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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22406 | Prazosin | Prazosine,Furazosin,Prazocin | Adrenergic Receptor |
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension. | |||
T1050 | Prazosin hydrochloride | Prazosin hydrochloride,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,Minipress | Potassium Channel , MRP , Adrenergic Receptor , ABC , Autophagy |
Prazosin hydrochloride (Vasoflex) reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not completely known. Prazosin hydrochloride is a synthetic ... | |||
T63980 | BODIPY FL prazosin | ||
BODIPY FL prazosin is a fluorescent α1-adrenergic antagonist that acts on α1a-AR (Ki: 14.5 nM) and α1b-AR (Ki: 43.3 nM). BODIPY FL prazosin can be used for the study of subcellular localization differences in α1-adrenoce... | |||
T10998 | Deriglidole | SL 86-0715 | Adrenergic Receptor |
Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does not show activity against prazosin and rat co... | |||
T0993 | Methoxamine hydrochloride | Methoxamine HCl | Adrenergic Receptor |
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION. | |||
T22232 | Alfuzosin | ||
Alfuzosin, a quinazoline derivative, is a selective and competitive antagonist of the α1 adrenergic receptor, primarily used to manage benign prostatic hyperplasia (BPH). It effectively targets and mitigates alpha1-adren... | |||
T67790 | Biricodar dicitrate | VX 710,VX 710-3 | NF-κB , AChR |
Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer. | |||
T25793 | Metazosin | Kenosin | |
Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex. | |||
T31022 | CP 59430 | CP-59430,CP59430 | |
CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist. | |||
T62476 | Trimazosin | ||
Trimazosin is an orally active quinazoline derivative, structurally related to prazosin. trimazosin has hypotensive activity by selectively blocking alpha1-adrenoceptors. | |||
T22680 | CP-100356 hydrochloride | CP-100356 HCl,CP 100356 hydrochloride | BCRP |
CP-100356 hydrochloride is an orally active and low micromolar dual inhibitor of MDR1 (P-gp) and BCRP, a nucleotide-derived substrate analogue with inhibitory effects on MDR1-mediated Calcein-AM transporter and BCRP-medi... | |||
T71122 | Carsatrin (free base) | ||
Carsatrin is purinylpiperazine derivative. as cardiotonic and antiarrhythmic. Carsatrin acts as positive inotropic agent that increases twitch tension and prolongs the action potential (AP) duration of ventricular muscle... | |||
T70975 | Carsatrin succinate | ||
Carsatrin succinate is the salt form of Carsatin, a purinylpiperazine derivative used as a cardiotonic and antiarrhythmic. Carsatrin acts as positive inotropic agent that increases twitch tension and prolongs the action ... |