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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60075 | Dopamine D2 receptor agonist-2 | Dopamine D2 Receptor | Dopamine Receptor |
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor. | |||
T11077 | Dopamine D2 receptor antagonist-1 | Others | |
Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity. | |||
T7635 | Raclopride | Dopamine Receptor | |
Raclopride is a selective antagonist of dopamine D2/D3 receptor. | |||
T4007 | Eticlopride hydrochloride | Dopamine Receptor | |
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM). | |||
T16392 | ONC206 | Dopamine Receptor | |
ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and possesses broad-spectrum anti-tumor activity. | |||
TQ0084 | Lumateperone Tosylate | ITI-007 | Dopamine Receptor , 5-HT Receptor |
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki: 32 nM). | |||
T0280 | Spiperone | Spiroperidol,Spiropitan | Dopamine Receptor |
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds. It has been recommended in the treatment of SCHIZOPHRENIA. | |||
T21069 | Lumateperone | ITI 722,ITI722,ITI-007,ITI007 | 5-HT Receptor |
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM). | |||
T7943 | Fluphenazine decanoate | Dopamine Receptor | |
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia. | |||
T2226 | Pergolide mesylate | Pergolide mesylate salt,LY127809,Pergolide methanesulfonate | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor |
Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to potential for HEART VALVE DISEASES. | |||
T8136 | Perospirone hydrochloride | Perospirone HCl,SM-9018 hydrochloride | Dopamine Receptor , 5-HT Receptor |
Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia. It also displays affinity towards 5HT1A receptors as a partial agonist. | |||
T1045 | Trimipramine maleate | Surmontil maleate | Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor |
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal... | |||
T10683 | Carmoxirole hydrochloride | EMD 45609 hydrochloride | Dopamine Receptor |
Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity in vivo. | |||
T9228 | Propionylpromazine hydrochloride | Propiopromazine hydrochloride | Dopamine Receptor |
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist. | |||
T70302 | Fallypride | Dopamine Receptor | |
Fallypride is a potent and selective dopamine D2/D3 receptor antagonist. | |||
T3497 | Ocaperidone | Ocaperidona,R79598 | Dopamine Receptor , 5-HT Receptor |
Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist. | |||
T22817 | GSK 789472 hydrochloride | GSK-789472 HCl,1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride,4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one | Dopamine Receptor |
GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist. | |||
T0302 | Triflupromazine hydrochloride | Neoprin,Fluopromazine hydrochloride,Fluorofen,Flumazin | Dopamine Receptor , 5-HT Receptor , AChR , Autophagy |
Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists. | |||
T7180 | Sultopride hydrochloride | LIN-1418 hydrochloride | Dopamine Receptor |
Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist. | |||
T6142 | PD128907 HCl | Dopamine Receptor | |
PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor. |