20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6713 | Ulipristal | Estrogen/progestogen Receptor , Progesterone Receptor | |
Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure. | |||
T1560 | Prednisolone | Predonine,Hydroretrocortine,Metacortandralone | Glucocorticoid Receptor , Endogenous Metabolite |
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. | |||
T2527 | Ulipristal acetate | Ulipristal,CDB-2914 | Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy |
Ulipristal acetate (CDB-2914) is an orally bioavailable, acetate salt of ulipristal, a selective progesterone receptor modulator with anti-progesterone activity. Ulipristal binds to the progesterone receptor (PR), thereb... | |||
T21404 | Fluticasone furoate | Veramyst,Allermist,Avamys,Fluticasone furoate | Glucocorticoid Receptor |
Fluticasone furoate (Avamys) is a synthetic trifluorinated corticosteroid derived from fluticasone with a Kd of 0.3 nM. Fluticasone furoate has potent anti-inflammatory, anti-asthmatic activity, and low systemic exposure... | |||
T0094 | Budesonide | Entocort,Pulmicort,Rhinocort | Glucocorticoid Receptor |
Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. According to reports, Budesonide has extensively inhibitory effects agai... | |||
T2884 | Cortisone | Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone | Glucocorticoid Receptor , Endogenous Metabolite |
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity. | |||
T1531 | Mometasone furoate | Sch32088 | Glucocorticoid Receptor |
Mometasone furoate (Sch32088) is a pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA and ALLERGIC RHINITIS. It is also used as a topical treatment for ski... | |||
T0034 | Cortisone acetate | Cortisone 21-acetate,NSC 49420 | Glucocorticoid Receptor , Endogenous Metabolite |
Cortisone Acetate is a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal glands with anti-inflammatory and immunomodulating properties. Cortisone acetate (NSC-49420) d... | |||
T6503 | Fluorometholone Acetate | NSC 47438,Flarex,Eflone,Oxylone acetate | Glucocorticoid Receptor , Carbonic Anhydrase |
Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye. | |||
T0188 | Fluticasone (propionate) | CCI-187881,Fluticasone propionate | Glucocorticoid Receptor , Virus Protease , Estrogen/progestogen Receptor , Phospholipase , Endogenous Metabolite |
Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist. | |||
T4602 | Hydrocortisone hemisuccinate | Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate | Glucocorticoid Receptor , Others , Interleukin |
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent. | |||
T15102 | Dexamethasone palmitate | DXP | Glucocorticoid Receptor |
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexamethasone palmitate is a glucocorticoid receptor agonist and an... | |||
T0208 | Prednisolone disodium phosphate | Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium | Glucocorticoid Receptor |
Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties. | |||
T22367 | Methylprednisolone succinate | Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate | Glucocorticoid Receptor |
Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent. | |||
T0977 | Medrysone | Gimeracil,6α-Methyl-11β-hydroxyprogesterone | Glucocorticoid Receptor , Others |
Medrysone (6α-Methyl-11β-hydroxyprogesterone) is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone exerts its effect by interacting with specific intracellular ... | |||
T9047 | Fluprednisolone | NSC-47439,NSC 47439,NSC47439 | Others |
Fluprednisolone (NSC-47439) is a synthetic glucocorticoid that has anti-inflammatory properties. | |||
T1168 | Desonide | Tridesilon,Locapred,Prednacinolone | Glucocorticoid Receptor |
Desonide (Prednacinolone) is a synthetic glucocorticosteroid for topical use, with anti-inflammatory activity. Desonide binds to glucocorticoid receptors in the cytoplasm, and the ligand-receptor complex is translocated ... | |||
T6502 | Fluocinonide | Lidex,Metosyn,Topsyn | Glucocorticoid Receptor |
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent. | |||
T0269 | Dichlorisone Acetate | Diloderm | Endogenous Metabolite , AChE |
Dichlorisone Acetate (Diloderm) is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity. | |||
T8396 | Prednisone acetate | Prednisone 21-acetate | Glucocorticoid Receptor |
Prednisone acetate (Prednisone 21-acetate) is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory. |