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Search Results for " subfamily "

20

Compounds

Cat No. Product Name Synonyms Targets
T16483 PF-05105679 TRP/TRPV Channel
PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.
T9776 TRPM4 inhibitor 8 TRP/TRPV Channel
TRPM4 inhibitor 8 is an inhibitor of Transient receptor potential melastatin 4(TRPM4) which contributes to viability, migration, cell cycle shift, and adhesion.
T9335 1,1'-Methylenedi-2-naphthol Squoxin Others
1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).
T3719 Daminozide Succinic Acid,DMASA,Aminozide Histone Demethylase
Daminozide (Succinic Acid) is a plant growth regulator, selectively inhibits the KDM2/7 JmjC subfamily.
T28020 Mesendogen TRP/TRPV Channel
Mesendogen is an inhibitor of TRPM6. Mesendogen alters magnesium homeostasis, promotes mesoderm and definitive endoderm differentiation.
T62204 NR2F6 modulator-1 Others
NR2F6 modulator-1 is a potent modulator of nuclear receptor subfamily 2, group F, member 6 (NR2F6). NR2F6 modulator-1 can be used to study immune regulation and modulation of tumour stem cell activity.
T10616 BRM/BRG1 ATP Inhibitor-1 Epigenetic Reader Domain
BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A member 2 (SMARCA2) and BRG1/SMARCA4 ATPase activity inhibitor (IC50...
T16763 RN-1747 TRP/TRPV Channel
RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: 0.77 μM, 4.0 μM, and 4.1 μM for hTRPV4, mTRPV4, and rTRPV4 respectively). RN-1747 also antagonizes TRPM8 (IC50: 4 μM...
T16745 Rhosin hydrochloride Apoptosis , Rho , Ras
Rhosin hydrochloride is an effective and specific RhoA subfamily Rho GTPases inhibitor, which specifically binds to RhoA to inhibit RhoA-GEF interaction (Kd: ~ 0.4 uM). Rhosin hydrochloride does not interact with Cdc42 o...
T2024 A-803467 A 803467,A803467 Sodium Channel
A-803467 is a selective NaV1.8 channel blocker.
TP2158 TRV-120027 TFA TRV-120027 TFA (1234510-46-3 free base) RAAS , Arrestin
TRV120027 TFA is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1R) and engages ß-arrestins while blocking G-protein signaling.
T23429 KDM2/7-IN-1 TC-E 5002 Others
Selective histone demethylase KDM2/7 subfamily inhibitor
T68693 AZ12099548
AZ12099548 is a transient receptor potential cation channel subfamily V member 1 (TRPV1) antagonist.
T71359 ArgTX-93 TFA
ArgTX-93 is a highly potent and subfamily selective antagonist of the NMDARs and AMPARs.
T70716 ArgTX-48 TFA
ArgTX-48 is a highly potent and subfamily selective antagonist of the NMDARs and AMPARs.
T63411 CCG258747
CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.
T82579 Dermaseptin-B9
Dermaseptin-B9, an antimicrobial peptide, has been isolated from the Phyllomedusinae subfamily of frogs [1].
T16746 Rhosin Rho
Rhosin is an effective and specific RhoA subfamily Rho GTPases inhibitor, which specifically binds to RhoA to inhibit RhoA-GEF interaction (Kd: ~ 0.4 uM). Rhosin does not interact with Cdc42 or Rac1, nor the GEF, LARG. R...
T37086 PDDHV
PDDHV is a resiniferatoxin-type phorboid vanilloid with capsaicin-like selectivity for the cloned rat transient receptor potential cation channel subfamily V member 1 (TRPV1), formerly known as vanilloid receptor 1. It i...
TP2287 Rac GTPase fragment Others
Rac GTPase fragment is a peptide with the sequence H2N-Val-Phe-Asp-Glu-Ala-Ile-Arg-Ala-Val-OH, MW= 1019.15. Rac is a subfamily of the Rho family of GTPases, small signaling G proteins (more specifically a GTPase).
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TargetMol