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Search Results for " third-generation "

20

Compounds

Cat No. Product Name Synonyms Targets
T9865 Almonertinib mesylate EGFR
Almonertinib mesylate is an irreversible inhibitor of EGFR tyrosine kinase with high selectivity for EGFR-sensitizing and T790M resistance mutations. Almonertinib mesylate can be used in the non-small cell lung cancer st...
T60076 Oritinib SH-1028 EGFR
Oritinib (SH-1028) is an inhibitor of EGFR with IC50s of 18, 0.7, 4, 0.1, 1.4 and 0.89 nM for EGFR (wt), EGFR (L858R), EGFR (L861Q), EGFR (L858R/T790M), EGFR (d746-750), EGFR (d746-750/T790M), respectively. Oritinib can ...
T1223 Ceftriaxone sodium hydrate Ceftriaxone Sodium Trihydrate,Ceftriaxone disodium hemiheptahydrate,Ceftriaxone sodium Others , Antibacterial , Antibiotic
Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.
T3061 Lorlatinib PF-6463922,PF-06463922,Loratinib Apoptosis , Tyrosine Kinases , ROS , ALK , ROS Kinase
Lorlatinib (PF-6463922) is an orally available, ATP-competitive inhibitor of the receptor tyrosine kinases, anaplastic lymphoma kinase (ALK) and C-ros oncogene 1 (Ros1), with potential antineoplastic activity.
T30787 Cefetamet sodium Ro 15-8074/001,Ro15-8074/001,Ro-15-8074/001
Cefetamet sodium is a third-generation cephalosporin.
T1599 Ibandronic acid Bonviva,Bondronat,Boniva Others , HBV
Ibandronic acid (Bonviva) is a third-generation amino-bisphosphonate with anti-resorptive and anti-hypercalcemic activities.
T0138 Cefpiramide acid Cefpiramidum,Cefpiramido Antibacterial
Cefpiramide acid (Cefpiramidum) is a third-generation cephalosporin antibiotic.
T0198 Ceftiofur sodium Naxcel,Sodium ceftiofur Antibacterial , Antibiotic
Ceftiofur sodium (Naxcel), an antibiotic of the cephalosporin type (third generation), is used as veterinary medicine.
T7120 Cefetamet pivoxil hydrochloride Ro 15-8075 Antibacterial , Antibiotic
Cefetamet pivoxil hydrochloride (Ro 15-8075) is a third generation cephalosporin antibiotic with oral activity.
T7839 Lasofoxifene Tartrate CP-336156 Estrogen Receptor/ERR
Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.
T0127 Glimepiride Glimperide,HOE-490 Potassium Channel
Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.
T0911 Cefotaxime sodium Cefotaxim sodium salt,Cefotaxime sodium salt,Cefotaxim (sodium salt),HR-756 (sodium salt) Antibacterial , Antibiotic
Cefotaxime is a third-generation cephalosporin antibiotic. Like other third-generation cephalosporins, it has broad spectrum activity against Gram positive and Gram negative bacteria. In most cases, it is considered to b...
T9073 SRS16-86 Ferroptosis
SRS16-86 is a novel third-generation ferrostatin, is an inhibitor of ferroptosis.
T1405 Cefditoren pivoxil ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl Antibacterial , Antibiotic
Cefditoren pivoxil (ME 1207) is a semi-synthetic, broad-spectrum, beta-lactamase resistant, third-generation cephalosporin antibiotic with bactericidal activity.
T8126 Cefodizime Sodium Others , Antibacterial , Antibiotic
Cefodizime Sodium is a third generation cephalosporin antibiotic, has broad-spectrum activity
T5024 Cefotiam Hexetil Hydrochloride Antibacterial , Antibiotic
Cefotiam Hexetil Hydrochloride is a third-generation, semi-synthetic, beta-lactam cephalosporin antibiotic with antibacterial activity.
T6268 Ceftiofur hydrochloride Ceftiofur HCl,U-67279A,Excenel hydrochloride Antibacterial , Antibiotic
Ceftiofur hydrochloride (U-67279A) is the hydrochloride salt form of ceftiofur, a semisynthetic, beta-lactamase-stable, broad-spectrum, third-generation cephalosporin with antibacterial activity.
T4405 Ceftibuten dihydrate Sch-39720 dihydrate Antibacterial , Antibiotic
Ceftibuten dihydrate (Sch-39720 dihydrate) is the dihydrate form of ceftibuten, and is a third-generation cephalosporin with antibacterial activity.
T2490 Osimertinib AZD-9291,Mereletinib EGFR
Osimertinib (AZD-9291) is an EGFR third-generation inhibitor that inhibits the T790M resistance mutation produced by second-generation EGFR inhibitors with irreversible and oral activity. Osimertinib has antitumor activi...
T4990 Cefcapene pivoxil hydrochloride hydrate Cefcapene Pivoxil Hydrochloride Antibacterial , Antibiotic
Cefcapene pivoxil hydrochloride hydrate is the pivalate ester prodrug form of cefcapene, a semi-synthetic third-generation cephalosporin with antibacterial activity. After oral administration of cefcapene pivoxil, the es...

Compounds

Almonertinib mesylate
T9865
Synonym:
Target: EGFR
Oritinib
T60076
Synonym: SH-1028
Target: EGFR
Ceftriaxone sodium hydrate
T1223
Synonym: Ceftriaxone Sodium Trihydrate,Ceftriaxone disodium hemiheptahydrate,Ceftriaxone sodium
Target: Others, Antibacterial, Antibiotic
Lorlatinib
T3061
Synonym: PF-6463922,PF-06463922,Loratinib
Target: Apoptosis, Tyrosine Kinases, ROS, ALK, ROS Kinase
Cefetamet sodium
T30787
Synonym: Ro 15-8074/001,Ro15-8074/001,Ro-15-8074/001
Target:
Ibandronic acid
T1599
Synonym: Bonviva,Bondronat,Boniva
Target: Others, HBV
Cefpiramide acid
T0138
Synonym: Cefpiramidum,Cefpiramido
Target: Antibacterial
Ceftiofur sodium
T0198
Synonym: Naxcel,Sodium ceftiofur
Target: Antibacterial, Antibiotic
Cefetamet pivoxil hydrochloride
T7120
Synonym: Ro 15-8075
Target: Antibacterial, Antibiotic
Lasofoxifene Tartrate
T7839
Synonym: CP-336156
Target: Estrogen Receptor/ERR
Glimepiride
T0127
Synonym: Glimperide,HOE-490
Target: Potassium Channel
Cefotaxime sodium
T0911
Synonym: Cefotaxim sodium salt,Cefotaxime sodium salt,Cefotaxim (sodium salt),HR-756 (sodium salt)
Target: Antibacterial, Antibiotic
SRS16-86
T9073
Synonym:
Target: Ferroptosis
Cefditoren pivoxil
T1405
Synonym: ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl
Target: Antibacterial, Antibiotic
Cefodizime Sodium
T8126
Synonym:
Target: Others, Antibacterial, Antibiotic
Cefotiam Hexetil Hydrochloride
T5024
Synonym:
Target: Antibacterial, Antibiotic
Ceftiofur hydrochloride
T6268
Synonym: Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
Ceftibuten dihydrate
T4405
Synonym: Sch-39720 dihydrate
Target: Antibacterial, Antibiotic
Osimertinib
T2490
Synonym: AZD-9291,Mereletinib
Target: EGFR
Cefcapene pivoxil hydrochloride hydrate
T4990
Synonym: Cefcapene Pivoxil Hydrochloride
Target: Antibacterial, Antibiotic
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TargetMol