Powder: -20°C for 3 years | In solvent: -80°C for 1 year
NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
100 mg | In stock | $ 81.00 | |
200 mg | In stock | $ 98.00 | |
500 mg | In stock | $ 126.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 50.00 |
Description | NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM). |
Targets&IC50 | Ca2+ channel, N-type:0.11 μM |
In vitro | NP118809 with a total linker length of 3 carbons (n = 1) and which exhibited approximately a 500-fold increased N-type channel blockade compared to compounds in this series with linkers either shorter (n = 0, 2a) or longer (n = 2 4, (2c e). Examination of the effect of NP118809 on functional L-type calcium channel activity showed that this compound was approximately 111-fold more selective for N-type channels[1] |
Synonyms | 39-1B4 |
Molecular Weight | 460.61 |
Formula | C32H32N2O |
CAS No. | 41332-24-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (108.55 mM)
You can also refer to dose conversion for different animals. More
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NP118809 41332-24-5 Membrane transporter/Ion channel Metabolism Calcium Channel NP 118809 Inhibitor inhibit 39-1B4 Ca2+ channels NP-118809 Ca channels inhibitor