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Search Results for " mpa "

20

Compounds

Cat No. Product Name Synonyms Targets
T1171L Methylprednisolone Aceponate MPA,SH 440,SH-440,SH440,Advantan Others
Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.
T19416 Medroxyprogesterone acetate D3 MPA D3,Medroxyprogesterone 17-acetate D3 Others
Medroxyprogesterone acetate D3 is deuterium labeled Medroxyprogesterone acetate. Medroxyprogesterone acetate is a widely used synthetic steroid by its interaction with progesterone, androgen and glucocorticoid receptors.
T67798 (2RS)-FPMPA FPMPA HIV Protease
(2RS)-FPMPA(FPMPA) has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).
T13173 TMPA Others , AMPK
TMPA is a nuclear receptor Nur77 and LKB1 interaction antagonist.
T11186 EMPA OX Receptor
EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM respectively)
T1766 Empagliflozin BI 10773 SGLT
Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6. Empagliflozin is used for the treatment of type 2 diabetes.
T61813 AMPA receptor antagonist-3 iGluR
AMPA receptor antagonist-3 is an AMPA receptor antagonist.
T3440 2-PMPA 2-(Phosphonomethyl)pentanedioic acid Carboxypeptidase
2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).
T34609 Selurampanel BGG-492,BGG 492,BGG492 iGluR
Selurampanel (BGG492) is an orally active and selective competitive AMPA glutamate receptor antagonist, a quinazoline-dione sulfonamide. selurampanel is used in the study of epilepsy, migraine and tinnitus.
T17179 Tulrampator CX-1632,S-47445 iGluR
Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.
T16977 Talampanel GYKI-53773,LY-300164 Apoptosis , GluR
Talampanel (LY-300164) is an orally and selective α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptor antagonist with anti-seizure activity. Talampanel (IVAX) has neuroprotective effects in rodent stroke models.
T61068 AMPA receptor antagonist-2 iGluR
AMPA receptor antagonist-2 is an AMPA receptor antagonist.
T37734 AMPA receptor modulator-2 GluR
AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor[1]. pIC50 = -lgIC50. [1]. BERRY CYNTHIA G B (US), et al. AZABENZIMIDAZOLES AND THEIR USE AS AM...
T21761 HNMPA IGF-1R
HNMPA is a membrane impermeable inhibitor of insulin receptor tyrosine kinase. HNMPA inhibits tyrosine and serine autophosphorylation by the human insulin receptor. HNMPA exhibits no effect on cyclic AMP-dependent prote...
T19232 CMC-Na (Viscosity:800-1200 mPa.s) CMC-Na (Viscosity:800-1200 mPa.s) Others
Sodium carboxymethyl cellulose (CMC-Na) (Viscosity:800-1200 mPa.s) is a water-soluble cellulose, commonly used as a co-solvent in animal experiments, and is essentially non-toxic to animals.
T3957 Farampator Org24448,CX-691 GluR , iGluR
Farampator (CX-691) (CX-691;Org24448) is a positive modulator of AMPA receptor.
T10307 AMPA receptor modulator-1 iGluR
AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.
T31208 Dasolampanel NGX-426,NGX 426,NGX426 GluR , iGluR
Dasolampanel (NGX-426) is an orally available ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders, including neuropathic pain and migraine.
T15820 Mibampator LY451395 iGluR
Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.
T79191 AMPA receptor modulator-5 iGluR
AMPA Receptor Modulator-5 (Example 217) serves as an AMPA receptor modulator, utilized in neurological disease research [1].
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TargetMol