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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7736 | 2-Chloroadenosine | Adenosine Receptor | |
2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively) | |||
T11014 | DFP00173 | Aquaporin | |
DFP00173 is a potent and selective aquaporin 3 (AQP3) inhibitor. DFP00173 inhibits mouse and human AQP3 with IC50 of ~0.1-0.4 μM. Compared with the homologous AQP subtypes AQP7 and AQP9, DFP00173 is selective for AQP3. | |||
T5239 | Cholesteryl sulfate sodium | Cholesterol 3-Sulfate Sodium Salt,Sodium Cholesteryl Sulfate | Endogenous Metabolite , PKC |
Cholesteryl sulfate sodium (Sodium Cholesteryl Sulfate) is a sterol sulfate in human plasma. Cholesteryl sulfate sodium is a component of cell membrane and has a regulatory function. Cholesteryl sulfate sodium also activ... | |||
T4466 | Pitofenone hydrochloride | Baralgin Ketone Hydrochloride,Pitophenone hydrochloride | AChE |
Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively. | |||
TN1369 | Alloimperatorin | Prangenidin | Others |
Alloimperatorin (Prangenidin) exhibits in vitro antitumor activity in HL-60 acute myeloid leukemia cancer cells via inducing apoptosis, cell cycle disruption and inhibition of cell migration. It photosensitizes efficient... | |||
TN3790 | Dehydroabietinol | Pomiferin A,Dehydroabietyl alcohol | Antifection |
Dehydroabietinol (Pomiferin A) inhibits growth of chloroquine-sensitive as well as chloroquine-resistant strains of Plasmodium falciparum cultivated in erythrocytes in vitro (IC 50 26-27 microM). | |||
TN3601 | Carminic acid | ROS | |
Carminic acid, the well-known red dyestuff from cochineal insects (Dactylopius spp.), is a potent feeding deterrent to ants. Carminic acid is an antioxidant to protect erythrocytes and DNA against radical-induced oxidati... | |||
T25588 | L589-420 | L 589-420,L-589-420,L-589 420,L 589 420,L589 420 | |
L589-420 is a sodium pump inhibitor in human erythrocytes. | |||
TN1007 | 3-Epidehydrotumulosic acid | Others | |
3-Epidehydrotumulosic acid exhibits inhibitory effects on AAPH-induced haemolysis of erythrocytes. | |||
T69131 | Pitofenone | ||
Pitofenone is an inhibitor of the acetylcholinesterase activity from bovine erythrocytes and electric eel. | |||
T71422 | S6821 | ||
S6821 is a TAS2R8 antagonist. S6821 was not found to be mutagenic or clastogenic in vitro, and did not induce micronuclei in bone marrow polychromatic erythrocytes in vivo. | |||
T71806 | Tenellin | ||
Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells. | |||
T82827 | Bombolitin III | ||
Bombolitin III, an antimicrobial peptide sourced from bumblebee venom, possesses lytic activity against erythrocytes and liposomes [1]. | |||
T6432 | Calpeptin | Apoptosis , Cysteine Protease , Proteasome | |
Calpeptin is a potent, cell-permeable calpain inhibitor. | |||
T82826 | Bombolitin IV | ||
Bombolitin IV, an antimicrobial peptide obtained from bumblebee venom, has the ability to lyse erythrocytes and liposomes [1]. | |||
T36795 | Donepezil N-oxide | ||
Donepezil N-oxide is an active metabolite of the acetylcholinesterase inhibitor donepezil . Donepezil N-oxide inhibits cholinesterase (ChE) activity in human erythrocytes in a concentration-dependent manner, exhibiting 4... | |||
T36766 | Palmitoylcholine (chloride) | ||
Palmitoylcholine is an acyl choline.1It inhibits protein kinase C activity when used at a concentration of 100 μM.2Palmitoylcholine induces hemolysis in rat erythrocytes.3Plasma levels of palmitoylcholine are decreased i... | |||
T82829 | Bombolitin I | ||
Bombolitin I, an antimicrobial peptide originating from bumblebee venom, possesses the ability to lyse erythrocytes and liposomes [1]. | |||
TN1728 | Hellebrigenin | PARP , Akt , CDK | |
Hellebrigenin has anti-hepatoma activities, it induces cell cycle arrest and apoptosis in human hepatocellular carcinoma HepG2 cells through inhibition of Akt. Hellebrigenin exhibites moderate to strong activity against ... | |||
T82828 | Bombolitin II | ||
Bombolitin II, an antimicrobial peptide originating from bumblebee venom, possesses the ability to lyse erythrocytes and liposomes [1]. |