active — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
TP1555L1	Fibronectin Active Fragment Control acetate	Fibronectin Active Fragment Control acetate(97461-84-2 Free base)
	Fibronectin Active Fragment Control acetate is an active fragment of fibronectin which is a glycoprotein.
T5401	GSK2983559 active metabolite	GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1	RIP kinase
	GSK2983559 active metabolite (RIPK2-IN-1) is a potent, selective receptor-interacting protein-2 (RIP2) kinase inhibitor.		RIP kinase
TP1555	Fibronectin Active Fragment Control
	Fibronectin is a high-molecular weight (~440kDa) extracellular matrix glycoprotein that binds to membrane-spanning receptor proteins called integrins.In addition to integrins, fibronectin also binds extracellular matrix ...
T14122	Active-mono-sulfone-PEG8-acid		Others
	Active-mono-sulfone-PEG8-acid is a polyethylene glycol (PEG) derivative serving as a linker for PROTAC synthesis[1].		Others
T10480	Bay 41-4109 (less active enantiomer)		HBV
	Bay 41-4109 less active enantiomer shows less activity than Bay 41-4109. BAY 41-4109 is a potent HBV inhibitor (IC50: 53 nM).		HBV
T19667	R-138727	Prasugrel active metabolite
	R-138727 is a novel P2Y12 receptor inhibitor.
T29705	AG-2000 Free Base	Lansoprazole sulfenamide active metabolite
	AG-2000 Free Base is a bio-active chemical. Detailed information has not been published.
T13646	Desisobutyryl-ciclesonide	CIC-AP,Ciclesonide active principle	Others
	Desisobutyryl-ciclesonide has an affinity for glucocorticoid receptors. Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide.		Others
T29704	AG-1812 free base	UNII-6RI44GB0V9,HE078804,AC1MIZB6,Lansoprazole disulfide active metabolite
	ABT-1812 is a bio-active chemical.
T9966	GSK-1520489A		Wee1
	GSK-1520489A is an active PKMYT1 inhibitor.		Wee1
T8348	Phentolamine		Adrenergic Receptor
	Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist		Adrenergic Receptor
T8580	Bupranolol		Adrenergic Receptor
	Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.		Adrenergic Receptor
T9565	OSBPL7-IN-1		Others
	OSBPL7-IN-1 is an orally active inhibitor of oxysterol binding protein like 7 (OSBPL7). OSBPL7-IN-1 promotes an increase of ABCA1 at the plasma membrane without affecting mRNA expression[1].		Others
T9732	VY-3-135		Fatty Acid Synthase
	VY-3-135 is a metastasis inhibitor and an acetyl-CoA synthetase 2 (ACSS2) modulator.		Fatty Acid Synthase
T1292	Tiapride hydrochloride		Dopamine Receptor
	Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing dyskinesia, negative symptoms of psychosis, alcohol withdraw...		Dopamine Receptor
T8734	Choline		Others
	Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins		Others
T20525	Chloramphenicol palmitate		Antibacterial , Antibiotic
	Chloramphenicol palmitate is a broad-spectrum antibiotic with activity against gram-positive and gram-negative bacteria. Chloramphenicol palmitate can be used in studies about acting as a bacterial selection agent in tra...		Antibacterial , Antibiotic
T34896	Tofisopam	Emandaxin,Grandaxin	Others
	Tofisopam (Grandaxin) is a 2,3-benzodiazepine compound with anxiolytic activity that can be taken orally.		Others
T11351	Galanthamine N-Oxide		AChE
	Galanthamine N-Oxide, an alkaloid extracted from Zephyranthes concolor bulbs, effectively inhibits acetylcholinesterase (AChE) from electric eel with an EC50 of 26.2 μM. It acts as a significant inhibitor of substrate ac...		AChE
T40732	TMPD dihydrochloride
	TMPD dihydrochloride is an active substrate of enzymatically convert redox and an electron donor for the reduction of heme peroxidases.