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20

Compounds

Cat No. Product Name Synonyms Targets
TN7054 N-Formylcytisine (-)-N-Formylcytisine Others
N-Formylcytisine ((-)-N-Formylcytisine) is a natural product isolated from the stem bark of Maackia amurensis.
T12153 N-type calcium channel blocker-1 Calcium Channel
N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.
T12039 Miglustat N-Butyldeoxynojirimycin,OGT918,NB-DNJ Others
Miglustat (NB-DNJ) is an alkylated product of imino sugar deoxynojirimycin.It is an inhibitor of glucosylceramide synthase, primarily to treat Type I Gaucher disease (GD1).
TQ0155 Miglustat hydrochloride NB-DNJ hydrochloride,N-Butyldeoxynojirimycin hydrochloride,OGT918 hydrochloride Transferase
Miglustat hydrochloride (N-Butyldeoxynojirimycin hydrochloride) is an inhibitor of glucosylceramide synthase and can be used for studies about Type I Gaucher disease.
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T21900 ML-336 Others
ML-336 is an inhibitor of of the Venezuelan equine encephalitis virus (VEEV) strain TC-83.
TP1559L Ziconotide Acetate (107452-89-1 free base) Prialt,Ziconotide Acetate Calcium Channel
Ziconotide Acetate (107452-89-1 free base) (Prialt) is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide Acetate (107452-89-1 free base) acts by binding to N-type calcium chan...
T7334 NP118809 39-1B4 Calcium Channel
NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).
T11517 GV-58 Calcium Channel
GV-58 is a selective N- and P/Q-type Ca2+ channels agonist (EC50: 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel). The inhibitory of GV-58 is 20-fold fewer for CDK kinases activity.
T10659 Ca2+ channel agonist 1 Calcium Channel , CDK
Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.
T12385 PD0176078 PD176078 Calcium Channel
PD0176078 () is a newly blocker of N-type Calcium channel.
T4462 Roflumilast N-oxide PDE
Roflumilast N-oxide is an inhibitor of PDE type 4.
T6S1500 Ginsenoside Rf Ginsenoside-Rf,Panaxoside Rf Calcium Channel , Endogenous Metabolite
Ginsenoside Rf (Panaxoside Rf) is a trace component of ginseng root. Ginsenoside Rf inhibits N-type Ca2+ channel.
T10690 Cav 2.2 blocker 1 Calcium Channel
Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
T0388 Cilnidipine FRC-8653 Calcium Channel
Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.
T36061 N-Desmethyl Sildenafil Desmethylsildenafil,UK-103,320 Drug Metabolite
N-Desmethyl Sildenafil (UK-103,320) (Desmethylsildenafil) is a prominent metabolite of Sildenafil, a potent inhibitor of phosphodiesterase type 5 (PDE5).
T16339 Norverapamil hydrochloride (±)-Norverapamil hydrochloride,D591 hydrochloride Calcium Channel , P-gp , Drug Metabolite
Norverapamil hydrochloride (D591 hydrochloride) ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor.
T16240 N,N'-Diacetyl-L-cystine (Ac-Cys-OH)2,DiNAC Others
N,N'-Diacetyl-L-cystine (DiNAC) is the disulphide dimer of N-acetylcysteine with immunomodulating properties. N,N'-diacetyl-L-cystine also has antiatherosclerotic effects in Watanabe-heritable hyperlipidemic rabbit (WHHL...
T16448 PD173212 Calcium Channel
PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2). PD173212 (0.0017-1.7 μmol/kg, Intraperitoneal Injection.) dose-dependently reduced DNBS-induced visceral hypersensitivity in mice.
T16164 MY-5445 N-(3-chlorophenyl)-4-phenylphthalazin-1-amine PDE
MY-5445 (N-(3-chlorophenyl)-4-phenylphthalazin-1-amine) is a specific inhibitor of phosphodiesterase type 5 (PDE5). MY-5445 selectively inhibits cGMP PDE (Ki:1.3 μM).

Compounds

N-Formylcytisine
TN7054
Synonym: (-)-N-Formylcytisine
Target: Others
N-type calcium channel blocker-1
T12153
Synonym:
Target: Calcium Channel
Miglustat
T12039
Synonym: N-Butyldeoxynojirimycin,OGT918,NB-DNJ
Target: Others
Miglustat hydrochloride
TQ0155
Synonym: NB-DNJ hydrochloride,N-Butyldeoxynojirimycin hydrochloride,OGT918 hydrochloride
Target: Transferase
OMDM-1
T12302
Synonym: (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide
Target: Endogenous Metabolite
ML-336
T21900
Synonym:
Target: Others
Ziconotide Acetate (107452-89-1 free base)
TP1559L
Synonym: Prialt,Ziconotide Acetate
Target: Calcium Channel
NP118809
T7334
Synonym: 39-1B4
Target: Calcium Channel
GV-58
T11517
Synonym:
Target: Calcium Channel
Ca2+ channel agonist 1
T10659
Synonym:
Target: Calcium Channel, CDK
PD0176078
T12385
Synonym: PD176078
Target: Calcium Channel
Roflumilast N-oxide
T4462
Synonym:
Target: PDE
Ginsenoside Rf
T6S1500
Synonym: Ginsenoside-Rf,Panaxoside Rf
Target: Calcium Channel, Endogenous Metabolite
Cav 2.2 blocker 1
T10690
Synonym:
Target: Calcium Channel
Cilnidipine
T0388
Synonym: FRC-8653
Target: Calcium Channel
N-Desmethyl Sildenafil
T36061
Synonym: Desmethylsildenafil,UK-103,320
Target: Drug Metabolite
Norverapamil hydrochloride
T16339
Synonym: (±)-Norverapamil hydrochloride,D591 hydrochloride
Target: Calcium Channel, P-gp, Drug Metabolite
N,N'-Diacetyl-L-cystine
T16240
Synonym: (Ac-Cys-OH)2,DiNAC
Target: Others
PD173212
T16448
Synonym:
Target: Calcium Channel
MY-5445
T16164
Synonym: N-(3-chlorophenyl)-4-phenylphthalazin-1-amine
Target: PDE
1 2 3 4 5
TargetMol