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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13491 | Neuromuscular-targeting compound 1 | Others | |
Neuromuscular-targeting compound 1 can be used to study muscular dystrophy and neuromuscular-related diseases. | |||
T10059 | Neuromuscular Disorder-Targeting Compound 1 | Others | |
Neuromuscular Disorder-Targeting Compound 1 is a compound used in the research of neuromuscular disorders, for example, symptoms of chronic fatigue syndrome and fibromyalgia syndrome. | |||
T0166 | Pancuronium dibromide | Pancuronium bromide,Pavulon | AChR |
Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) blocking neuromuscular transmission is achieved by competing ... | |||
T21793 | CGP 35348 | GABA Receptor | |
CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after neonatal brain damage in albino mice. | |||
T5326 | Sugammadex sodium | Org25969,Sugammadex (sodium) | Others |
Sugammadex sodium (Org25969) , a synthetic derivative of γ-cyclodextrin, is a steroid-based neuromuscular blocker reversing agent. | |||
T1234 | 5,5-Dimethyloxazolidine-2,4-dione | Dimethadion,Dimethadione,Dimethyloxazolidinedione | Calcium Channel |
5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE. | |||
T2227 | Hemicholinium 3 | Hemicholinium-3,Hemicholine | Others , AChE |
Hemicholinium 3 is a potent and selective choline uptake blocker. | |||
T6397 | Atracurium besylate | Tracrium,51W89,BW-33A | AChR |
Atracurium besylate (51W89) is a non-depolarizing neuromuscular blocking agent with short duration of action. Its lack of significant cardiovascular effects and its lack of dependence on good kidney function for eliminat... | |||
T22371 | Mivacurium dichloride | Mivacurium chloride | AChR |
Mivacurium dichloride (Mivacurium chloride) is a non-depolarising, rapid neuromuscular blocker of short duration, used therefore as anesthetic, to provide skeletal muscle relaxation in minor surgical operations, in emerg... | |||
T4497 | Amifampridine | 3,4-Pyridinediamine,Pyridine-3,4-Diamine,3,4-Diaminopyridine | Others |
Amifampridine (3,4-Diaminopyridine) is predominantly in the treatment of a number of rare muscle diseases. Amifampridine works by blocking potassium channel efflux in nerve terminals so that action potential duration is ... | |||
T0818 | Decamethonium bromide | Decacuran,Syncurine | AChR , AChE |
Decamethonium bromide (Syncurine) is a neuromuscular blocker and nicotinic AChR partial agonist. | |||
T6S0084 | Tuberostemonine | Tuberstemonine | Parasite |
1. Tuberostemonine (Tuberstemonine) exhibits relatively higher intestinal permeabilities. 2. Tuberostemonine acts in part as an open-channel blocker at the crayfish neuromuscular junction. | |||
T12481 | Pipecuronium bromide | RGH-1106 | AChR |
Pipecuronium bromide (RGH-1106) is a selective and potent nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker, causing muscle relaxation, often in conjunction with antibiotics. | |||
T6684 | Succinylcholine Chloride Dihydrate | choline chloride succinate,Succinyldicholine dichloride,Suxamethonium Chloride Dihydrate | AChR |
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker. | |||
TP1868 | Proctolin | Others | |
Proctolin is a bioactive neuropeptide that modulates interneuronal and neuromuscular synaptic transmission in a wide variety of arthropods. | |||
T1259 | Pyrantel pamoate | Pyrantel embonate | Others , Antibiotic , Parasite |
Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent. | |||
T6751 | Acetylcholine iodide | Acetylcolina | Others |
Acetylcholine iodide (Acetylcolina) is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the cent... | |||
T1594 | Vecuronium bromide | ORG NC 45 | AChR |
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle relaxant activity. | |||
T3966 | Tirasemtiv | CK-2017357 | Others |
Tirasemtiv (CK-2017357)(CK 2017357) is a small-molecule fast-skeletal-troponin activator, with a potential treatment for muscle weakness and neuromuscular dysfunction. | |||
T14094 | Acetamiprid | AChR | |
Acetamiprid is a nicotinic acetylcholine receptor (nAChR) agonist. Acetamiprid is a neonicotinoid insecticide used worldwide. It is shown to be associated with neuromuscular and reproductive disorders. |