bicyclic — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T9609	GRK5-IN-2		GRK
	GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. It regulates the expression and/or release of insulin and is useful for the metabolic disease research.		GRK
T8242	Sabinene		Others
	Sabinene is a natural product that has antifungal and anti-inflammatory properties		Others
T5734	(+)-BORNEOL	d-Borneol	GABA Receptor
	(+)-BORNEOL (d-Borneol) is a natural bicyclic monoterpene used for analgesia and anesthesia in traditional Chinese medicine; enhances GABA receptor activity with an EC50 of 248 μM.		GABA Receptor
TN1114	Carabrone		Antibacterial , Antifection
	Carabrone, a botanical bicyclic sesquiterpenic lactone, is a promising fungicidal agent that can effectively control G. tritici.		Antibacterial , Antifection
T2952	Camphor	(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa	Influenza Virus , TRP/TRPV Channel
	Camphor (2-Camphanone) is a bicyclic monoterpene ketone found widely in plants, especially CINNAMOMUM CAMPHORA. It is used topically as a skin antipruritic and as an anti-infective agent.		Influenza Virus , TRP/TRPV Channel
T8279	Isobornyl acetate		Others
	Isobornyl acetate is a natural product derived from the essential oil of the lemongrass plant and is a bicyclic monoterpene. It is used in a variety of applications, including as a flavoring agent, a fragrance ingredient...		Others
TN1641	(-)-Fenchone		Others , Antioxidant , Antifungal
	(-)-Fenchone is a bicyclic monoterpenoid widely distributed in plants and can be extracted from Foeniculum vulgare and Peumus boldus. (-)-Fenchone has a wide range of biological activities including antioxidant, wound he...		Others , Antioxidant , Antifungal
T9043	AS1810722		P450 , STAT
	AS1810722, a fused bicyclic pyrimidine derivative, is an orally active and potent inhibitor of STAT6, demonstrating an IC50 of 1.9 nM. It exhibits effective inhibition of CYP3A4, positioning it as a promising candidate f...		P450 , STAT
T10109	3-Carene	Delta-3-Carene	COX , Antifungal
	3-Carene（Delta-3-Carene） is a bicyclic monoterpene extracted from western larch and Douglas-fir that acts as a phytofungicide.3-Carene inhibits inflammatory infiltrates and COX-2 overexpression induced by nociceptive sti...		COX , Antifungal
T4799	Indole		Others , Endogenous Metabolite
	Indole has a bicyclic structure, consisting of a six-membered benzene ring fused to a five-membered nitrogen-containing pyrrole ring. It can be produced by bacteria as a degradation product of the amino acid tryptophan. ...		Others , Endogenous Metabolite
T1483	Citalopram hydrobromide	Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,Citalopram HBr	5-HT Receptor , Serotonin Transporter , Autophagy
	Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby potentiating serotonergic activity in the central nervous system...		5-HT Receptor , Serotonin Transporter , Autophagy
T27886	LY 186826	LY-186826,LY186826
	LY 186826 is an antibacterial agent with bicyclic pyrazolidinone properties.
T26028	RA VII	Methylether of TPC-A,RAVII,RA-VII
	RA VII is used as an antitumor bicyclic hexapeptide of plant origin.
T27882	LY 173013	LY-173013,LY173013
	LY 173013 is a bicyclic pyrazolidinone, it has antibacterial properties.
T40715	3-Butenoic acid	Vinylacetic acid
	3-Butenoic acid, also known as Vinylacetic acid, is utilized in the synthesis of 3,6-dihydro-1,2-oxazine that possesses a bicyclic structure. This strained bicyclic compound, when combined with an external alkene, acts a...
T26175	Salinamide A
	Salinamide A is an effective anti-inflammatory bicyclic depsipeptide.
T35653	2’-O,4’-C-Methyleneuridine
	2'-O,4'-C-Methyleneuridine (Compound 15a) is a bicyclic nucleoside. [1]. Sharma VK, et al. Chemoenzymatic convergent synthesis of 2'-O,4'-C-methyleneribonucleosides. J Org Chem. 2014 Jul 3;79(13):6336-41.
T19086	1-(2'-O-4-C-Methylene-beta-D-ribofuranosyl)thymine		Others
	1-(2'-O-4-C-Methylene-beta-D-ribofuranosyl)thymine is a bicyclic nucleoside.		Others
T31575	Drimane
	Drimane is a bicyclic sesquiterpene. It is the parent structure of many natural products with various biological activity.
T74647	BT5528
	BT5528, a bicyclic peptide toxin conjugate and an EphA2 activator derived from BCY6099, consists of a bicyclic peptide and Auristatin E. This compound demonstrates significant anti-tumor efficacy without inducing bleedin...