eta — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T12157	ETA antagonist 1		Others
	ETA antagonist 1 is an antagonist of ETA selective (IC50 of 0.08 μM).		Others
T31672	Erythrofuranosyladenine	9-β-D-Erythrofuranosyladenine,ETA
	Erythrofuranosyladenine(9-beta-D-Erythrofuranosyladenine, ETA) is a nontoxic MTAP substrate. Erythrofuranosyladenine is an effective salvage agent for methylthioadenosine phosphorylase–selective therapy of T-cell acute l...
T6258	Zibotentan	ZD4054	Apoptosis , Endothelin Receptor
	Zibotentan (ZD4054) (ZD4054) is a specific Endothelin (ET)A antagonist with IC50 of 21 nM, exhibiting no activity at ETB. Phase 3.		Apoptosis , Endothelin Receptor
T2561	Macitentan	ACT-064992	Apoptosis , Endothelin Receptor
	Macitentan (ACT-064992) is an endothelin receptor antagonist that is used in the therapy of pulmonary arterial hypertension (PAH).		Apoptosis , Endothelin Receptor
T15595L	IRL-1620 acetate	IRL-1620 acetate（142569-99-1 free base）	Endothelin Receptor
	IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a Ki of 16 pM which is more selective than ETA with a Ki of 19 μM.		Endothelin Receptor
T19309L1	Endothelin 1 (swine, human) acetate	Endothelin 1 (swine, human) acetate(117399-94-7 free base)	Endothelin Receptor
	Endothelin 1 (swine, human) acetate is a synthetic peptide with the sequence of human and swine Endothelin 1. Endothelin 1 is a potent endogenous vasoconstrictor and acts through two types of receptors ETA and ETB.		Endothelin Receptor
T22540L	Ac-Endothelin-1 (16-21), human acetate		Others
	Ac-Endothelin-1 (16-21), human acetate, the principal peptide of the endothelin family, has been shown to have a variety of biological activities in both vascular and nonvascular tissues. The C-terminal fragment, which i...		Others
TNU0758	2-Aminopurine-9-beta-D-(2’-deoxy)riboside		Others
	2-Aminopurine-9-beta-D-(2’-deoxy)riboside is a derivative of 2-Aminopurine.		Others
T5146	Eptifibatide acetate (148031-34-9 free base)	Eptifibatide acetate	Others
	Eptifibatide acetate (148031-34-9 free base) (Eptifibatide acetate) , an antiplatelet drug of the glycoprotein IIb/IIIa inhibitor class, is a cyclic heptapeptide constructed from 6 amino acids and a mercaptopropionyl res...		Others
T12710	Retagliptin Phosphate	SP 2086	Proteasome , DPP-4
	Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.		Proteasome , DPP-4
T1070	Cefmetazole sodium	Sodium cefmetazole	Antibacterial , Antibiotic
	Cefmetazole sodium (Sodium cefmetazole) is a semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types...		Antibacterial , Antibiotic
TN7071	Ergosterol Acetate	Ergosta-5,7,22-trien-3-beta-yl acetate	Others
	Ergosterol Acetate (Ergosta-5,7,22-trien-3-beta-yl acetate) is one of the acetate derivatives of Ergosterol from Monascus anka.		Others
T20366	Beta-Nicotyrine	Nicotyrine,alpha-Nicotyrine	Others
	beta-Nicotyrine is a tobacco alkaloids Metabolite in the liver.		Others
T35372	Zinc acetate	Dicarbomethoxyzinc	Others
	Zinc acetate (Dicarbomethoxy) can induce the expression of metallothionein in intestinal cells.		Others
T3272	Metamizole magnesium	Metamizolemagnesiumsalt	Antibiotic
	Metamizole magnesium (Metamizolemagnesiumsalt) is a pain reliever, which can antispasmodic.		Antibiotic
T68052	Delmetacin	Demethacin	CXCR
	Delmetacin (Demethacin) is a non-steroidal anti-inflammatory compound with anti-inflammatory and analgesic activity and inhibitory effects on the CXC chemokine receptor CXCR1.		CXCR
T8832	Eledoisin trifluoroacetate (69-25-0 free base)	Eledoisin trifluoroacetate	Others
	Eledoisin trifluoroacetate (69-25-0 free base) is a peptide extracted from the posterior salivary glands of certain small octopi (Eledone spp., Mollusca), or obtained by synthesis. Its actions resemble those of SUBSTANCE...		Others
TN3500	Beta-Amyrone	β-Amyron	COX , AChR , PPAR , Antifection
	beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM. beta-Amyrone has anti-inflammatory activity through inhibiting the expression of COX-2. beta-Amyrone exhibits a...		COX , AChR , PPAR , Antifection
T37422L	Ras Inhibitory Peptide acetate	Ras Inhibitory Peptide acetate(159088-48-9 Free base)	Ras
	Ras Inhibitory Peptide acetate is a peptide involved in the Ras-dependent signaling pathway that plays an important role in human cancers initiated by oncogenic receptors.		Ras
T5817	PKC-theta inhibitor hcl	PKC-theta inhibitor	PKC
	PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM).		PKC