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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4563 | Thonzylamine | neohetramine | Histamine Receptor |
Thonzylamine (neohetramine) is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of symptoms of common cold, hay fever (allergic rhin... | |||
T1269 | Tripelennamine hydrochloride | Pyribenzamine hydrochloride,Tripelennamine HCl,Pyribenzamine HCl | Histamine Receptor |
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation. | |||
T67953 | Elbanizine | Others | |
Elbanizine showed antiallergic, antiasthmatic, antihistaminic, and spasmolytic activity. | |||
T25180 | Bromodiphenhydramine hydrochloride | Others | |
Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous. | |||
T22508 | 3-CPMT | Chlortropbenzyl hydrochloride,3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octane hydrochloride,SL6057,Wy 2149,FC-1 | Dopamine Receptor |
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent. | |||
T22354 | Levocetirizine Dihydrochloride | Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride | Histamine Receptor |
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro... | |||
T1470L | Fexofenadine hydrochloride | Histamine Receptor | |
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic activity. | |||
T0776 | Phenothiazine | ENT 38 | Dopamine Receptor , Antibacterial , Antibiotic , Antifungal |
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities. Phenothiazines antagonize the dopamine D2-receptor in the chemoreceptor trigger zone (CTZ)... | |||
T1266 | Terfenadine | (±)-Terfenadine,MDL-991 | Apoptosis , Potassium Channel , 5-HT Receptor , Caspase , Na+/Ca2+ Exchanger , HER , AChR , Histamine Receptor |
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects. | |||
T0370 | Pheniramine maleate | Daneral,Inhiston,Trimetose | 5-HT Receptor , Histamine Receptor |
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of the endothelium-derived re... | |||
T1278 | Astemizole | Laridal,Histaminos,Paralergin | Potassium Channel , Histamine Receptor |
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re... | |||
T32707 | Levomequitazine | ||
Levomequitazine is an antihistaminic drug candidate. | |||
T20709 | Levocabastine hydrochloride | R50,547,R-50,547,Levocabastine HCl,R 50,547,Livostin | |
Levocabastine HCl is an agent with antihistaminic activity. | |||
T23679 | AHR-13268D | AHR 13268D,AHR13268D | |
AHR-13268D is a new agent of antiallergic/antihistaminic. | |||
T69016 | Piprinhydrinate | ||
Piprinhydrinate is a Histamine H₁-receptor antagonist (H₁-antihistaminic). | |||
T82476 | Embramine hydrochloride | ||
Embramine hydrochloride is a monoethanolamine derivative utilized for its antihistaminic and anticholinergic properties [1]. | |||
T70773 | Noberastine citrate | ||
Noberastine citrate, a histamine H1 antagonist, has potent and specific peripheral antihistaminic activity. Noberastine, a furan derivative of nor-astemizole (an astemizole metabolite), has been shown to have a more rapi... | |||
T69071 | Secoverine | ||
Secoverine is a selective muscarinic receptor antagonist that was studied as a neurotropic spasmolytic agent. It was shown that the drug had no nicotinolytic or antihistaminic activity, a moderate antisterotonic activity... | |||
T71425 | Noberastine maleate | ||
Noberastine maleate, a histamine H1 antagonist, has potent and specific peripheral antihistaminic activity. Noberastine, a furan derivative of nor-astemizole (an astemizole metabolite), has been shown to have a more rapi... |