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Search Results for " neuromuscular "

20

Compounds

Cat No. Product Name Synonyms Targets
T13491 Neuromuscular-targeting compound 1 Others
Neuromuscular-targeting compound 1 can be used to study muscular dystrophy and neuromuscular-related diseases.
T10059 Neuromuscular Disorder-Targeting Compound 1 Others
Neuromuscular Disorder-Targeting Compound 1 is a compound used in the research of neuromuscular disorders, for example, symptoms of chronic fatigue syndrome and fibromyalgia syndrome.
T0166 Pancuronium dibromide Pancuronium bromide,Pavulon AChR
Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) blocking neuromuscular transmission is achieved by competing ...
T21793 CGP 35348 GABA Receptor
CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after neonatal brain damage in albino mice.
T5326 Sugammadex sodium Org25969,Sugammadex (sodium) Others
Sugammadex sodium (Org25969) , a synthetic derivative of γ-cyclodextrin, is a steroid-based neuromuscular blocker reversing agent.
T1234 5,5-Dimethyloxazolidine-2,4-dione Dimethadion,Dimethadione,Dimethyloxazolidinedione Calcium Channel
5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.
T2227 Hemicholinium 3 Hemicholinium-3,Hemicholine Others , AChE
Hemicholinium 3 is a potent and selective choline uptake blocker.
T6397 Atracurium besylate Tracrium,51W89,BW-33A AChR
Atracurium besylate (51W89) is a non-depolarizing neuromuscular blocking agent with short duration of action. Its lack of significant cardiovascular effects and its lack of dependence on good kidney function for eliminat...
T22371 Mivacurium dichloride Mivacurium chloride AChR
Mivacurium dichloride (Mivacurium chloride) is a non-depolarising, rapid neuromuscular blocker of short duration, used therefore as anesthetic, to provide skeletal muscle relaxation in minor surgical operations, in emerg...
T4497 Amifampridine 3,4-Pyridinediamine,Pyridine-3,4-Diamine,3,4-Diaminopyridine Others
Amifampridine (3,4-Diaminopyridine) is predominantly in the treatment of a number of rare muscle diseases. Amifampridine works by blocking potassium channel efflux in nerve terminals so that action potential duration is ...
T0818 Decamethonium bromide Decacuran,Syncurine AChR , AChE
Decamethonium bromide (Syncurine) is a neuromuscular blocker and nicotinic AChR partial agonist.
T6S0084 Tuberostemonine Tuberstemonine Parasite
1. Tuberostemonine (Tuberstemonine) exhibits relatively higher intestinal permeabilities. 2. Tuberostemonine acts in part as an open-channel blocker at the crayfish neuromuscular junction.
T12481 Pipecuronium bromide RGH-1106 AChR
Pipecuronium bromide (RGH-1106) is a selective and potent nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker, causing muscle relaxation, often in conjunction with antibiotics.
T6684 Succinylcholine Chloride Dihydrate choline chloride succinate,Succinyldicholine dichloride,Suxamethonium Chloride Dihydrate AChR
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
TP1868 Proctolin Others
Proctolin is a bioactive neuropeptide that modulates interneuronal and neuromuscular synaptic transmission in a wide variety of arthropods.
T1259 Pyrantel pamoate Pyrantel embonate Others , Antibiotic , Parasite
Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.
T6751 Acetylcholine iodide Acetylcolina Others
Acetylcholine iodide (Acetylcolina) is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the cent...
T1594 Vecuronium bromide ORG NC 45 AChR
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle relaxant activity.
T3966 Tirasemtiv CK-2017357 Others
Tirasemtiv (CK-2017357)(CK 2017357) is a small-molecule fast-skeletal-troponin activator, with a potential treatment for muscle weakness and neuromuscular dysfunction.
T14094 Acetamiprid AChR
Acetamiprid is a nicotinic acetylcholine receptor (nAChR) agonist. Acetamiprid is a neonicotinoid insecticide used worldwide. It is shown to be associated with neuromuscular and reproductive disorders.
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