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PEPA

Name: PEPA
Brand: TargetMol
SKU: T12406
Price: 32 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T12406Cas No. 141286-78-4

PEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.

PEPA

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Purity: 97.31%

Catalog No. T12406Cas No. 141286-78-4

PEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.

Pack Size	Price	Availability
5 mg	$32	In Stock
10 mg	$48	In Stock
25 mg	$106	In Stock
50 mg	$208	In Stock
100 mg	$309	In Stock
1 mL x 10 mM (in DMSO)	$34	In Stock

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Batch Information

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Purity:97.31%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description

PEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.

Chemical Properties

Molecular Weight	402.44
Formula	C₁₆H₁₆F₂N₂O₄S₂
Cas No.	141286-78-4
Smiles	NC(=O)COc1c(F)cc(SCCNS(=O)(=O)c2ccccc2)cc1F
Relative Density.	1.47 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (124.24 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4848 mL	12.4242 mL	24.8484 mL	124.2421 mL
5 mM	0.4970 mL	2.4848 mL	4.9697 mL	24.8484 mL
10 mM	0.2485 mL	1.2424 mL	2.4848 mL	12.4242 mL
20 mM	0.1242 mL	0.6212 mL	1.2424 mL	6.2121 mL
50 mM	0.0497 mL	0.2485 mL	0.4970 mL	2.4848 mL
100 mM	0.0248 mL	0.1242 mL	0.2485 mL	1.2424 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc