peptide-competitive — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T3624	A-366	A 366,A366	Epigenetic Reader Domain , Histone Methyltransferase
	A-366 is a highly selective peptide-competitive histone methyltransferase G9a inhibitor with IC50s of 3.3 and 38 nM for G9a and GLP, respectively.It is more than 1,000-fold selective for G9a and GLP over the other 21 met...		Epigenetic Reader Domain , Histone Methyltransferase
T26645	Aptiganel	CNS 1102,CNS-1102,CNS1102	NMDAR
	Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.		NMDAR
TP1523	PKG inhibitor peptide TFA (82801-73-8 free base)	PKG inhibitor peptide TFA	PKA
	PKG inhibitor peptide TFA (82801-73-8 free base) is an inhibitor of ATP-competitive cGMP-dependent protein kinase (PKG).		PKA
TP2100	Avexitide	Exendin-3 (9-39) amide,Exendin (9-39)	Glucagon Receptor
	Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.		Glucagon Receptor
TP2103L	[D-p-Cl-Phe6,Leu17]-VIP acetate		Others
	[D-p-Cl-Phe6,Leu17]-VIP acetate is a competitive and selective antagonist of vasoactive intestinal peptide (VIP) receptor (IC50 = 125.8 nM).		Others
T78223	γ-Glu-Tyr	gamma-Glutamyltyrosine,gamma-GLU-TYR
	γ-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide with competitive inhibition of dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.
TP1785L	Peptide T acetate(106362-32-7 free base)		Others , HIV Protease
	Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120. Peptide T is a synthetic octapeptide whose possible mechanism of action is the competitive inhibition of gp120 to the CD4 receptor as well as binding...		Others , HIV Protease
TP1887L1	[Ala107]-MBP (104-118) acetate	[Ala107]-MBP (104-118) acetate(99026-77-4 free base)	PKC
	[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).		PKC
T15387	GLP-1R Antagonist 1		Glucagon Receptor
	GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).		Glucagon Receptor
TP1890L1	MLCK inhibitor peptide 18 acetate	MLCK inhibitor peptide 18 acetate(224579-74-2 free base)	Serine/threonin kinase
	MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA. Cell permeable.		Serine/threonin kinase
T8313	HCH6-1		Others
	HCH6-1 is a competitive Formyl peptide receptor 1 (FPR1) antagonist.		Others
T8691	PD 168368	PD168368	Bombesin Receptor
	PD 168368 is a novel, potent, competitive and selective nonpeptide neuromodulin B receptor (NMB-R) antagonist with inhibitory effects on the gastrin-releasing peptide receptor (GRPR).PD 168368 is a potent mixed agonist o...		Bombesin Receptor
T71280	S 8308
	S 8308 is a weak, but specific and competitive, non-peptide antagonist of AII exerting its inhibitory action at the receptor level.
T69621	BIIE-0246 HCl
	BIIE-0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor. BIIE-0246 displays > 650-fold selectivity over Y1, Y4 and Y5 receptors.
T17281	Z-Ile-Leu-aldehyde	Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII	Others
	Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.		Others
T81448	PKG inhibitor peptide TFA
	PKG inhibitor peptide TFA is an ATP-competitive antagonist of cGMP-dependent protein kinase (PKG), exhibiting a K_i value of 86 μM [1].
TP1887	[Ala107]MBP(104-118)	[Ala107]-MBP (104-118)
	Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).
TP1888	[Ala113]MBP(104-118)	[Ala113]-MBP (104-118)
	Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 28 - 62 mM).
TP1785	Peptide T
	Peptide T is an octapeptide from the V2 region of HIV-1 gp120. Peptide T is a synthetic octapeptide whose possible mechanism of action is the competitive inhibition of gp120 to the CD4 receptor as well as binding to vaso...
T38460	SN52
	SN52 is a powerful, competitive, and cell-permeable inhibitor of NF-κB2. It is a variant of the SN50 peptide. SN52 effectively prevents the nuclear translocation of p52-RelB heterodimers, exhibiting a robust radiosensiti...