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Search Results for " nr3c3 "

20

Compounds

Cat No. Product Name Synonyms Targets
T3036 Dydrogesterone Progesterone Receptor
Dydrogesterone is a potent progestogen which can be used in progesterone deficiency studies.
T13703 Gestonorone Capronate Prostaglandin Receptor
Gestonorone Capronate  is a progesterone used to treat benign prostatic hyperplasia and endometrial cancer.
T1514 Norethindrone Norethisterone Estrogen/progestogen Receptor , Progesterone Receptor
Norethindrone (Norethisterone) is a synthetic progestational hormone with actions similar to those of PROGESTERONE but functioning as a more potent inhibitor of ovulation. It has weak estrogenic and androgenic properties...
T0478 Progesterone Pregn-4-ene-3,20-dione Estrogen/progestogen Receptor , Progesterone Receptor , Opioid Receptor , Endogenous Metabolite
Progesterone (Pregn-4-ene-3,20-dione) is the major progestational steroid that is secreted primarily by the CORPUS LUTEUM and the PLACENTA. Progesterone acts on the UTERUS, the MAMMARY GLANDS and the BRAIN. It is require...
T1263 Levonorgestrel D-Norgestrel Others , Estrogen/progestogen Receptor , Progesterone Receptor
Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device. The physiologic effect of levonorgestrel is by means of Inhibit Ovum Fertilization.
T1596 Chlormadinone acetate Gestafortin Progesterone Receptor , Androgen Receptor
Chlormadinone acetate (Gestafortin) is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive.
T5040 Medroxyprogesterone Estrogen/progestogen Receptor , Progesterone Receptor
Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.
T8395 Nomegestrol acetate Others , Progesterone Receptor
Nomegestrol acetate is a widely used progestin-like drug,which is characterized as a full agonist at the progesterone receptor
T1541 Drospirenone ZK 3059,Dihydrospirorenone Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , COX
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T7537 Norgestimate Progesterone Receptor
Norgestimate is an acetylated progestinused in combination with ethinyl estradiol as an oral contraceptive.
T28362 PF-02413873 PF02413873 Progesterone Receptor
PF-02413873 is a competitive antagonist of nonsteroidal progesterone receptor with a Ki of 2.6 nM. PF-02413873 can be used in studies about the treatment of gynecological conditions such as endometriosis.
T6819 Desogestrel Org-2969,Desogen,Desogestrelum,Cerazette Estrogen/progestogen Receptor , Progesterone Receptor
Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
T0996 Ethynodiol diacetate Ethynodiol acetate,8080 CB Estrogen/progestogen Receptor , Progesterone Receptor
Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with estrogens as an oral contraceptive.
T6713 Ulipristal Estrogen/progestogen Receptor , Progesterone Receptor
Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.
T2577 Dienogest STS 557 Apoptosis , Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy
Dienogest (STS 557) is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic activities that is used in hormone therap...
T1490 Gestodene SHB 331,WL 70 Estrogen/progestogen Receptor , Progesterone Receptor
Gestodene (WL 70) is a progestogen hormonal contraceptive.
T5174 Nestoron ST-1435,Segesterone Acetate,Nestorone,Elcometrine Estrogen/progestogen Receptor , Progesterone Receptor
Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).
T0870 Altrenogest R2267,RU2267,Allyltrenbolone,A35957 Estrogen/progestogen Receptor , Progesterone Receptor
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.
T14975 CJ-42794 CJ-042794 Others
CJ-42794 (CJ-042794) is a selective antagonist of prostaglandin E receptor subtype 4 (EP4). It inhibits [3H]-PGE2 binding to the human EP4 receptor (a mean pKi: 8.5). CJ-42794 is a binding affinity that was at least 200-...
T2527 Ulipristal acetate Ulipristal,CDB-2914 Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy
Ulipristal acetate (CDB-2914) is an orally bioavailable, acetate salt of ulipristal, a selective progesterone receptor modulator with anti-progesterone activity. Ulipristal binds to the progesterone receptor (PR), thereb...

Compounds

Dydrogesterone
T3036
Synonym:
Target: Progesterone Receptor
Gestonorone Capronate
T13703
Synonym:
Target: Prostaglandin Receptor
Norethindrone
T1514
Synonym: Norethisterone
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Progesterone
T0478
Synonym: Pregn-4-ene-3,20-dione
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite
Levonorgestrel
T1263
Synonym: D-Norgestrel
Target: Others, Estrogen/progestogen Receptor, Progesterone Receptor
Chlormadinone acetate
T1596
Synonym: Gestafortin
Target: Progesterone Receptor, Androgen Receptor
Medroxyprogesterone
T5040
Synonym:
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Nomegestrol acetate
T8395
Synonym:
Target: Others, Progesterone Receptor
Drospirenone
T1541
Synonym: ZK 3059,Dihydrospirorenone
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, COX
Norgestimate
T7537
Synonym:
Target: Progesterone Receptor
PF-02413873
T28362
Synonym: PF02413873
Target: Progesterone Receptor
Desogestrel
T6819
Synonym: Org-2969,Desogen,Desogestrelum,Cerazette
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Ethynodiol diacetate
T0996
Synonym: Ethynodiol acetate,8080 CB
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Ulipristal
T6713
Synonym:
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Dienogest
T2577
Synonym: STS 557
Target: Apoptosis, Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Gestodene
T1490
Synonym: SHB 331,WL 70
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Nestoron
T5174
Synonym: ST-1435,Segesterone Acetate,Nestorone,Elcometrine
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Altrenogest
T0870
Synonym: R2267,RU2267,Allyltrenbolone,A35957
Target: Estrogen/progestogen Receptor, Progesterone Receptor
CJ-42794
T14975
Synonym: CJ-042794
Target: Others
Ulipristal acetate
T2527
Synonym: Ulipristal,CDB-2914
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
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TargetMol