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Search Results for " sedative "

20

Compounds

Cat No. Product Name Synonyms Targets
T36949 Niaprazine 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...
T3563 Lvguidingan Others
Lvguidingan is an Anticonvulsant agent.
T8887 2'MeO6MF GABA Receptor
2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional recovery and dampens the stroke-induced inflammatory response...
T6464 Detomidine hydrochloride MPV-253 AII,Domosedan,Detomidine HCl Adrenergic Receptor
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
T2S2109 Skimmianine beta-Fagarine,Skimmianin,Chloroxylonine,Skimmiamine Others
1. Skimmianine (Chloroxylonine) is a spasmolytic agent. 2. Skimmianine (Chloroxylonine) shows pharmacol. props. similar to 2-(Methylamino)-1-phenyl-1-propanol BCJ45-G.
T7699 AZD7325 AZD-7325 P450 , GABA Receptor
AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
T14983 Clomethiazole Distraneurin,Chlormethiazole,5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE P450 , GABA Receptor
Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It also has the potential for treating convulsive status epilepticus. Chlormethiazole inhibits cytochrome P450 isoforms: C...
T0370 Pheniramine maleate Daneral,Inhiston,Trimetose 5-HT Receptor , Histamine Receptor
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of the endothelium-derived re...
T0205 Brompheniramine maleate Dimotane,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane 5-HT Receptor , Histamine Receptor
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
TN2865 (E)-3,4,5-Trimethoxycinnamic acid O-Methylsinapic acid,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid Others
(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.
T23445 Anxiolytic/nonsedative agent-1 TCS 1205 GABA Receptor
Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α...
T11506 Guaiapate Mg 5454,Klamar Others
Guaiapate has an antitussive and sedative effect.
T30248 AZD 3043 AZD-3043,THRX 918661,AZD3043
AZD 3043 is a propofol derivative which acts as a sedative-hypnotic agent.
T31724 Etoxybamide Others
Etoxybamide is a drug candidate for sedative (hypnotic).
T28887 Suriclone RP-31264,RP31264,RP 31264 GABA Receptor
Suriclone (RP 31264) is a selective cyclic pyrrolidone analog with sedative and anxiolytic activity, but not significant sedative effects.Suriclone shows its effects by modulating GABA-A receptors.
T14314 Apronal Apronalide,Allylisopropylacetylurea Others
Apronal (Apronalide) has the hypnotic and sedative capacity and can be used for studies about neuropsychiatry disorders.
T83647 (Z)-Tenilapine Others
(Z)-Tenilapine is trans-Tenilapine, cis-Tenilapine has sedative activity.
T28303 Pazinaclone A-77000,DN-2327,DN2327,DN 2327,A 77000,A77000 GABA Receptor
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
T0227 Bromisoval 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,BRN 1773255,Bromovalerylurea,Bromaral Others
Bromisoval (Isobromyl) is a mild hypnotic and sedative with potential toxicity.
T7521 Azaphen Pipofezin hydrochloride,Pipofezine hydrochloride,Azafen 5-HT Receptor , Serotonin Transporter
Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.

Compounds

Niaprazine
T36949
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Lvguidingan
T3563
Synonym:
Target: Others
2'MeO6MF
T8887
Synonym:
Target: GABA Receptor
Detomidine hydrochloride
T6464
Synonym: MPV-253 AII,Domosedan,Detomidine HCl
Target: Adrenergic Receptor
Skimmianine
T2S2109
Synonym: beta-Fagarine,Skimmianin,Chloroxylonine,Skimmiamine
Target: Others
AZD7325
T7699
Synonym: AZD-7325
Target: P450, GABA Receptor
Clomethiazole
T14983
Synonym: Distraneurin,Chlormethiazole,5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE
Target: P450, GABA Receptor
Pheniramine maleate
T0370
Synonym: Daneral,Inhiston,Trimetose
Target: 5-HT Receptor, Histamine Receptor
Brompheniramine maleate
T0205
Synonym: Dimotane,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
(E)-3,4,5-Trimethoxycinnamic acid
TN2865
Synonym: O-Methylsinapic acid,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid
Target: Others
Anxiolytic/nonsedative agent-1
T23445
Synonym: TCS 1205
Target: GABA Receptor
Guaiapate
T11506
Synonym: Mg 5454,Klamar
Target: Others
AZD 3043
T30248
Synonym: AZD-3043,THRX 918661,AZD3043
Target:
Etoxybamide
T31724
Synonym:
Target: Others
Suriclone
T28887
Synonym: RP-31264,RP31264,RP 31264
Target: GABA Receptor
Apronal
T14314
Synonym: Apronalide,Allylisopropylacetylurea
Target: Others
(Z)-Tenilapine
T83647
Synonym:
Target: Others
Pazinaclone
T28303
Synonym: A-77000,DN-2327,DN2327,DN 2327,A 77000,A77000
Target: GABA Receptor
Bromisoval
T0227
Synonym: 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,BRN 1773255,Bromovalerylurea,Bromaral
Target: Others
Azaphen
T7521
Synonym: Pipofezin hydrochloride,Pipofezine hydrochloride,Azafen
Target: 5-HT Receptor, Serotonin Transporter
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TargetMol