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Search Results for " 5-ht2 "

20

Compounds

Cat No. Product Name Synonyms Targets
T12597 5-HT2 antagonist 1 5-HT Receptor
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
T36949 Niaprazine 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...
T15270 Fananserin RP 62203 Dopamine Receptor , 5-HT Receptor
Fananserin is an effective, selective and oral active antagonist of 5-HT2 (Ki = 0.37 nM for the rat 5-HT2A). Fananserin is an antagonist of human D4 receptor (Ki = 2.93 nM).
T0137 Mirtazapine 6-Azamianserin,Org3770 Dopamine Receptor , 5-HT Receptor , Opioid Receptor , Adrenergic Receptor , Histamine Receptor
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevations in serum aminotransferase levels and h...
T79804 5-HT2 agonist-1 5-HT Receptor
Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively. The free base form of this compound is utilized in research pertaini...
T14968 Cinanserin hydrochloride SQ 10643 Influenza Virus , 5-HT Receptor
Cinanserin hydrochloride (SQ 10643) is a high affinity antagonist of the 5-HT2 receptor (Ki: 41 nM) and a 3C-like protease inhibitor of severe acute respiratory syndrome coronavirus.
T1045 Trimipramine maleate Surmontil maleate Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal...
T4369 SCH-23390 hydrochloride R-(+)-SCH23390 hydrochloride Potassium Channel , Dopamine Receptor , 5-HT Receptor
SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).
T79805 5-HT2 agonist-1 free base 5-HT Receptor
Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C receptors, exhibiting IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively. It is utilized in research pertaining to depression...
T1567 Olanzapine LY170053 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR
Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T22904 L-745870 trihydrochloride L-745,870 trihydrochloride Dopamine Receptor , Sigma receptor , 5-HT Receptor , Adrenergic Receptor
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
T12865 SCH-23390 maleate R-(+)-SCH-23390 maleate Potassium Channel , Dopamine Receptor , 5-HT Receptor
SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM, respectively).
T5389 Volinanserin M 100907,MDL100907 5-HT Receptor
Volinanserin (MDL100907) (MDL 100907) is a potent and selective antagonist of the serotonin receptor 5-HT2 (Ki: 0.36 nM) and shows 300-fold selectivity for 5-HT2 receptor over 5-HT1c, alpha-1 adrenergic and sigma recepto...
T22029 AL 34662 5-HT Receptor , Adrenergic Receptor
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a low affinity α-1D adrenergic agonist, with an EC50 of 0.4 μM....
T23382 Spiroxatrine R 5188 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2, and dopamine receptors.Spiroxatrine may be used in the stu...
T16759 Ritanserin R 55667 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
T8702 SKF-83566 Dopamine Receptor , 5-HT Receptor , AChR
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 nM
T21855 AMI-193 Espiramida,Spiramide Dopamine Receptor , 5-HT Receptor
AMI-193 (Spiramide) is an effective and selective antagonist of 5-HT2 and D2 receptor with Kis of 2, 3, 50, 2530, and 4300 nM for 5-HT2, D2 Receptor, 5-HT1A, D1 Receptor, and 5-HT1C Receptor. AMI-193 shows antipsychotic ...
T22959 M-Chlorophenylbiguanide hydrochloride 1-(3-Chlorophenyl)biguanidehydrochloride 5-HT Receptor
5-HT3 receptor agonist
T2599 Pirenperone 5-HT Receptor
Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.

Compounds

5-HT2 antagonist 1
T12597
Synonym:
Target: 5-HT Receptor
Niaprazine
T36949
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Fananserin
T15270
Synonym: RP 62203
Target: Dopamine Receptor, 5-HT Receptor
Mirtazapine
T0137
Synonym: 6-Azamianserin,Org3770
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
5-HT2 agonist-1
T79804
Synonym:
Target: 5-HT Receptor
Cinanserin hydrochloride
T14968
Synonym: SQ 10643
Target: Influenza Virus, 5-HT Receptor
Trimipramine maleate
T1045
Synonym: Surmontil maleate
Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor
SCH-23390 hydrochloride
T4369
Synonym: R-(+)-SCH23390 hydrochloride
Target: Potassium Channel, Dopamine Receptor, 5-HT Receptor
5-HT2 agonist-1 free base
T79805
Synonym:
Target: 5-HT Receptor
Olanzapine
T1567
Synonym: LY170053
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR
L-745870 trihydrochloride
T22904
Synonym: L-745,870 trihydrochloride
Target: Dopamine Receptor, Sigma receptor, 5-HT Receptor, Adrenergic Receptor
SCH-23390 maleate
T12865
Synonym: R-(+)-SCH-23390 maleate
Target: Potassium Channel, Dopamine Receptor, 5-HT Receptor
Volinanserin
T5389
Synonym: M 100907,MDL100907
Target: 5-HT Receptor
AL 34662
T22029
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor
Spiroxatrine
T23382
Synonym: R 5188
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Ritanserin
T16759
Synonym: R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
SKF-83566
T8702
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, AChR
AMI-193
T21855
Synonym: Espiramida,Spiramide
Target: Dopamine Receptor, 5-HT Receptor
m-Chlorophenylbiguanide hydrochloride
T22959
Synonym: 1-(3-Chlorophenyl)biguanidehydrochloride
Target: 5-HT Receptor
Pirenperone
T2599
Synonym:
Target: 5-HT Receptor
1 2 3 4 5
TargetMol