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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3278 | Piribedil | EU-4200,Trivastan,ET-495,Trivastal | Dopamine Receptor , Histone Methyltransferase , Adrenergic Receptor |
Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease. | |||
T21935L | AMN082 free base | AMN082 | GluR |
AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist. | |||
T6140 | SB-334867 free base | SB334867A free base,SB-334867,SB 334867,SB334867 | OX Receptor |
SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist. | |||
T21935 | AMN082 | AMN 082 dihydrochloride | GluR |
AMN082 (AMN 082 dihydrochloride) is a selective metabotropic glutamate mGlu7 receptor agonist reported to exhibit antidepressant activity. | |||
T35033 | Vamicamide | FK 176,FK-176,FK176 | AChE |
Vamicamide (FK 176) is a novel anticholinergic compound. Vamicamide increases spontaneous locomotor activity in mice at 32 mg/kg (p.o.) or higher and inhibits cataleptic convulsions in mice at 100 mg/kg. | |||
T35033L | (S)-Vamicamide | (S)-Vamicamide (Iso-132373-81-0) | AChE |
(S)-Vamicamide is a novel anticholinergic compound.Vamicamide increases spontaneous locomotor activity in mice at 32 mg/kg or higher (p.o.) and inhibits tonic convulsions in mice at 100 mg/kg.CAS 번호13483-86-1 | |||
TP1940L1 | Ac-RYYRIK-NH2 acetate | Opioid Receptor | |
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the sti... | |||
TMS1461 | Qingyangshengenin B | Otophylloside B | Beta Amyloid |
Qingyangshengenin B (Otophylloside B) is a C-21 steroidal glycoside isolated from Qingyangshen. Qingyangshengenin B protects against Aβ toxicity, which decreases Aβ deposition by decreasing the expression of Aβ at the mR... | |||
T21792 | CGP 3466B maleate | Omigapil (Maleate),Omigapil maleate | Apoptosis |
CGP 3466B maleate (Omigapil maleate) is an orally bioavailable GAPDH nitrosylation inhibitor. Omigapil maleate abrogates Aβ1-42-induced tau acetylation, memory impairment, and locomotor dysfunction in mice. Omigapil male... | |||
T3685 | SR9009 | Stenabolic,REV-ERB Agonist II | Autophagy |
SR9009 (Stenabolic), a REV-ERB agonist, increases the constitutive repression of genes regulated by REV-ERBα/ERBβ (IC50: 670/800 nM). Through activation of REV-ERB, SR9009 can decrease circadian locomotor activity during... | |||
T37190 | L-Allylglycine | Dehydrogenase , GABA Receptor | |
L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo in mouse brain preparations. L-Allylglycine (1.2 mmol/kg, ... | |||
T32440 | L 363572 | L363-572,L-363572,L-363-572,L363572,L 363-572 | |
L 363572, a hexapeptide analog of MK 678, does not effect locomotor acitivity in rats. | |||
T81659 | NocII TFA | ||
NocII TFA, an orphan neuropeptide, stimulates locomotor activity in mice [1]. | |||
TP1982 | Neuropeptide S(Rat) | Neuropeptide S (Rat) | |
Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM). Increases locomotor activity and wakefulness in mice. Also reduces anxiety-like behavior in mice. | |||
TN4722 | Otophylloside F | Others | |
Otophylloside F can suppress the seizure-like locomotor activity caused by pentylenetetrazole in zebrafish. | |||
T75951 | Neuropeptide S(Rat) TFA | ||
Neuropeptide S(Rat) TFA, a robust endogenous agonist for the neuropeptide S receptor (NSPR) with an EC50 of 3.2 nM, enhances locomotor activity and promotes wakefulness while concurrently diminishing anxiety-like behavio... | |||
TP1983 | Neuropeptide S (human) | ||
Potent endogenous neuropeptide S receptor agonist (EC50 = 9.4 nM). Increases locomotor activity and wakefulness in mice. Also reduces anxiety-like behavior in mice. | |||
T28313 | PD 117302 | PD-117302,PD117302 | |
PD 117302 is a nonpeptide opioid compound. It is a selective kappa-opioid agonist. PD 117302 causes naloxone-reversible locomotor impairment and diuresis. It is an Anti-Arrhythmia Agent, an Anticonvulsants, a Cardiovascu... | |||
T29230 | ZK-95962 | ||
ZK-95962 is an agonist gamma-aminobutyric acid (GABA) receptor. ZK-95962 had selective effects on releasing exploratory locomotor activity suppressed by footshock (punished crossings). ZK-95962 had weak effects on the me... | |||
TP1981 | Neuropeptide S(Mouse) | Neuropeptide S (Mouse) | |
Potent endogenous neuropeptide S receptor (NPSR) agonist (EC50 = 3 nM). Induces mobilization of intracellular Ca2+. Increases locomotor activity and wakefulness in mice. Also reduces anxiety-like behavior in mice. |