Home Tools
Log in
Cart

Search Result

Search Results for " napa "

Targets

21

Compounds

4

Natural Products

4

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T3575 Acecainide hydrochloride ASL 601,NAPA Others
Acecainide hydrochloride (NAPA) is a major metabolite of PROCAINAMIDE. Its anti-arrhythmic action may cause cardiac toxicity in kidney failure.
T0249 N-Acetylprocainamide NAPA,Acecainide Potassium Channel , Sodium Channel , Drug Metabolite
N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmic drug.
T6763 Xevinapant ARRY-334543,SM-406,AT406,Debio-1143 IAP
Xevinapant (Debio-1143) is a potent Smac mimetic and an antagonist of IAP (inhibitor of apoptosis protein via E3 ubiquitin ligase), binding to XIAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3 with Ki of 66.4 nM, 1.9 nM, and 5.1 nM, ...
T7587 Tenapanor RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722 Sodium Channel
Tenapanor (RDX 5791) is an inhibitor of the sodium-proton (Na(+)/H(+)) exchanger NHE3, which plays a prominent role in sodium handling in the gastrointestinal tract and kidney. Tenapanor possesses an excellent preclinica...
T0113 Mebhydrolin napadisylate Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline 5-HT Receptor , AChR , Histamine Receptor
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.
T3218 Napabucasin BBI608 STAT
Napabucasin (BBI608) is an orally available Stat3 and Y cell stemness inhibitor.
T16802 Lonapalene RS4317 Others
Lonapalene is a topically effective inhibitor of 5-lipoxygenase.
T9593 Senaparib IMP4297 PARP
Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.
T6007 Birinapant TL32711 Apoptosis , IAP , HIV Protease
Birinapant (TL32711) is a synthetic small molecule that is both a peptidomimetic of second mitochondrial-derived activator of caspases (SMAC) and inhibitor of IAP (Inhibitor of Apoptosis Protein) family proteins, with po...
T60097 Methyl (E)-sinapate Others
Methyl (E)-sinapate is isolated from the Polygala sibirica L.var. megalopha Fr.
T40572 Lesogaberan napadisylate AZD-3355 napadisylate
Lesogaberan (AZD-3355) napadisylate is a potent and selective agonist of GABA B receptors, with an EC 50 of 8.6 nM for human recombinant GABA B receptors. It demonstrates an affinity (Ki) of 5.1 nM for rat GABA B recepto...
T35940 Darinaparsin Dimethylarsinic glutathione,Darinaparsin
Darinaparsin is a dimethylated arsenic linked to glutathione. It is cytotoxic to DU145, LNCaP, and PC3 prostate cancer cells (IC50s = 5-10 &#181M) and patient-derived primary prostate cancer cells (IC50s = 2.5-20 &#181M)...
T26553 Aclatonium Napadisilate Acaltonium napadisilate
Aclatonium Napadisilate, a cholinergic agonist, has been shown to stimulates endocrine and exocrine pancreatic secretion.
T24995 Abediterol napadisylate LAS100977 napadisylate
Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.
T13405L Fanapanel MPQX,ZK200775 Others
Fanapanel is a highly selective AMPA/kainate antagonist with little activity against NMDA. It also has Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.
T70762 Senaparib hydrochloride
Senaparib hydrochloride is a potent and selective oral PARP1/2 inhibitor with strong antitumor activity.
T13405 Fanapanel hydrate MPQX hydrate,ZK200775 (hydrate) Others
Fanapanel hydrate is a highly selective antagonist of AMPA/kainate with little activity against NMDA(Ki of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively).
T3299 Xevinapant hydrochloride AT-406 HCl,SM-406 Apoptosis , IAP
Xevinapant hydrochloride (AT-406 HCl) , an orally active antagonist of multiple inhibitor of apoptosis proteins(IAP), inhibits progression of human ovarian Y binding to XIAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3 with Ki of 66....
T28131 Napamezole WIN51181,WIN-51181,WIN 51181
Napamezole is an α2 adrenergic receptor antagonist. Napamezole antagonizes methoxamine-induced contractions (alpha-1) of the rat vas deferens with a Kb of 135 nM. Napamezole reverses clonidine-induced decreased in twitch...
T7587L Tenapanor HCl RDX-5791,AZD 1722,AZD-1722,AZD1722,RDX5791,RDX 5791
Tenapanor( AZD-1722, RDX 5791) is an inhibitor of the sodium-proton (Na(+)/H(+)) exchanger NHE3, which is used for sodium handling in the gastrointestinal tract and kidney.
T32827 L-Napamp
L-Napamp is a bioactive chemical.

Compounds

Acecainide hydrochloride
T3575
Synonym: ASL 601,NAPA
Target: Others
N-Acetylprocainamide
T0249
Synonym: NAPA,Acecainide
Target: Potassium Channel, Sodium Channel, Drug Metabolite
Xevinapant
T6763
Synonym: ARRY-334543,SM-406,AT406,Debio-1143
Target: IAP
Tenapanor
T7587
Synonym: RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722
Target: Sodium Channel
Mebhydrolin napadisylate
T0113
Synonym: Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline
Target: 5-HT Receptor, AChR, Histamine Receptor
Napabucasin
T3218
Synonym: BBI608
Target: STAT
Lonapalene
T16802
Synonym: RS4317
Target: Others
Senaparib
T9593
Synonym: IMP4297
Target: PARP
Birinapant
T6007
Synonym: TL32711
Target: Apoptosis, IAP, HIV Protease
Methyl (E)-sinapate
T60097
Synonym:
Target: Others
Lesogaberan napadisylate
T40572
Synonym: AZD-3355 napadisylate
Target:
Darinaparsin
T35940
Synonym: Dimethylarsinic glutathione,Darinaparsin
Target:
Aclatonium Napadisilate
T26553
Synonym: Acaltonium napadisilate
Target:
Abediterol napadisylate
T24995
Synonym: LAS100977 napadisylate
Target:
Fanapanel
T13405L
Synonym: MPQX,ZK200775
Target: Others
Senaparib hydrochloride
T70762
Synonym:
Target:
Fanapanel hydrate
T13405
Synonym: MPQX hydrate,ZK200775 (hydrate)
Target: Others
Xevinapant hydrochloride
T3299
Synonym: AT-406 HCl,SM-406
Target: Apoptosis, IAP
Napamezole
T28131
Synonym: WIN51181,WIN-51181,WIN 51181
Target:
Tenapanor HCl
T7587L
Synonym: RDX-5791,AZD 1722,AZD-1722,AZD1722,RDX5791,RDX 5791
Target:
L-Napamp
T32827
Synonym:
Target:
Cat No. Product Name Synonyms Targets
TN2281 Sinapaldehyde trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde Antibacterial
Sinapaldehyde (trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde) is a natural product. Sinapaldehyde exhibits moderate antibacterial against Methicillin resistant S. aureus (MRSA) and E. coli with MIC values of 128 and 128 μ...
TN1929 Methyl sinapate Others
Methyl sinapate can increase the frequency of cells with chromosome aberrations in the CHO K-1 cells treated with MMC, 4NQO or UV.
TN5027 Sinapaldehyde glucoside Others
Sinapaldehyde glucoside is a natural product of Phellodendron, Rutaceae. The catalog number is TN5027 and the CAS number is 154461-65-1. Sinapaldehyde glucoside can be used as a reference standard.
TN6365 3-Deoxy-11,13-dihydroisosecotanapartholide
3-Deoxy-11,13-dihydroisosecotanapartholide is a natural product for research related to life sciences. The catalog number is TN6365 and the CAS number is 572924-43-7.

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPH-02997 Dps Protein, Mycobacterium smegmatis, Recombinant (His & SUMO) Mycobacterium smegmatis E. coli
Protects DNA from oxidative damage by sequestering intracellular Fe(2+) ion and storing it in the form of Fe(3+) oxyhydroxide mineral. One hydrogen peroxide oxidizes two Fe(2+) ions, which prevents hydroxyl radical produ...
TMPH-00794 Dps Protein, Helicobacter pylori, Recombinant (His & SUMO) Helicobacter pylori E. coli
Protects DNA from oxidative damage by sequestering intracellular Fe(2+) ion and storing it in the form of Fe(3+) oxyhydroxide mineral. One hydrogen peroxide oxidizes two Fe(2+) ions, which prevents hydroxyl radical produ...
TMPY-00151 Alpha SNAP Protein, Human, Recombinant (His) Human E. coli
NAPA (NSF Attachment Protein Alpha) is a Protein Coding gene. This gene encodes a member of the soluble NSF attachment protein (SNAP) family. SNAP proteins play a critical role in the docking and fusion of vesicles to ta...
TMPH-02697 GNA12 Protein, Mouse, Recombinant (His & Myc) Mouse E. coli
Guanine nucleotide-binding proteins (G proteins) are involved as modulators or transducers in various transmembrane signaling systems. Activates effector molecule RhoA by binding and activating RhoGEFs (ARHGEF12/LARG). G...
TargetMol