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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1281 | Bombesin | ||
Bombesin is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in mammals called neuromedin B and gastrin-releasing peptide. | |||
TP2239L | [D-Phe12]-Bombesin acetate | [D-Phe12]-Bombesin acetate(108437-87-2 free base) | Bombesin Receptor |
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion. | |||
TP1916L1 | [D-Phe12,Leu14]-Bombesin acetate | [D-Phe12,Leu14]-Bombesin acetate(108437-88-3 Free base) | Bombesin Receptor |
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion. | |||
TP1281L1 | Bombesin acetate(31362-50-2 free base) | Bombesin Receptor | |
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in mammals called neuromedin B and gastrin-releasing peptide. | |||
TP2239 | [D-Phe12]-Bombesin | Others | |
Bombesin receptor antagonist | |||
TP1916 | [D-Phe12,Leu14]-Bombesin | ||
Bombesin receptor antagonist that inhibits bombesin binding to rat brain with an IC50 value of 2 μM. Inhibits amylase release in vitro (IC50 = 4 μM) and attenuates bombesin-mediated suppression of food intake in vivo. | |||
T83490 | [Lys3]-Bombesin | ||
[Lys3]-Bombesin is a biologically active peptide used in PET (Positron Emission Tomography) imaging to identify GRPR (gastrin-releasing peptide receptor) positive prostate cancer. The compound, when conjugated with a cor... | |||
TN1849 | Kuwanon H | GPR , Bombesin Receptor | |
Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the physiological and pathological role of GRP. | |||
T2126 | MK-5046 | Bombesin Receptor | |
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). | |||
T4540 | ML-18 | Bombesin Receptor | |
ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM. | |||
T76601 | (D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14) | ||
(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14), a bombesin (BBN) antagonist, holds potential for cancer research applications [1]. | |||
T3S1612 | Kuwanon G | Moracenin B,Kuwanone G | Phosphatase , Antibacterial , Bombesin Receptor , AChR , AChE , Glucosidase |
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for Type II diabetes mellitus. 2. Kuwanon G has a... | |||
TP1701 | RC-3095 TFA | RC-3095 (TFA) | Bombesin Receptor |
RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity. | |||
TP2219L | Alytesin acetate | Others | |
Alytesin acetate is an amphibian bombesin-like peptide. | |||
T20604L | Litorin acetate(55749-97-8 Free base) | Bombesin Receptor | |
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the n... | |||
T20603L | Ranatensin acetate | Others | |
Ranatensin acetate, a undecapeptide isolated from skin of Rana pipiens, is a naturally occurring bombesin-like peptide. | |||
T28740 | SDZ-62-434 | SDZ 62 434,SDZ62434 | Platelet aggregation |
SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity that inhibits bombesin- and platelet-derived growth factor-induced DNA synthesis in quiescent Swiss 3T3 cells for the study of leukemia, human ... | |||
TP1442 | Neuromedin B | Endogenous Metabolite | |
Neuromedin B (NMB) is one of the bombesin (BN)-related peptides in mammals. It was originally purified from pig spinal cords, and it has been shown to be present in central nervous system as well as in gastrointestinal t... | |||
TP1913L1 | BA 1 acetate(183241-31-8 free base) | Bombesin Receptor | |
BA 1 acetate is a potent bombesin receptor agonist (IC50 values are 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively). Enhances glucose transport in obese and diabetic primary myocytes. Also stimulates NCI-H1299 ... | |||
TP1931L1 | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) | cholecystokinin |
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ... |