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Search Results for " mepi "

Targets

24

Compounds

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T2078 Fimepinostat CUDC-907,PI3K/HDAC Inhibitor,CUDC 907 Apoptosis , PI3K , HDAC
Fimepinostat (CUDC 907) is an orally bioavailable inhibitor of both phosphoinositide 3-kinase (PI3K) class I and pan-histone deacetylase (HDAC) enzymes, with potential antineoplastic activity. Upon oral administration, C...
T0946 Mepivacaine hydrochloride Mepivacaine HCl Sodium Channel
Mepivacaine hydrochloride (Mepivacaine HCl) is the hydrochloride salt form of mepivacaine, an amide derivative with local anesthetic properties.
T0765 Fomepizole Antizol-Vet,4-Methylpyrazole,Antizol P450 , CAT , AChR
Fomepizole (4-Methylpyrazole) is used as an antidote in confirmed or suspected methanol or ethylene glycol poisoning. Fomepizole(4-Methylpyrazole) is a competitive inhibitor of alcohol dehydrogenase, the enzyme that cata...
T22361 Mepivacaine Carbocaine Sodium Channel
Mepivacaine (Carbocaine) is an amide compound for local anaesthesia that causes transient loss of self-consciousness in humans or animals. mepivacaine acts by binding to specific voltage-gated sodium channels in nerve ce...
T0264 Zomepirac sodium salt Zomepirac Sodium,McN-2783-21-98 PGE Synthase , PDE
Zomepirac sodium salt (McN-2783-21-98) is a prostaglandin synthetase inhibitor.
T1860 Imepitoin AWD 131-138,ELB-138 GABA Receptor
Imepitoin (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist. It shows potent anticonvulsant and anxiolytic properties in rodent models.
T0257 Mepiroxol Mepyroxol,Lysateril Others
Mepiroxol (Lysateril), an antihyperlipidemic, is also called 3-PYRIDINEMETHANOL N-OXIDE.
T0127 Glimepiride Glimperide,HOE-490 Potassium Channel
Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.
T64332 Glimepiride sulfonamide Immunology/Inflammation related
Glimepiride sulfonamide is an antiinflammatory agent.
T69424 Zomepirac free acid
Zomepirac is a prostaglandin synthetase inhibitor. Zomepirac is an orally effective nonsteroidal anti-inflammatory drug (NSAID) that has antipyretic actions.
T37727 Methimepip dihydrobromide
Methimepip dihydrobromide is a selective H3R agonist.
T19921 Dimepiperate Yukamate,MUW 1193,MUW-1193,MUW1193,MY 93
Dimepiperate is an agent of biochemical.
T60329 Mepixetil
Mepixetil is a potent angiotensin II receptor antagonist[1].
T72245 Fomepizole hydrochloride 4-Methylpyrazole hydrochloride
Fomepizole hydrochloride (4-Methylpyrazole), a potent, orally active inhibitor of cytochrome P450 (CYP2E1) and a competitive inhibitor of alcohol dehydrogenase, prevents the conversion of methanol and ethylene glycol int...
T73408 Immepip
Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.
T78657 Azilsartan mepixetil potassium QR-01019K
Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more pronounced and enduring reduction in heart rate, and a high sa...
T16041 Mepixanox Pimexone Others
Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.
T35641 Trans-hydroxy Glimepiride
trans-hydroxy Glimepiride is an active metabolite of the sulfonylurea glimepiride .1It is formed from glimepiride primarily in the liver by the cytochrome P450 (CYP) isoform CYP2C9. 1.Langtry, H.D., and Balfour, J.A.Glim...
T35640 Trans-carboxy Glimepiride
trans-carboxy Glimepiride is a metabolite of the sulfonylurea glimepiride .1It is formed from glimepiride in a two-step process mediated by the cytochrome P450 (CYP) isoform CYP2C9 and cytosolic enzymes. 1.Noh, K., Kim, ...
T22863 Immepip dihydrobromide Others
Immepip dihydrobromide is a histamine H3 receptor agonist.
T71284 Glimepiride urethane
Glimepiride urethane is a third generation sulfonylurea compound, which increases the release of insulin from pancreatic beta cells. In addition, glimepiride increases the activity of intracellular insulin receptors. Gli...
T39063 Azilsartan mepixetil
Azilsartan mepixetil is a potent angiotensin II receptor antagonist with enhanced efficacy and prolonged duration of action. It exhibits more prominent and sustained effects in lowering blood pressure and heart rate, whi...
T12825 Timepidium bromide SA504,Sesden AChR
Timepidium bromide is an agent of anticholinergic.
T30205 Atromepine Dispan,Levomepat,TMT,Atromepinum
Atromepine is a bioactive chemical.

Compounds

Fimepinostat
T2078
Synonym: CUDC-907,PI3K/HDAC Inhibitor,CUDC 907
Target: Apoptosis, PI3K, HDAC
Mepivacaine hydrochloride
T0946
Synonym: Mepivacaine HCl
Target: Sodium Channel
Fomepizole
T0765
Synonym: Antizol-Vet,4-Methylpyrazole,Antizol
Target: P450, CAT, AChR
Mepivacaine
T22361
Synonym: Carbocaine
Target: Sodium Channel
Zomepirac sodium salt
T0264
Synonym: Zomepirac Sodium,McN-2783-21-98
Target: PGE Synthase, PDE
Imepitoin
T1860
Synonym: AWD 131-138,ELB-138
Target: GABA Receptor
Mepiroxol
T0257
Synonym: Mepyroxol,Lysateril
Target: Others
Glimepiride
T0127
Synonym: Glimperide,HOE-490
Target: Potassium Channel
Glimepiride sulfonamide
T64332
Synonym:
Target: Immunology/Inflammation related
Zomepirac free acid
T69424
Synonym:
Target:
Methimepip dihydrobromide
T37727
Synonym:
Target:
Dimepiperate
T19921
Synonym: Yukamate,MUW 1193,MUW-1193,MUW1193,MY 93
Target:
Mepixetil
T60329
Synonym:
Target:
Fomepizole hydrochloride
T72245
Synonym: 4-Methylpyrazole hydrochloride
Target:
Immepip
T73408
Synonym:
Target:
Azilsartan mepixetil potassium
T78657
Synonym: QR-01019K
Target:
Mepixanox
T16041
Synonym: Pimexone
Target: Others
trans-hydroxy Glimepiride
T35641
Synonym:
Target:
trans-carboxy Glimepiride
T35640
Synonym:
Target:
Immepip dihydrobromide
T22863
Synonym:
Target: Others
Glimepiride urethane
T71284
Synonym:
Target:
Azilsartan mepixetil
T39063
Synonym:
Target:
Timepidium bromide
T12825
Synonym: SA504,Sesden
Target: AChR
Atromepine
T30205
Synonym: Dispan,Levomepat,TMT,Atromepinum
Target:

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-01841 Serpin I2 Protein, Human, Recombinant (His) Human HEK293 Cells
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in some fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesis, infl...
TargetMol