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Search Results for " mycobacteria "

20

Compounds

Cat No. Product Name Synonyms Targets
T14830 Bromperidol R-11333 5-HT Receptor
Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic. Which is used as an antipsychotic in the treatment of schizophrenia.
T0972 Isoniazid INH,Isonicotinic acid hydrazide,Isonicotinic hydrazide Mitophagy , Dehydrogenase , CAT , Antibacterial , Autophagy
Isoniazid (Isonicotinic hydrazide) is an antibacterial agent used primarily as a tuberculostatic.
T0793 Kanamycin sulfate Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan ribosome , Antibacterial , Antibiotic
Kanamycin sulfate (Kanamycin monosulfate) is an aminoglycoside bacteriocidal antibiotic.
T60073 Antimycobacterial agent-4 4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide Antibacterial
Antimycobacterial agent-4 (4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide) has antibacterial activity against Mycobacterium tuberculosis.
T63420 Antimycobacterial agent-2
Antimycobacterial agent-2 is an effective anti-mycobacterial agent with a MIC99 of 0.8 μM against Mycobacterium tuberculosis (M.tb) H37Rv. Antimycobacterial agent-2 is cytotoxic, acting on CHO cells (IC50: 48.1 μM).
T61853 Antimycobacterial agent-1
Antimycobacterial agent-1 (compound 33) demonstrates potent antimycobacterial activity against Mycobacterium tuberculosis H37Ra, with a minimal inhibitory concentration (MIC) value of 1 μg/ml. Notably, antimycobacterial ...
T72306 Mycobacterial Zmp1-IN-1
Mycobacterial Zmp1-IN-1, a zinc metalloprotease-1 (Zmp1) inhibitor, demonstrates dose-dependent anti-mycobacterial activity against Mtb H37Ra, making it suitable for tuberculosis (TB) research.
T79281 Antimycobacterial agent-6
Antimycobacterial agent-6 (compound 25) effectively inhibits Mycobacterium tuberculosis, including wild-type and fluoroquinolone-resistant strains, by targeting the Mtb DprE1-C387S mutant. It displays minimal inhibitory ...
T63865 Antimycobacterial agent-3
Antimycobacterial agent-3 is an antimycobacterial agent with low cytotoxicity. antimycobacterial agent-3 is effective against sensitive MTB strain H37Rv and resistant clinical isolates (MIC < 0.029-0.110 μ M).
T7518 Deoxycytidine triphosphate trisodium salt 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE TRISODI Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis , Endogenous Metabolite , Antibiotic
Deoxycytidine triphosphate trisodium salt (2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE TRISODI) contributes to antibiotic lethality in stationary-phase mycobacteria.
T21023 Bedaquiline fumarate TMC 207,R403323,TMC-207,TMC207,R-403323,R 403323 Antibacterial , Antibiotic
Bedaquiline fumarate (TMC207), a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections. It blocks the proton pump for ATP synthase of mycobacteria. ...
T0377 Clofazimine NSC-141046 DNA , Antibacterial , Antibiotic
Clofazimine (NSC-141046) is a phenazine dye with anti-mycobacterial and anti-inflammatory activities. Clofazimine has a slow bactericidal effect on Mycobacterium leprae and is active against various other Mycobacteria.
T23979 Deoxypheganomycin D
Deoxypheganomycin D is a specific mycobacteria inhibitor.
T26189 Setomimycin AM 2947,Antibiotic A 39183B,AM2947,AM-2947
Setomimycin is an antibiotic against Gram positive bacteria, including mycobacteria.
T25955 Picromycin Antibiotic B 62169A,Amaromycin,Albomycetin,Pikromycin
Picromycin is a 14-membered macrolide antibiotic and Prolyl endopeptidase (PREP) inhibitor. Pikromycin shows activity against gram-positive bacteria including mycobacteria.
TN6057 1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone (Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one
(Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one shows strong inhibitory activity on leukotriene biosynthesis in human polymorphonuclear granulocytes, and it is very effective against mycobacteria.
T33537 Mycobactin P
Mycobactin P is one of iron(III) chelating compounds produced by most species of Mycobacteria which act as growth factors.
T62840 Bromperidol hydrochloride
Bromperidol hydrochloride (R-11333 hydrochloride) is an antipsychotic agent with good affinity for the central dopamine receptors D2. Spectinomycin synergistically kills mycobacteria.
T40520 Thiophene-2 Thiophene-2,TP2
Thiophene-2 (TP2) is a targeted inhibitor of polyketide synthase 13 (Pks13), specifically designed to disrupt mycolic acid biosynthesis. By doing so, it effectively induces rapid cell death in mycobacteria. Thiophene-2 d...
T16749 Rifalazil KRM-1648,ABI-1648 DNA/RNA Synthesis
Rifalazil is a rifamycin derivative, inhibits the bacterial DNA-dependent RNA polymerase and kills bacterial cells by blocking off the β-subunit in RNA polymerase. Rifalazil is an antibiotic, exhibits high potency agains...

Compounds

Bromperidol
T14830
Synonym: R-11333
Target: 5-HT Receptor
Isoniazid
T0972
Synonym: INH,Isonicotinic acid hydrazide,Isonicotinic hydrazide
Target: Mitophagy, Dehydrogenase, CAT, Antibacterial, Autophagy
Kanamycin sulfate
T0793
Synonym: Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan
Target: ribosome, Antibacterial, Antibiotic
Antimycobacterial agent-4
T60073
Synonym: 4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide
Target: Antibacterial
Antimycobacterial agent-2
T63420
Synonym:
Target:
Antimycobacterial agent-1
T61853
Synonym:
Target:
Mycobacterial Zmp1-IN-1
T72306
Synonym:
Target:
Antimycobacterial agent-6
T79281
Synonym:
Target:
Antimycobacterial agent-3
T63865
Synonym:
Target:
Deoxycytidine triphosphate trisodium salt
T7518
Synonym: 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE TRISODI
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, Endogenous Metabolite, Antibiotic
Bedaquiline fumarate
T21023
Synonym: TMC 207,R403323,TMC-207,TMC207,R-403323,R 403323
Target: Antibacterial, Antibiotic
Clofazimine
T0377
Synonym: NSC-141046
Target: DNA, Antibacterial, Antibiotic
Deoxypheganomycin D
T23979
Synonym:
Target:
Setomimycin
T26189
Synonym: AM 2947,Antibiotic A 39183B,AM2947,AM-2947
Target:
Picromycin
T25955
Synonym: Antibiotic B 62169A,Amaromycin,Albomycetin,Pikromycin
Target:
1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone
TN6057
Synonym: (Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one
Target:
Mycobactin P
T33537
Synonym:
Target:
Bromperidol hydrochloride
T62840
Synonym:
Target:
Thiophene-2
T40520
Synonym: Thiophene-2,TP2
Target:
Rifalazil
T16749
Synonym: KRM-1648,ABI-1648
Target: DNA/RNA Synthesis
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TargetMol