Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 117.00 | |
5 mg | In stock | $ 470.00 | |
10 mg | In stock | $ 683.00 | |
25 mg | In stock | $ 987.00 | |
50 mg | In stock | $ 1,390.00 | |
100 mg | In stock | $ 1,880.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 447.00 |
Description | DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM). |
Targets&IC50 | LTA4H:47 nM (IC50) |
In vitro | DG051 is a potent inhibitor of LTA4H aminopeptidase activity against L-alanine p-nitroanilide (IC50: 72 nM). DG051 inhibits human whole blood (HWB) with IC50 of 37 nM [1]. DG-051 is an LTA4H inhibitor, currently in Phase II clinical development for the prevention of heart attack [2]. |
Molecular Weight | 426.33 |
Formula | C21H25Cl2NO4 |
CAS No. | 929915-58-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 317 mg/mL (743.56 mM)
You can also refer to dose conversion for different animals. More
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DG051 929915-58-2 Metabolism Aminopeptidase inhibit Inhibitor DG 051 DG-051 inhibitor