rat | E. coli |
Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD... | |||
TMPK-00246 | MICB Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
MICB (MHC class I chain-related gene B) is a transmembrane glycoprotein that functions as a ligand for NKG2D. A closely related protein, MICA, shares 85% amino acid identity with MICB.MICB Seems to have no role in antige... | |||
TMPK-00247 | MICB Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
MICB (MHC class I chain-related gene B) is a transmembrane glycoprotein that functions as a ligand for NKG2D. A closely related protein, MICA, shares 85% amino acid identity with MICB.MICB Seems to have no role in antige... | |||
TMPK-01246 | GDF-15 Protein, Mouse, Recombinant (His) | Mouse | E. coli |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-00245 | MICB Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
MICB (MHC class I chain-related gene B) is a transmembrane glycoprotein that functions as a ligand for NKG2D. A closely related protein, MICA, shares 85% amino acid identity with MICB.MICB Seems to have no role in antige... | |||
TMPY-06711 | B7-1 Protein, Mouse, Recombinant (His & Avi), Biotinylated | Mouse | HEK293 Cells |
B7-1 Protein, Mouse, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 26.94 kDa and the accession number is Q00609-1. | |||
TMPY-02363 | B7-1 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
B7-1 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 50.7 kDa and the accession number is Q00609-1. | |||
TMPY-05811 | B7-1 Protein, Mouse, Recombinant (His), Biotinylated | Mouse | HEK293 Cells |
B7-1 Protein, Mouse, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.1 kDa and the accession number is Q00609-1. | |||
TMPY-02307 | B7-1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
B7-1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.1 kDa and the accession number is Q00609-1. | |||
TMPK-00664 | GDF-15 Protein (Primary Amine Labeling), Cynomolgus, Recombinant (hFc), Biotinylated | Cynomolgus | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-00198 | GDF-15 Protein (Primary Amine Labeling), Human, Recombinant (hFc), Biotinylated | Human | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-00663 | GDF-15 Protein, Cynomolgus, Recombinant (hFc) | Cynomolgus | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-01245 | GDF-15 Protein (Primary Amine Labeling), Mouse, Recombinant (hFc), Biotinylated | Mouse | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-00196 | GDF-15 Protein, Human, Recombinant (His & Avi), Biotinylated | Human | E. coli |
Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD... | |||
TMPK-00197 | GDF-15 Protein (Primary Amine Labeling), Human, Recombinant (H202D, hFc), Biotinylated | Human | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-01244 | GDF-15 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-00569 | GDF-15 Protein, Canine, Recombinant (His) | Canine | E. coli |
Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD... | |||
TMPK-00665 | GDF-15 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | E. coli |
Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t... | |||
TMPK-01416 | HLA-B*15:01&B2M&SARS-CoV-2 epitope (NQKLIANQF) Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
HLA-B*15:01 is strongly associated with asymptomatic infection with SARS-CoV-2 and is likely to be involved in the mechanism underlying early viral clearance. T cells from pre-pandemic individuals carrying HLA-B*15:01 we... | |||
TMPK-01413 | H-2K (b) &B2M&OVA (SIINFEKL) Monomer Protein, Mouse, MHC (His & Avi) | Mouse | HEK293 Cells |
Ovalbumin (OVA) has been historically a popular source of such antigens, since OVA can induce both humoral and cellular immune responses based on well-characterised peptide epitopes. The OVA257-264 octapeptide was one of... | |||
TMPK-01412 | HLA-B*15:01&B2M&SARS-CoV-2 epitope (NQKLIANQF) Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
HLA-B*15:01 is strongly associated with asymptomatic infection with SARS-CoV-2 and is likely to be involved in the mechanism underlying early viral clearance. T cells from pre-pandemic individuals carrying HLA-B*15:01 we... |