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20

Compounds

Cat No. Product Name Synonyms Targets
T10003 α1 adrenoceptor-MO-1 Others
α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.
T12643 (R)-Terazosin Adrenergic Receptor
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively).
T13016 SR59230A Adrenergic Receptor
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T2524 Dexmedetomidine Adrenergic Receptor
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of dexmedetomidine is by means of General Anesthesia.
T1132 Nicergoline Nicergolinum,Nimergoline Adrenergic Receptor
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T22033 ARC 239 dihydrochloride Norepinephrine
ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).
T20898 (R)-Propranolol hydrochloride Dexpropranolol hydrochloride,(R)-(+)-Propranolol Adrenergic Receptor
(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol. Propranolol is a nonselective β-adrenergic receptor (βAR) antag...
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T22236 Alprenolol hydrochloride 5-HT Receptor
Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.
T5S2059 Glaucine Calcium Channel , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , PDE
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 production. Glaucine can inhibit the migration and invasion of h...
T6579 Medetomidine hydrochloride MPV785,Medetomidine HCl,Domitor Adrenergic Receptor
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
T6466 Dexmedetomidine hydrochloride Precedex,(+)-Medetomidine hydrochloride,(S)-Medetomidine hydrochloride,Dexmedetomidine HCl Adrenergic Receptor
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is the racemic form of this compound.
T3046 BMY 7378 dihydrochloride BMY7378 HCl Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T0137 Mirtazapine 6-Azamianserin,Org3770 Dopamine Receptor , 5-HT Receptor , Opioid Receptor , Adrenergic Receptor , Histamine Receptor
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevations in serum aminotransferase levels and h...
T0197 Terazosin hydrochloride Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic Adrenergic Receptor
Terazosin hydrochloride (Hytrin) , a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for patients with prostate enlargement and h...
T6701 Terazosin hydrochloride dihydrate Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate Adrenergic Receptor
Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
T11286 Fiduxosin A 185980.1,ABT 980 Adrenergic Receptor
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin...
T9220 Naftopidil hydrochloride 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride Adrenergic Receptor
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, respective...
T1239 Indacaterol maleate QAB149 Adrenergic Receptor
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
T11015 Midaglizole hydrochloride (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128 Adrenergic Receptor
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenocepto...

Compounds

α1 adrenoceptor-MO-1
T10003
Synonym:
Target: Others
(R)-Terazosin
T12643
Synonym:
Target: Adrenergic Receptor
SR59230A
T13016
Synonym:
Target: Adrenergic Receptor
Dexmedetomidine
T2524
Synonym:
Target: Adrenergic Receptor
Nicergoline
T1132
Synonym: Nicergolinum,Nimergoline
Target: Adrenergic Receptor
ARC 239 dihydrochloride
T22033
Synonym:
Target: Norepinephrine
(R)-Propranolol hydrochloride
T20898
Synonym: Dexpropranolol hydrochloride,(R)-(+)-Propranolol
Target: Adrenergic Receptor
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Alprenolol hydrochloride
T22236
Synonym:
Target: 5-HT Receptor
Glaucine
T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
Medetomidine hydrochloride
T6579
Synonym: MPV785,Medetomidine HCl,Domitor
Target: Adrenergic Receptor
Dexmedetomidine hydrochloride
T6466
Synonym: Precedex,(+)-Medetomidine hydrochloride,(S)-Medetomidine hydrochloride,Dexmedetomidine HCl
Target: Adrenergic Receptor
BMY 7378 dihydrochloride
T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Mirtazapine
T0137
Synonym: 6-Azamianserin,Org3770
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
Terazosin hydrochloride
T0197
Synonym: Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic
Target: Adrenergic Receptor
Terazosin hydrochloride dihydrate
T6701
Synonym: Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate
Target: Adrenergic Receptor
Fiduxosin
T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Naftopidil hydrochloride
T9220
Synonym: 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride
Target: Adrenergic Receptor
Indacaterol maleate
T1239
Synonym: QAB149
Target: Adrenergic Receptor
Midaglizole hydrochloride
T11015
Synonym: (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128
Target: Adrenergic Receptor
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TargetMol