acetate-dependent — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
TP1271L	Calmodulin-Dependent Protein Kinase II 290-309 acetate	Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)	CaMK
	Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).		CaMK
T75959	Calmodulin-Dependent Protein Kinase II(290-309) acetate
	Calmodulin-Dependent Protein Kinase II (290-309) acetate is a potent antagonist of CaMK, exhibiting an IC50 of 52 nM for the inhibition of Ca2+/calmodulin-dependent protein kinase II [1].
T4380	Ac-CoA Synthase Inhibitor1	ACSS2 inhibitor	RSV , Fatty Acid Synthase
	Ac-CoA Synthase Inhibitor1 (ACSS2 inhibitor) is the most potent and specific inhibitor of acetate-dependent acetyl-CoA synthetase 2 (ACSS2).		RSV , Fatty Acid Synthase
TP1485L	Calcineurin substrate acetate		Autophagy
	Calcineurin substrate acetate is from the regulatory RII subunit of cAMP-dependent protein kinase.		Autophagy
T21470L	Davunetide acetate	Davunetide acetate(211439-12-2 Free base)	Beta Amyloid , Microtubule Associated
	Davunetide acetate is derived from activity-dependent neuroprotective protein existing in the mammalian CNS. Davunetide acetate is a microtubule-stabilizing peptide and inhibits Aβ aggregation and Aβ-induced neurotoxicit...		Beta Amyloid , Microtubule Associated
T40437L	Caloxin 2A1 acetate		Proton pump
	Caloxin 2A1 acetate is an inhibitor of extracellular plasma membrane Ca2+-ATPase (PMCA) peptide. Caloxin 2A1 acetate inhibits Ca2+-dependent formation of the 140-kDa acid-stable acylphosphate.		Proton pump
T4946	(+)-Columbianetin acetate	COLUMBIANETIN ACETATE	Others
	(+)-Columbianetin acetate (COLUMBIANETIN ACETATE) may be helpful in regulating mast cell-mediated allergic inflammatory responses.The absorption of (+)-Columbianetin acetate is a passive diffusion process without pH-depe...		Others
T37422L	Ras Inhibitory Peptide acetate	Ras Inhibitory Peptide acetate(159088-48-9 Free base)	Ras
	Ras Inhibitory Peptide acetate is a peptide involved in the Ras-dependent signaling pathway that plays an important role in human cancers initiated by oncogenic receptors.		Ras
TP1403L	Syntide 2 acetate(108334-68-5 free base)		CaMK
	Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).		CaMK
TP2018L	GIP (human) acetate	GIP (human) acetate(100040-31-1 Free base)	IGF-1R
	GIP (human) acetate is a stimulator of glucose-dependent insulin secretion and a weak inhibitor of gastric acid secretion. GIP (human) acetate plays a vital role in lipid metabolism and the development of obesity.		IGF-1R
T37588L	GIP (1-30) amide, porcine acetate		IGF-1R
	GIP (1-30) amide, porcine acetate is an agonist of fully glucose-dependent insulinotropic polypeptide (GIP) receptor. GIP (1-30) amide, porcine acetate can weakly inhibit gastric acid secretion and strongly stimulate ins...		IGF-1R
T21983L	PKI 14-22 amide, myristoylated Acetate	PKI 14-22 amide, myristoylated Acetate(201422-03-9 Free base)	PKA
	PKI 14-22 amide, myristoylated Acetate inhibit cAMP-dependent protein kinase (PKA) and blocks hyperalgesia produced by spinal administration of 8-bromo-cAMP.		PKA
TP1914L1	BAM (8-22) acetate	BAM (8-22) acetate(412961-36-5 free base)	Others
	BAM (8-22) acetate is a proteolytically cleaved product of proenkephalin A. BAM (8-22) acetate activates Mas-related G-protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces scratching in mice in an Mrgpr...		Others
TP1220L	Carperitide acetate	Carperitide acetate (89213-87-6 Free base),Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate	Endothelin Receptor
	Carperitide acetate (Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate), a 28-amino acid hormone, is naturally produced and released by the human heart upon cardiac injury or mechanical stretch. This compou...		Endothelin Receptor
TP1909L1	CALP2 acetate(261969-04-4 free base)		CaMK , PDE
	CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM. CALP2 acetate potently inhibits of adhesion and degranulation. CALP2 acetate is als...		CaMK , PDE
T21309	Nafarelin acetate(76932-56-4 free base)	RS-94991-298,Nafarelin acetate,Nafarelin acetate hydrate,Synarel	GNRH Receptor
	Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing h...		GNRH Receptor
T3650	STO-609 acetate		CaMK
	STO-609 acetate is selective, cell-permeable inhibitor of Ca2+-calmodulin-dependent protein kinase kinase (Ki: 80/15 ng/ml, for CaM-KKα/KKβ); competes for the ATP-binding site. It displays > 80-fold selectivity over CaMK...		CaMK
TP1789L	Malantide acetate(86555-35-3 free base)		PKA , PKC
	Malantide acetate is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activ...		PKA , PKC
TP1787L	PKG Substrate acetate（81187-14-6 free base)		PKA
	PKG Substrate acetate is a selective substrate for cGMP-dependent protein kinase (PKG).PKG Substrate is a selective substrate for protein kinase G (PKG) with a strong preference for PKG Iα (Km = 59 μM) over PKG II (Km = ...		PKA
TP1051L	Protein Kinase C Peptide Substrate acetate	Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)	Others
	Protein Kinase C Peptide Substrate acetate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-couple...		Others