Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
50 mg | In stock | $ 36.00 | |
100 mg | In stock | $ 50.00 | |
200 mg | In stock | $ 75.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 50.00 |
Description | Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects. |
Targets&IC50 | ERG (human):204 nM |
Synonyms | (±)-Terfenadine, MDL-991 |
Molecular Weight | 471.67 |
Formula | C32H41NO2 |
CAS No. | 50679-08-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 47.2 mg/mL(100 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Terfenadine 50679-08-8 Angiogenesis Apoptosis GPCR/G Protein Immunology/Inflammation JAK/STAT signaling Membrane transporter/Ion channel Neuroscience Proteases/Proteasome Tyrosine Kinase/Adaptors Potassium Channel 5-HT Receptor Caspase Na+/Ca2+ Exchanger HER AChR Histamine Receptor inhibit MDL 991 MDL991 (±)-Terfenadine Inhibitor MDL-991 KcsA inhibitor