t9 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T13246	UCT943		Parasite , PI4K
	UCT943 is an inhibitor of Plasmodium falciparum PI4K (IC50 = 23 nM).		Parasite , PI4K
T7302	CU-CPT9b	CU-CPT-9b,TLR8-specific antagonist 1	TLR
	CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM). It inhibits activation of NF- B induced by the TLR8 agonist R-848 in TLR8-overexpressing HEK-Blue cells with an IC50 valu...		TLR
T5207	LIT927	LIT 927,LIT-927	CXCR
	LIT927 (LIT-927) is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to CXCR4).		CXCR
T14841	BVT948		Phosphatase , P450 , Histone Methyltransferase
	BVT948 is a protein tyrosine phosphatase (PTP) inhibitor. It can also inhibit several CYP450 isoforms and lysine methyltransferase SETD8 (KMT5A).		Phosphatase , P450 , Histone Methyltransferase
T3068	AT9283	J-504568	Apoptosis , FLT , JAK , Bcr-Abl , Aurora Kinase , Autophagy
	AT9283 (J-504568) is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora B and Abl(T315I).		Apoptosis , FLT , JAK , Bcr-Abl , Aurora Kinase , Autophagy
T4354	KPT9274	KPT-9274,KPT 9274,PAK4-IN-1	NAMPT , PAK
	KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.		NAMPT , PAK
T33616	NDT9520492	NDT 9520492,NDT-9520492
	NDT9520492 is a bioactive chemical.
T76593	(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)
	Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon), a gonadotropin-releasing hormone (GnRH) analog, effectively induces ovulation and/or spawning in farmed fish [1].
T69227	GT951
	GT951 is a EAAT2 activator.

Compounds

UCT943

T13246

Synonym:

Target: Parasite, PI4K

CU-CPT9b

T7302

Synonym: CU-CPT-9b,TLR8-specific antagonist 1

Target: TLR

LIT927

T5207

Synonym: LIT 927,LIT-927

Target: Phosphatase, P450, Histone Methyltransferase

AT9283

T3068

Synonym: J-504568

Target: Apoptosis, FLT, JAK, Bcr-Abl, Aurora Kinase, Autophagy

KPT9274

T4354

Synonym: KPT-9274,KPT 9274,PAK4-IN-1

Target: NAMPT, PAK

NDT9520492

T33616

Synonym: NDT 9520492,NDT-9520492

Target:

(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)

Cat No.	Product Name	Synonyms	Targets
T81052	T988C	(+)-T988C
	T988C, a heptacyclic epidithiodioxopiperazine (ETP) natural product, exhibits potent cytotoxicity against cultured P388 leukemia cells [1].

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-05096	Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc)	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-01873	Transferrin Receptor/TFRC Protein, Human, Recombinant (His)	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-01897	PRSS3 Protein, Human, Recombinant (His)	Human	HEK293
	Trypsin-3, also known as Trypsin III, brain trypsinogen, Serine protease 3 and PRSS3, is a secreted protein that belongs to the peptidase S1 family. Trypsin-3 / PRSS3 is expressed is in pancreas and brain. It contains on...
TMPY-05617	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPK-00376	Transferrin R/CD71 Protein, Human, Recombinant (hFc)	Human	HEK293
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-00374	Transferrin R/CD71 Protein, Human, Recombinant (His & Avi)	Human	HEK293
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-01261	Transferrin R/CD71 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-00375	Transferrin R/CD71 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPJ-00378	Transferrin Receptor/TFRC Protein, Human, Recombinant (aa 101-760, His)	Human	Human Cells
	Transferrin receptor protein 1 (TFRC) belongs to the peptidase M28 family that is synthesized as a 172 amino acid (aa). TFRC regulated by cellular iron levels through binding of the iron regulatory proteins, IRP1 and IRP...
TMPY-06251	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06271	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His)	SARS-CoV-2	Baculovirus-Insect Cells
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06444	SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06395	SARS-CoV-2 Spike S1 Protein (L5F & T95I & D253G & S477N & E484K & D614G, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-02845	CST9L Protein, Human, Recombinant (hFc)	Human	HEK293
	Testatin is a member of the Cystatin family. Cystatins comprise genes that all show expression patterns that are strikingly restricted to reproductive tissue. Cystatins are a family of cysteine protease inhibitors with h...
TMPY-06287	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His & Avi), Biotinylated	SARS-CoV-2	Baculovirus-Insect Cells
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06293	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His & Avi), Biotinylated	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06393	SARS-CoV-2 Spike S1+S2 Protein (L5F & T95I & D253G & S477N & E484K & D614G & A701V, His)	SARS-CoV-2	Baculovirus-Insect Cells
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06443	SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06421	SARS-CoV-2 Spike S1 Protein (T95I & Y144S & Y145N & R346K & E484K & N501Y & D614G & P681H, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPY-06647	CHST9 Protein, Human, Recombinant (His)	Human	HEK293
	CHST9 Protein, Human, Recombinant (His) is expressed in HEK293 with His tag. The predicted molecular weight is 17.66 kDa. Accession number: NP_113610.2
TMPY-06422	SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His)	SARS-CoV-2	HEK293
	The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...