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20

Compounds

Cat No. Product Name Synonyms Targets
T3S0081 Oxypeucedanin (+-)-Oxypeucedanin,Oxypeucadanin Potassium Channel
1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocke...
T8118 Bekanamycin Kanamycin B Antibacterial , Antibiotic
Bekanamycin (Kanamycin B) is an aminoglycoside antibiotic.
T20766 Sulfisoxazole acetyl Gantrisin,Acetylsulfisoxazole,Gantrisin Pediatric,Lipo Gantrisin Antibacterial
Sulfisoxazole acetyl (Gantrisin) is an agent with antibacterial activity. Sulfisoxazole acetyl is a Sulfisoxazole derivative with antibacterial activity. Sulfisoxazole acetyl is an inhibitor of dihydropteroate synthase.
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T1320 Disopyramide Triombrin,Hypaque sodium,amidotrizoate sodium Potassium Channel , Sodium Channel , AChR
Disopyramide (Triombrin) is a class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the h...
T1676 Rosuvastatin ZD 4522 Potassium Channel , HMG-CoA Reductase , Autophagy
Rosuvastatin (ZD 4522) is an antilipemic agent that competitively inhibits hydroxymethyl-glutaryl-coenzyme A (HMG-CoA) reductase. HMG-CoA reductase catalyzes the conversion of HMG-CoA to mevalonic acid, the rate-limiting...
T7894 Tazarotenic acid AGN-190299 Others
Tazarotenic acid (AGN-190299) is a retinoid prodrug which is converted to its active form
T1510 Rosuvastatin calcium ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium Potassium Channel , HMG-CoA Reductase , Autophagy
Rosuvastatin calcium (ZD4522) , a selective and competitive inhibitor of hepatic hydroxymethyl-glutaryl coenzyme A (HMG-CoA) reductase, has antilipidemic activity.
T3189 B7/CD28 interaction inhibitor 1 CTLA-4 inhibitor Others
B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) is a potent CTLA-4 inhibitor.
T9044 SORT-PGRN interaction inhibitor 1 Neurotensin Receptor
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
T12350 P53 and MDM2 proteins-interaction-inhibitor dihydrochloride Others
p53 and MDM2 proteins-interaction-inhibitor dihydrochloride is a interaction inhibitor between p53 and MDM2 proteins.
T80381 SAAP Fraction 3
SAAP Fraction 3, an antimicrobial peptide, exhibits activity against P. haemolytica in Zn-saline buffer [1].
T28219 NusB-NusE interaction inhibitor-1
NusB-NusE interaction inhibitor-1 is a modulator of the NusB-NusE interaction.
T82245 HA-CD44 interaction inhibitor 1
Antitumor agent-109 (compound 6) is a dual-function inhibitor that targets hyaluronic acid and CD44, which are involved in tumor progression and invasion. It demonstrates potent antitumor activity, specifically inhibitin...
T82902 Beclin1-Bcl-2 interaction inhibitor 1
Beclin1-Bcl-2 Interaction Inhibitor 1 effectively disrupts the binding of Beclin 1 to Bcl-2, and is utilized in cancer and neurodegeneration research [1].
T79756 Beclin1-ATG14L interaction inhibitor 1 Autophagy
Beclin1-ATG14L Interaction Inhibitor 1 (COM 19) is a selective inhibitor targeting the specific interaction between Beclin1 and ATG14L. It impedes the formation of complex I in the lipid kinase VPS34, thus inhibiting aut...
T12351 P53 and MDM2 proteins-interaction-inhibitor (racemic) p53-and-mdm2-proteins-interaction-inhibitor-racemic Others
p53 and MDM2 proteins-interaction-inhibitor (racemic) is an inhibitor of the interaction between p53 and MDM2 proteins.
T82244 HA-CD44 interaction inhibitor 2
Antitumor Agent-108 (Compound 5), an inhibitor of the Hyaluronic Acid (HA)-CD44 interaction, effectively disrupts cancer spheroid integrity and exhibits antiproliferative activity against cancer cells [1].
T81126 SORT-PGRN interaction inhibitor 2
SORT-PGRN Interaction Inhibitor 2 is a compound that downregulates SORT1 protein expression and enhances extracellular progranulin (PGRN) secretion in various mammalian cell lines, and is utilized in the study of neurolo...
T79106 SORT-PGRN interaction inhibitor 3 Neurotensin Receptor
SORT-PGRN Interaction Inhibitor 3 (Compound 13), with an IC50 value of 0.17 μM, acts as an inhibitor of the SORT-PGRN interaction, and is utilized in the study of neurodegenerative diseases [1].

Compounds

Oxypeucedanin
T3S0081
Synonym: (+-)-Oxypeucedanin,Oxypeucadanin
Target: Potassium Channel
Bekanamycin
T8118
Synonym: Kanamycin B
Target: Antibacterial, Antibiotic
Sulfisoxazole acetyl
T20766
Synonym: Gantrisin,Acetylsulfisoxazole,Gantrisin Pediatric,Lipo Gantrisin
Target: Antibacterial
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Disopyramide
T1320
Synonym: Triombrin,Hypaque sodium,amidotrizoate sodium
Target: Potassium Channel, Sodium Channel, AChR
Rosuvastatin
T1676
Synonym: ZD 4522
Target: Potassium Channel, HMG-CoA Reductase, Autophagy
Tazarotenic acid
T7894
Synonym: AGN-190299
Target: Others
Rosuvastatin calcium
T1510
Synonym: ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium
Target: Potassium Channel, HMG-CoA Reductase, Autophagy
B7/CD28 interaction inhibitor 1
T3189
Synonym: CTLA-4 inhibitor
Target: Others
SORT-PGRN interaction inhibitor 1
T9044
Synonym:
Target: Neurotensin Receptor
p53 and MDM2 proteins-interaction-inhibitor dihydrochloride
T12350
Synonym:
Target: Others
SAAP Fraction 3
T80381
Synonym:
Target:
NusB-NusE interaction inhibitor-1
T28219
Synonym:
Target:
HA-CD44 interaction inhibitor 1
T82245
Synonym:
Target:
Beclin1-Bcl-2 interaction inhibitor 1
T82902
Synonym:
Target:
Beclin1-ATG14L interaction inhibitor 1
T79756
Synonym:
Target: Autophagy
p53 and MDM2 proteins-interaction-inhibitor (racemic)
T12351
Synonym: p53-and-mdm2-proteins-interaction-inhibitor-racemic
Target: Others
HA-CD44 interaction inhibitor 2
T82244
Synonym:
Target:
SORT-PGRN interaction inhibitor 2
T81126
Synonym:
Target:
SORT-PGRN interaction inhibitor 3
T79106
Synonym:
Target: Neurotensin Receptor
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TargetMol