aminopeptidase — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T9345	Aminopeptidase M		Others
	Aminopeptidase M (AMP) inhibition is of interest for several diseases, such as highly vascularized cancer types.		Others
T61278	Aminopeptidase-IN-1		Aminopeptidase
	Aminopeptidase-IN-1 is a potent inhibitor of insulin-regulated aminopeptidase (IRAP) (Ki: 7.7 μM).Aminopeptidase-IN-1 can be used in studies of cognitive and memory disorders.		Aminopeptidase
T36943	Aminopeptidase N Inhibitor
	Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM). It is selective for AP-N/CD13 over matrix metalloproteinase-9 (MMP-9), angiotensin converting enzyme (ACE), neutral endopeptidase (...
T76568	Aminopeptidase N Ligand (CD13) NGR peptide
	Aminopeptidase N Ligand (CD13) NGR peptide, a polypeptide that targets CD13, functions as a carrier for mediating intracellular transmission and is commonly utilized in cancer research [1] [2].
TQ0047	DG051		Aminopeptidase
	DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).		Aminopeptidase
T1257	Bestatin	Ubenimex	Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
	Bestatin (Ubenimex) competitively inhibits many aminopeptidases, including B, N and leucine aminopeptidases. Ubenimex is a microbial metabolite and dipeptide with potential immunomodulatory and antitumor activities. Amin...		Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
T11221	ERAP1-IN-1		Others
	ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activi...		Others
T6301	Tosedostat	CHR-2797	Aminopeptidase , AChR
	Tosedostat (CHR-2797) is an orally bioavailable inhibitor of the M1 family of aminopeptidases with potential antineoplastic activity. Tosedostat is converted intracellularly into a poorly membrane-permeable active metabo...		Aminopeptidase , AChR
T3715	Acebilustat	CTX-4430	Aminopeptidase , LTR
	Acebilustat (CTX-4430) (ZK322) is an effective and specific leukotriene B4 hydrolase inhibitor.		Aminopeptidase , LTR
T21859	ARM1		Aminopeptidase , Epoxide Hydrolase
	ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.		Aminopeptidase , Epoxide Hydrolase
T7958	Methyl arachidate	Methyl Icosanoate	Others , Aminopeptidase
	Methyl arachidate (Methyl Icosanoate) is an esterified form of arachidic acid		Others , Aminopeptidase
T3529	Bestatin hydrochloride	Ubenimex hydrochloride	Integrin , Aminopeptidase , Antibacterial , Antibiotic
	Bestatin hydrochloride (Ubenimex hydrochloride) is an inhibitor of aminopeptidase N (APN)/CD13 and aminopeptidase B.		Integrin , Aminopeptidase , Antibacterial , Antibiotic
T16684	Puromycin aminonucleoside	NSC 3056	Apoptosis , Proteasome , Aminopeptidase , Antibacterial , Antibiotic
	Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner.
T21696	SC-57461A		Aminopeptidase
	SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor.		Aminopeptidase
T28482	Firibastat	QGC 001,QGC-001,RB-150,RB150,QGC001,RB 150	Aminopeptidase
	Firibastat (RB150) is a glutamyl aminopeptidase antagonist and an orally active brain penetrating prodrug of EC33. It is a first-in-class brain aminopeptidase A (APA) inhibitor with a Ki of 200 nM. Firibastat selectively...		Aminopeptidase
T5652	L(+)-Leucinol		Aminopeptidase
	L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase.		Aminopeptidase
T18997	GPDA	Glycylproline p-nitroanilide tosylate,GPN	Others
	GPDA (Glycylproline p-nitroanilide tosylate) is a substrate of X-Prolyl dipeptidyl-aminopeptidase in the enzyme assay.		Others
TP1181	Bradykinin (2-9)	Des-Arg1-bradykinin	Bradykinin Receptor
	Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P.		Bradykinin Receptor
T60021	EcMetAP-IN-1		Others
	ecMetAP-IN-1 can be used as a QSAR model to study methionine aminopeptidase inhibitor as an anticancer agent using multiple linear regression.		Others
T64341	H-β-Ala-AMC TFA		Others
	H-β-Ala-AMC TFA is a substrate for aminopeptidase. Building block for synthesizing the fluorogenic vanin I substrate pantothenate-AMC.		Others