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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T24840 | STS-E412 | STS E412,STSE412 | Others |
STS-E412 is a tissue-protective and selective EPOR/CD131 receptor activator for the study of neurological disorders. | |||
T2577 | Dienogest | STS 557 | Apoptosis , Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy |
Dienogest (STS 557) is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic activities that is used in hormone therap... | |||
T6680 | Staurosporine | Antibiotic AM-2282,AM-2282,CGP 41251 | Apoptosis , PKA , Antibacterial , Antibiotic , Src , PKC , Antifungal |
Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-Fgr, phosphorylase kinase and TAOK2. Staurosporine also induces... | |||
T11416 | Glucagon receptor antagonists-5 | Others | |
Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM). | |||
T126527 | Poststerone | ||
Poststerone is a useful organic compound for research related to life sciences and the catalog number is T126527. | |||
TP2421 | Ysdspstst peptide | ||
Ysdspstst peptide is a biochemical. | |||
T11415 | Glucagon receptor antagonists-3 | Others | |
Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist. | |||
T11414 | Glucagon receptor antagonists-2 | Others | |
Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist. | |||
T25973 | Poststatin | ||
Poststatin is a prolyl endopeptidase inhibitor produced by Streptomyces viridochromogenes MH534-30F3. | |||
T11413 | Glucagon receptor antagonists-1 | Others | |
Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist. | |||
T15584 | Integrin Antagonists 27 | Others | |
Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist. It has a binding affinity of 18 nM and as a novel anticancer agent. | |||
T10665 | Calcium-Sensing Receptor Antagonists I | Others | |
Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium. | |||
T72470 | Estrone O-sulfamate | Estrone 3-O-sulfamate | Others |
Estrone O-sulfamate (Estrone 3-O-sulfamate) is a potent inhibitor of steroid sulfatase (STS). Estrone O-sulfamate is a placental microsomal inhibitor (P.M.) with IC50 values of 18 nM. Estrone O-sulfamate showed inhibitor... | |||
T36857 | Estrone sulfate sodium | Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate | Endogenous Metabolite |
Estrone sulfate sodium (17β-Estrone 3-sulfate) is an endogenous steroid and an estrogen ester that is biologically inactive. It is converted by steroid sulfatase into estrone . Estrone sulfate sodium has been investigate... | |||
T81089 | Steroid sulfatase-IN-7 | ||
Steroid sulfatase-IN-7 is an irreversible inhibitor of steroid sulfatase (STS), demonstrating potent activity with an IC50 of 0.05 nM against human placental STS, rendering it suitable for application in cancer research ... | |||
T81090 | Steroid sulfatase-IN-6 | ||
Steroid Sulfatase-IN-6 (Compound 10c) serves as an irreversible steroid sulfatase (STS) inhibitor, exhibiting a K i value of 0.4 nM against human placenta STS, and is applicable in tumor disease research [1]. | |||
T62236 | Steroid sulfatase/17β-HSD1-IN-3 | ||
Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1). Steroid sulfatase/17β-HSD1-IN-3 can be used to study endometriosis and ... | |||
T62237 | Steroid sulfatase-IN-4 | ||
Steroid sulfatase-IN-4 (Compound 16) is an irreversible inhibitor of steroid sulfatase (STS) that acts on human STS (IC50: 25 nM). steroid sulfatase-IN-4 can be used to study endometriosis. | |||
TN5091 | Tagitinin A | PPAR , Antifection | |
Tagitinin A is a plant insecticidal compound, it has phytotoxic activity, it shows significant inhibition of wheat coleoptile growth, seed germination, and the growth of STS and weeds. Tagitinin A is also a PPARα/γ dual ... | |||
T61979 | Steroid sulfatase/17β-HSD1-IN-4 | ||
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ). Steroid sulfatase/17β-HSD1-IN-4 irreversibly inhibits hSTS a... |