Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α2β2γ2, α5β3γ2, respectively. Anxiolytic/nonsedative agent-1 shows α2 selective efficacy in vitro and anxioselective effects in vivo.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 98.00 | |
2 mg | In stock | $ 147.00 | |
5 mg | In stock | $ 195.00 | |
10 mg | In stock | $ 256.00 | |
25 mg | In stock | $ 581.00 | |
50 mg | In stock | $ 829.00 | |
100 mg | In stock | $ 1,150.00 | |
500 mg | In stock | $ 2,280.00 |
Description | Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α2β2γ2, α5β3γ2, respectively. Anxiolytic/nonsedative agent-1 shows α2 selective efficacy in vitro and anxioselective effects in vivo. |
Synonyms | TCS 1205 |
Molecular Weight | 337.33 |
Formula | C18H15N3O4 |
CAS No. | 355022-97-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 1mg/ml, Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Anxiolytic/nonsedative agent-1 355022-97-8 Membrane transporter/Ion channel Neuroscience GABA Receptor TCS-1205 TCS1205 TCS 1205 inhibitor inhibit