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SB-366791

Catalog No. T6977 CAS 472981-92-3

Synonyms: SB366791

SB-366791 is a new and selective cinnamide TRPV1 antagonist.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

SB-366791, CAS 472981-92-3

Pack Size	Availability	Price/USD
2 mg	In stock	$ 33.00
5 mg	In stock	$ 46.00
10 mg	In stock	$ 64.00
25 mg	In stock	$ 135.00
50 mg	In stock	$ 213.00
100 mg	In stock	$ 353.00
1 mL * 10 mM (in DMSO)	In stock	$ 47.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description	SB-366791 is a new and selective cinnamide TRPV1 antagonist.
Targets&IC50	TRPV1:5.7 nM

Synonyms	SB366791
Molecular Weight	287.74
Formula	C16H14ClNO2
CAS No.	472981-92-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 28.8 mg/mL (100 mM)

Ethanol: 2.9 mg/mL (10 mM)

References and Literature

1. Gunthorpe MJ,et al. Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist. Neuropharmacology. 2004 Jan;46(1):133-49.

Related compound libraries

This product is contained In the following compound libraries：

Highly Selective Inhibitor Library Membrane Protein-targeted Compound Library Inhibitor Library Anti-Cancer Compound Library Bioactive Compounds Library Max Target-Focused Phenotypic Screening Library NO PAINS Compound Library Bioactive Compound Library CNS-Penetrant Compound Library Neuronal Signaling Compound Library

Related Products

Related compounds with same targets

Oleoyl Serotonin Diphenyleneiodonium chloride AMG9810 ABT 102 GSK3395879 Pico145 M8-B Hydrochloride TRPM8 antagonist 2

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

SB-366791 472981-92-3 Membrane transporter/Ion channel TRP/TRPV Channel potential transient potent Transient receptor potential channels Inhibitor vanilloid SB 366791 inhibit receptor SB366791 selective TRP Channel inflammation inhibitor

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.