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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10876 | CPA inhibitor | Carboxypeptidase inhibitor | Carboxypeptidase |
CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM. | |||
T16263 | N6-Cyclopentyladenosine | UK-80882,CPA | Adenosine Receptor |
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 recepto... | |||
TP1560 | C(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm | ||
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively. | |||
T27138 | Declopramide | OXI-104,IMO-B,3-Chloroprocainamide | Apoptosis |
Declopramide (OXI-104) is a novel chemosensitizer with antitumor activity that induces apoptosis and can be used to study colorectal cancer and inflammatory bowel disease. | |||
TP1473 | Velmupressin | c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively. | |||
TP1205 | Velmupressin acetate | V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively. | |||
T2895 | Lupeol | Fagarasterol,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol | Apoptosis , Androgen Receptor , Akt |
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity. | |||
T20701 | MCPA | NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone | Others |
MCPA(Krezone) is a highly effective phenoxy herbicide. Use of MCPA would have impacts on nearby water and soil resources. | |||
T22489 | 2'-MeCCPA | 2-Chloro-N-cyclopentyl-2′-C-methyladenosine | HCV Protease , Adenosine Receptor |
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenylate cyclase activity with an IC value of 13.1 nM.2'-MeCCPA ... | |||
T21519 | CCPA | 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE | Adenosine Receptor |
CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor | |||
T1025 | Tranylcypromine (2-PCPA) hydrochloride | Tranylcypromine (2-PCPA) HCl,SKF-385 HCl | Histone Demethylase , MAO |
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression. | |||
T77567 | BCPA | Others | |
BCPA is a non-cytotoxic Pin1 modulator.BCPA modulates osteoclast activation and attenuates the reduction of Pin1 protein, thereby inhibiting RANKL-induced receptor activators of osteoclastogenesis.BCPA is used in the stu... | |||
T60359 | Cis-4-Br-2,5-F2-PCPA | ||
cis-4-Br-2,5-F2-PCPA (S1024) inhibits LSD1 and LSD2 with Ki values of 94 nM and 8.4 μM, respectively. There is aberrant expression of LSD1 in cancer stem cells, cis-4-Br-2,5-F2-PCPA inhibits LSD1 cell proliferation and b... | |||
T20948 | MCPA-thioethyl | HOK 7501,HOK7501,HOK-7501 | |
MCPA-thioethyl is a biochemical. | |||
T81054 | T-1-MCPAB | VEGFR | |
T-1-MCPAB, a VEGFR-2 inhibitor with an IC50 of 0.135 µM, effectively suppresses MCF7 cell migration and has applications in cancer research [1]. | |||
T41143 | PCPA methyl ester hydrochloride | 4-Chloro-DL-phenylalanine methyl ester hydrochloride | 5-HT Receptor , Hydroxylase |
pCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride) is an inhibitor of tryptophan hydroxylase inhibitor and 5-HT synthesis. pCPA methyl ester hydrochloride is permeable across the blood... | |||
T82765 | CcpA-IN-1 | Antibiotic | |
CcpA-IN-1 is a Staphylococcus aureus antibiotic exhibiting significant bactericidal activity (MICs=460 nM) [1]. | |||
T74170 | MOCPAC | ||
MOCPAC is an HDAC1 specific substrate [1] . | |||
T33228 | MCPA-potassium | ||
MCPA-potassium is a bioactive chemical. | |||
T33227 | MCPA-butyl | Yamaclean M | |
MCPA-butyl is a biochemical. |