Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 74.00 | |
5 mg | In stock | $ 178.00 | |
10 mg | In stock | $ 289.00 | |
25 mg | In stock | $ 572.00 | |
50 mg | In stock | $ 822.00 | |
100 mg | In stock | $ 1,130.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 209.00 |
Description | Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist. |
Synonyms | PF05212365, P -05212365, SAM-531, SAM531, PF-05212365, SAM 531, WAY-262,531 |
Molecular Weight | 409.5 |
Formula | C22H23N3O3S |
CAS No. | 925448-93-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 38 mg/mL (92.80 mM), when pH Adjusted to 3 with HCl. Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. More
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Cerlapirdine 925448-93-7 GPCR/G Protein Neuroscience 5-HT Receptor antagonist inhibit 5-hydroxytryptamine 5-HT6 oral PF05212365 selective Alzheimer's disease Serotonin Receptor P -05212365 SAM-531 SAM531 PF-05212365 5-hydroxytryptamine Receptor Inhibitor PF 05212365 SAM 531 WAY-262,531 inhibitor