progestin — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T39785L	TH5427		NUDIX hydrolase
	TH5427 is a lead NUDT5 inhibitor(MG assay IC50 = 29 nM).		NUDIX hydrolase
T7537	Norgestimate		Progesterone Receptor
	Norgestimate is an acetylated progestinused in combination with ethinyl estradiol as an oral contraceptive.		Progesterone Receptor
T2567	Etonogestrel	3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
	Etonogestrel (Implanon) is a steroidal progestin used as hormonal contraceptives.
T1263	Levonorgestrel	D-Norgestrel	Others , Estrogen/progestogen Receptor , Progesterone Receptor
	Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device. The physiologic effect of levonorgestrel is by means of Inhibit Ovum Fertilization.
T8094	16-Dehydroprogesterone	16-Dehydroprogesterone	Endogenous Metabolite
	16-Dehydroprogesterone is a endogenous Metabolite. 16-Dehydroprogesterone is a steroidal progestin.		Endogenous Metabolite
T1541	Drospirenone	ZK 3059,Dihydrospirorenone	Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , COX
	Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T8395	Nomegestrol acetate		Others , Progesterone Receptor
	Nomegestrol acetate is a widely used progestin-like drug,which is characterized as a full agonist at the progesterone receptor		Others , Progesterone Receptor
T5174	Nestoron	ST-1435,Segesterone Acetate,Nestorone,Elcometrine	Estrogen/progestogen Receptor , Progesterone Receptor
	Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).		Estrogen/progestogen Receptor , Progesterone Receptor
T1102	Mifepristone	C-1073,RU486,RU 38486	Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , NO Synthase , Autophagy
	Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
T16338	Norgestimate metabolite Norelgestromin	17-Deacetyl norgestimate,17-Deacylnorgestimate	Drug Metabolite
	Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen ethinyl es...		Drug Metabolite
T1261	Medroxyprogesterone Acetate	Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate)	Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite
	Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been...
T1429	17α-Hydroxyprogesterone	Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone	Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
	17α-Hydroxyprogesterone (17-OHP) is a physiological progestin that is produced during glucocorticoid and steroid hormone synthesis and is increased during the third trimester of pregnancy. Hydroxyprogesterone binds to th...
T2597	Norgestrel	SH-850,FH 122-A,WY-3707,SH-70850	Estrogen/progestogen Receptor , Reactive Oxygen Species
	Norgestrel (WY-3707) is a synthetic progestin commonly used alone or in combination with an estrogen for contraception. Norgestrel suppresses the secretion of luteinizing and follicle-stimulating hormones (LH and FSH), t...		Estrogen/progestogen Receptor , Reactive Oxygen Species
T7931	16a,17a-Epoxy-4-Pregnen-3,20-Dione		Others
	16a,17a-Epoxy-4-Pregnen-3,20-Dione is a synthetic progestin, a metabolite of the luteinizing hormone hormone, which acts by binding to the luteinizing hormone receptor. It has been used to study the effects of progestero...		Others
T33819	Org 2058	O-2058,Org-2058,Org2058
	Org 2058 is a synthetic progestin.
T30942	Cingestol
	Cingestol is a steroidal progestin of the 19-nortestosterone group that was never marketed.
T29248	(+)-Norgestrel	Dextronorgestrel,L-Norgestrel
	(+)-Norgestrel is a progestin medication for the treatment of birth control pills and in menopausal hormone therapy.
T34141	Promegestone	R5020,R-5020,RU 5020,R 5020,RU-5020
	Promegestone is a progestin medication used in menopausal hormone therapy and in the treatment of gynecological disorders.
T19811	Nomegestrol
	Nomegestrol is a progestin. It is used in the treatment of gynecological disorders, in menopausal hormone therapy for the treatment of menopausal symptoms, and in hormonal contraceptives.
T25304	Demegestone	R-2453,Lutionex,R 2453,RU 2453,R2453
	Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat lutea...