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Glimepiride

Catalog No. T0127 CAS 93479-97-1

Synonyms: HOE-490, Glimperide

Glimepiride is a long-acting, third-generation sulfonylurea with hypoglycemic activity.

Glimepiride, CAS 93479-97-1

Pack Size	Availability	Price/USD
25 mg	In stock	16.00
50 mg	In stock	22.00
100 mg	In stock	30.00
200 mg	In stock	40.00
500 mg	In stock	60.00
1 g	In stock	100.00
1 mL * 10 mM (in DMSO)	In stock	50.00

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Purity 97.84%

HNMR HPLC COA Datasheet MSDS

Purity 99.47%

HNMR HPLC COA Datasheet MSDS

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Glimepiride is a long-acting, third-generation sulfonylurea with hypoglycemic activity.
Targets&IC50	SUR1 :ic50 3nM, SUR2A :ic50 5.4nM, SUR2B :ic50 7.3nM,

Synonyms	HOE-490 , Glimperide
Purity	97.84%
Molecular Weight	490.62
Formula	C24H34N4O5S
CAS No.	93479-97-1

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

DMSO: 12.3 mg/mL (25 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Song DK, et al. Br J Pharmacol, 2001, 133(1), 193-199. 2. Müller G, et al. Horm Metab Res, 1996, 28(9), 469-487 3. Lawrence CL, et al. Br J Pharmacol, 2002, 136(5), 746-752. 4. Rabbani SI, et al. Indian J Exp Biol, 2009, 47(10), 804-810.

Related compound libraries

This product is contained In the following compound libraries：

Approved Drug Library Bioactive Compound Library Inhibitor Library Anti-cancer Compound Library Anti-diabetic Compound Library Ion Channel Inhibitor Library Protease Inhibitor Library FDA-approved Drug Library Anti-Metabolism Disease Compound Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Answers to questions you may have can be found in the Inhibitor Handling Instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.