Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CXD101 is a novel class I-selective HDACi (HDAC1 (IC50 : 63nM), HDAC2 (IC50 :570nM), HDAC3 (IC50 :550nM)). CXD101(CXD-101) has no activity against HDAC class II
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 54.00 | |
5 mg | In stock | $ 126.00 | |
10 mg | In stock | $ 198.00 | |
25 mg | In stock | $ 405.00 | |
50 mg | In stock | $ 597.00 | |
100 mg | In stock | $ 852.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 126.00 |
Description | CXD101 is a novel class I-selective HDACi (HDAC1 (IC50 : 63nM), HDAC2 (IC50 :570nM), HDAC3 (IC50 :550nM)). CXD101(CXD-101) has no activity against HDAC class II |
Targets&IC50 | HDAC1:63 nM , HDAC3:550 nM , HDAC2:570 nM |
Synonyms | CXD-101 |
Molecular Weight | 403.52 |
Formula | C24H29N5O |
CAS No. | 934828-12-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 31 mg/mL (76.82 mM)
You can also refer to dose conversion for different animals. More
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CXD101 934828-12-3 Chromatin/Epigenetic DNA Damage/DNA Repair HDAC antitumor HDAC2 orally Histone deacetylases histone CXD 101 inhibit CXD-101 HDAC1 HDAC3 acetylation Inhibitor inhibitor