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Search Results for " vanilloid "

20

Compounds

Cat No. Product Name Synonyms Targets
T9247 Vanilloid receptor antagonist 1 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile TRP/TRPV Channel
Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.
T1062 Capsaicin Qutenza,8-Methyl-N-vanillyl-trans-6-nonenamide,Vanilloid,(E)-Capsaicin,Zostrix Apoptosis , TRP/TRPV Channel , Autophagy
Capsaicin ((E)-Capsaicin) is a natural product extracted from Capsicum annuum, and is a TRPV1 agonist (EC50=0.29 μM). Capsaicin has antitumor, anti-inflammatory, antioxidant and neuroprotective activities.
T83701 TRPV1-Tat TFA Transient Receptor Potential Vanilloid 1-Tat,736-745-Tat
TRPV1-Tat, a peptide antagonist targeting transient receptor potential vanilloid 1 (TRPV1), is composed of amino acids 736-745 derived from TRPV1's A-kinase anchor protein (AKAP)-binding domain, combined with the HIV Tat...
T6977 SB-366791 SB366791 TRP/TRPV Channel
SB-366791 is a new and selective cinnamide TRPV1 antagonist.
T6848 GSK1016790A GSK101 Calcium Channel , TRP/TRPV Channel
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
T12306 OMDM-5 Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T23106 Olvanil N-Vanillyloleamide,N-Vannilyloleoylamide TRP/TRPV Channel
Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.
T23322 SB 452533 TRP/TRPV Channel
SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).
T29522 ABT 102 ABT102,CHEMBL398338,ABT-102 TRP/TRPV Channel
ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
T13214L TRPV4 agonist-1 free base OUN67600 TRP/TRPV Channel
TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).
T14087 ABT-239 TRP/TRPV Channel
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists. It also acts as a transient receptor potential vanilloid type 1 (TRPV1) antagonist.
T7189 AMG9810 TRP/TRPV Channel
AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6 nM for human and rat TRPV1, respectively).
T37097 SET 2 TRP/TRPV Channel
SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.
TN1377 α-Spinasterol alpha-Spinasterol COX , Antibacterial , TRP/TRPV Channel
α-Spinasterol is a transient receptor potential vanilloid 1 (TRPV1) antagonist, has anti-inflammatory, antidepressant, antioxidant and antinociceptive effects. α-Spinasterol inhibits COX-1 andCOX-2 activities with IC50 v...
T22360 MDR-652 TRP/TRPV Channel
MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1 respectively and EC50s for hTRPV1 and rTRPV1 ...
T2163 Dihydrocapsaicin CCRIS1589,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide Others , TRP/TRPV Channel
Dihydrocapsaicin (CCRIS1589) is isolated from Capsicum fruit. Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Like capsaicin, dihydrocapsaicin is an...
T22586 Arvanil Others
Cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist
T23178 PPAHV Others
vanilloid TRPV1 (VR1) receptor agonist
T22527 6'-Iodoresiniferatoxin Others
TRPV1 (VR1) vanilloid receptor partial agonist

Compounds

Vanilloid receptor antagonist 1
T9247
Synonym: 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
Target: TRP/TRPV Channel
Capsaicin
T1062
Synonym: Qutenza,8-Methyl-N-vanillyl-trans-6-nonenamide,Vanilloid,(E)-Capsaicin,Zostrix
Target: Apoptosis, TRP/TRPV Channel, Autophagy
TRPV1-Tat TFA
T83701
Synonym: Transient Receptor Potential Vanilloid 1-Tat,736-745-Tat
Target:
SB-366791
T6977
Synonym: SB366791
Target: TRP/TRPV Channel
GSK1016790A
T6848
Synonym: GSK101
Target: Calcium Channel, TRP/TRPV Channel
OMDM-5
T12306
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel
OMDM-1
T12302
Synonym: (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide
Target: Endogenous Metabolite
Olvanil
T23106
Synonym: N-Vanillyloleamide,N-Vannilyloleoylamide
Target: TRP/TRPV Channel
SB 452533
T23322
Synonym:
Target: TRP/TRPV Channel
ABT 102
T29522
Synonym: ABT102,CHEMBL398338,ABT-102
Target: TRP/TRPV Channel
TRPV4 agonist-1 free base
T13214L
Synonym: OUN67600
Target: TRP/TRPV Channel
ABT-239
T14087
Synonym:
Target: TRP/TRPV Channel
AMG9810
T7189
Synonym:
Target: TRP/TRPV Channel
SET 2
T37097
Synonym:
Target: TRP/TRPV Channel
α-Spinasterol
TN1377
Synonym: alpha-Spinasterol
Target: COX, Antibacterial, TRP/TRPV Channel
MDR-652
T22360
Synonym:
Target: TRP/TRPV Channel
Dihydrocapsaicin
T2163
Synonym: CCRIS1589,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide
Target: Others, TRP/TRPV Channel
Arvanil
T22586
Synonym:
Target: Others
PPAHV
T23178
Synonym:
Target: Others
6'-Iodoresiniferatoxin
T22527
Synonym:
Target: Others
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TargetMol