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Sulfisoxazole acetyl

Catalog No. T20766 CAS 80-74-0

Synonyms: Gantrisin, Acetylsulfisoxazole, Gantrisin Pediatric, Lipo Gantrisin

Sulfisoxazole acetyl (Gantrisin) is an agent with antibacterial activity. Sulfisoxazole acetyl is a Sulfisoxazole derivative with antibacterial activity. Sulfisoxazole acetyl is an inhibitor of dihydropteroate synthase.

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Sulfisoxazole acetyl, CAS 80-74-0

Pack Size	Availability	Price/USD
5 mg	In stock	$ 50.00
10 mg	In stock	$ 70.00
25 mg	In stock	$ 114.00
50 mg	In stock	$ 167.00
100 mg	In stock	$ 248.00
500 mg	In stock	$ 535.00
1 mL * 10 mM (in DMSO)	In stock	$ 61.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	Gantrisin, Acetylsulfisoxazole, Gantrisin Pediatric, Lipo Gantrisin
Molecular Weight	309.34
Formula	C13H15N3O4S
CAS No.	80-74-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 4.8 mg/mL (15.52 mM)

References and Literature

1. Eunyoung Kim, et al. Simultaneous determination of N(1)-acetyl sulfisoxazole and its metabolites, and relative bioavailability compare to sulfisoxazole in rats. J Pharm Biomed Anal. 2016 Sep 10;129:117-120. 2. Oh K, Baek MC, Kang W. Quantitative determination of sulfisoxazole and its three N-acetylated metabolites using HPLC-MS/MS, and the saturable pharmacokinetics of sulfisoxazole in mice. J Pharm Biomed Anal. 2016 Sep 10;129:332-338. 3. LOUGHLIN EH, MULLIN WG. The relative absorption and elimination of sulfisoxazole and acetyl sulfisoxazole. Antibiot Chemother (Northfield). 1955 Nov;5(11):609-15. 4. Bloedow DC, Hayton WL. Saturable first-pass metabolism of sulfisoxazole N1-acetyl in rats. J Pharm Sci. 1976 Mar;65(3):334-8.

Related compound libraries

This product is contained In the following compound libraries：

Drug Repurposing Compound Library Inhibitor Library Anti-Bacterial Compound Library Approved Drug Library FDA-Approved Drug Library Orally Active Compound Library ReFRAME Related Library Bioactive Compound Library Bioactive Compounds Library Max FDA-Approved & Pharmacopeia Drug Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Sulfisoxazole acetyl 80-74-0 Microbiology/Virology Antibacterial Inhibitor antibacterial action N1-Acetylsulfisoxazole inhibit Bacterial Gantrisin Acetylsulfisoxazole Sulfisoxazole derivative Gantrisin Pediatric Lipo Gantrisin orally active dihydropteroate synthase inhibitor

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