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Search Results for " ribosome "

20

Compounds

Cat No. Product Name Synonyms Targets
T1160 Fusidic acid Fusidine Others , CAT , Antibacterial , Antibiotic
Fusidic acid (Fusidine) is an antibiotic isolated from the fermentation broth of Fusidium coccineum.
T16674 Pseudouridine Endogenous Metabolite
Pseudouridine is the most abundant modified nucleoside in non-coding RNAs. It enhances the function of transfer RNA and ribosomal RNA by stabilizing RNA structure.
T8645 PF-06446846 Others
PF 06446846 is a potent and selective PCSK9 inhibitor
T12540 Pristinamycin IA Mikamycin IA,Mikamycin B Others , Antibiotic , P-gp
Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.
T4267 Tulathromycin A CP 472295,Draxxin,Tulathromycin Antibacterial , Antibiotic
Tulathromycin A (CP 472295) is a macrolide antibiotic.
T19459 N1-Methylpseudouridine 1-Methylpseudouridine Others
N1-Methylpseudouridine (1-Methylpseudouridine) is a methylpseudouridine and enhances translation through eIF2α-dependent and independent mechanisms by increasing ribosome density in mRNA.
T17143 Toyocamycin Vengicide Apoptosis , Others , IRE1 , Antibiotic , Antifungal
Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (IC50: 80 nM). Toyocamycin induces apoptosis.
T0788 Spectinomycin dihydrochloride Spectinomycin 2HCl,Actinospectacin ribosome , Antibacterial , Antibiotic
Spectinomycin dihydrochloride (Actinospectacin) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.
T1289 Fusidic acid sodium salt Sodium fusidate,Fusidate Sodium,Fucidin,SQ-16360 Others , CAT , Antibacterial , Antibiotic
Fusidic acid sodium salt (SQ-16360) is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections.
T0788L Spectinomycin dihydrochloride pentahydrate Trobicin,Spectogard,Spectinomycin hydrochloride hydrate ribosome , Antibacterial , Antibiotic
Spectinomycin dihydrochloride pentahydrate (Spectogard) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.
T7148 JOSAMYCIN EN-141 Antibacterial , Antibiotic
Josamycin (EN-141) is a macrolide antibiotic exhibiting antimicrobial activity. The dissociation constant Kd from ribosome for Josamycin is 5.5 nM.
T28506 Rbin-2 Phosphatase
Rbin-2 is a cell-permeable, potent, selective and reversible inhibitor of Midasin (Mdn1).Rbin-2 directly targets the AAA+ ATPase Midasin and inhibits eukaryotic ribosome production, making it a potent probe for the study...
T7411 Rbin-1 Ribozinoindole-1 ATPase , Phosphatase
Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.
T13767 MBX-4132 Others , Antibacterial
MBX-4132, inhibit trans translation by binding to the bacterial ribosome,is a member of a chemical class called oxadiazoles.
T4222 KKL-10 KKL 10 ribosome , Antibacterial
KKL-10, a ribosome rescue inhibitor, has broad-spectrum antimicrobial activity against bacteria.
T1557 Acetylspiramycin Spiramycin II,Foromacidin B,ASPM,Spiramycin B ribosome , Antibacterial , Antibiotic
Acetylspiramycin (Spiramycin B) targets 50S ribosome to inhibit protein synthesis.
T3265 Azathramycin Desmethyl Azithromycin,6-Demethylazithromycin,Azaerythromycin A,Azaerythromycin Antibacterial , Antibiotic
Azathramycin (Desmethyl Azithromycin) is an antibiotic derived from erythromycin, binding to the 50S subunit of the bacterial ribosome, and thus inhibits translation of mRNA.
T6758 Anisomycin Flagecidin,NSC 76712,Wuningmeisu C Apoptosis , DNA/RNA Synthesis , Antibacterial , Antibiotic , JNK
Anisomycin (NSC-76712) is an antibiotic isolated from various Streptomyces species. It interferes with protein and DNA synthesis by inhibiting peptidyl transferase or the 80S ribosome system.
T1214 Ribostamycin sulfate Vistamycin sulfate Antibacterial , Antibiotic
Ribostamycin sulfate (Vistamycin sulfate) , an aminoglycoside antibiotic, contains a neutral sugar moiety and is produced by Streptomyces ribosome.
T1747 Tedizolid TR 700,DA-7157,Torezolid MAO , Antibacterial , Antibiotic
Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of the ribosome.

Compounds

Fusidic acid
T1160
Synonym: Fusidine
Target: Others, CAT, Antibacterial, Antibiotic
Pseudouridine
T16674
Synonym:
Target: Endogenous Metabolite
PF-06446846
T8645
Synonym:
Target: Others
Pristinamycin IA
T12540
Synonym: Mikamycin IA,Mikamycin B
Target: Others, Antibiotic, P-gp
Tulathromycin A
T4267
Synonym: CP 472295,Draxxin,Tulathromycin
Target: Antibacterial, Antibiotic
N1-Methylpseudouridine
T19459
Synonym: 1-Methylpseudouridine
Target: Others
Toyocamycin
T17143
Synonym: Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
Spectinomycin dihydrochloride
T0788
Synonym: Spectinomycin 2HCl,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Fusidic acid sodium salt
T1289
Synonym: Sodium fusidate,Fusidate Sodium,Fucidin,SQ-16360
Target: Others, CAT, Antibacterial, Antibiotic
Spectinomycin dihydrochloride pentahydrate
T0788L
Synonym: Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
JOSAMYCIN
T7148
Synonym: EN-141
Target: Antibacterial, Antibiotic
Rbin-2
T28506
Synonym:
Target: Phosphatase
Rbin-1
T7411
Synonym: Ribozinoindole-1
Target: ATPase, Phosphatase
MBX-4132
T13767
Synonym:
Target: Others, Antibacterial
KKL-10
T4222
Synonym: KKL 10
Target: ribosome, Antibacterial
Acetylspiramycin
T1557
Synonym: Spiramycin II,Foromacidin B,ASPM,Spiramycin B
Target: ribosome, Antibacterial, Antibiotic
Azathramycin
T3265
Synonym: Desmethyl Azithromycin,6-Demethylazithromycin,Azaerythromycin A,Azaerythromycin
Target: Antibacterial, Antibiotic
Anisomycin
T6758
Synonym: Flagecidin,NSC 76712,Wuningmeisu C
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, JNK
Ribostamycin sulfate
T1214
Synonym: Vistamycin sulfate
Target: Antibacterial, Antibiotic
Tedizolid
T1747
Synonym: TR 700,DA-7157,Torezolid
Target: MAO, Antibacterial, Antibiotic
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TargetMol