Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Imepitoin (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist. It shows potent anticonvulsant and anxiolytic properties in rodent models.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 30.00 | |
2 mg | In stock | $ 44.00 | |
5 mg | In stock | $ 68.00 | |
10 mg | In stock | $ 101.00 | |
25 mg | In stock | $ 181.00 | |
50 mg | In stock | $ 328.00 | |
100 mg | In stock | $ 487.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 75.00 |
Description | Imepitoin (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist. It shows potent anticonvulsant and anxiolytic properties in rodent models. |
Kinase Assay | Cell-based determinations of mTOR inhibition: A high-throughput screening cell-based assay is developed using MDA-MB-468 cells to detect mTORC1 and mTORC2 activity. Cells are exposed for 2 hours to increasing concentrations of AZD8055. At the end of the incubation period, cells are fixed, washed, and probed with antibodies against S473 pAkt or against S235/236 phosphorylated S6 (pS6). Levels of phosphorylation are assessed using an Acumen laser scanning cytometer. |
Synonyms | AWD 131-138, ELB-138 |
Molecular Weight | 279.72 |
Formula | C13H14ClN3O2 |
CAS No. | 188116-07-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 13 mg/mL (46.48 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Imepitoin 188116-07-6 Membrane transporter/Ion channel Neuroscience GABA Receptor AWD 131-138 Inhibitor Gamma-aminobutyric acid Receptor ELB-138 ELB138 ELB 138 γ-Aminobutyric acid Receptor inhibit inhibitor