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Search Results for " ht1 "

20

Compounds

Cat No. Product Name Synonyms Targets
T24055 FAUC 213 FAUC213,FAUC-213 Dopamine Receptor
FAUC 213 is a selective full antagonist of the dopamine D4 receptor.
T1684 Nitisinone NTBC,SC0735,Nitisone Others , Reactive Oxygen Species
Nitisinone (SC0735)(SC0735) is an enzyme 4-hydroxyphenylpyruvate dioxygenase inhibitor.
T37197 5-HT1A modulator 2 hydrochloride 5-HT Receptor
5-HT1A modulator 2 hydrochloride, a derivative of 8-OH-DPAT , is a modulator of 5-HT1A with a Ki of 53 nM for 5-HT1A binding[1]. [1]. Naiman, N.,et al. 2-(Alkylamino)tetralin derivatives: interaction with 5-HT1A serotoni...
T10168 5-HT1A modulator 1 5-HT1Amodulator1 Phospholipase , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
T62843 5-HT1A antagonist 1
5-HT1A antagonist 1 (compound 6f) is a potent and selective 5-HT1Areceptor antagonist (Ki: 35 nM). 5-HT1A antagonist 1 can be used in the study of central nervous system disorders.
T27558 HT1042 HT 1042,HT-1042
HT1042 is an inhibitor of the β5i component of the 20S proteasome complex, it is used to aid in the treatment of inflammatory diseases, autoimmune and hematologic malignancies.
T0203 Sumatriptan succinate GR 43175 5-HT Receptor
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.
T8666 Naratriptan 5-HT Receptor
Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.
T12207 NEO 376 SPI-376 Dopamine Receptor , 5-HT Receptor , GABA Receptor
NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
T10872L CP 96021 5-HT Receptor
CP 96021 is a group of 5-HT1 receptors and 5-HT2 receptors antagonists that have anti-inflammatory properties and are non-non-self anti-ulcer compounds for the treatment of gastrointestinal tract and respiratory asthma.
T22534 8-Hydroxy-DPAT hydrobromide 8-OH-DPAT hydrobromide 5-HT Receptor
8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19. 8-Hydroxy-DPAT hydrobromide has a selectivity of almost 1000 fold for a subtype...
T23382 Spiroxatrine R 5188 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2, and dopamine receptors.Spiroxatrine may be used in the stu...
T21385 Cinitapride Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove 5-HT Receptor
Cinitapride (Blaston) is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia. Cinitapride acts as an antag...
T4978 Sarpogrelate hydrochloride MCI-9042 5-HT Receptor
Sarpogrelate hydrochloride (MCI-9042) , a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. Target: 5-HT2 Recepter Sarpogrelate is a drug which acts as an antagonist at ...
T1512 Rizatriptan benzoate MK-462 Benzoate 5-HT Receptor
Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine headaches.
T0162 Quetiapine ICI204636,Quetiapin Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR , Histamine Receptor
Quetiapine (ICI204636) is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapine' action is thought by mediated through antago...
T6602 Naratriptan hydrochloride Naratriptan HCl,Amerge,Naramig,GR-85548A hydrochloride 5-HT Receptor
Naratriptan Hydrochloride is the hydrochloride salt form of naratriptan, a sulfonamide with selective serotonin (5-HT) 1 receptor agonistic activity and anti-migraine property. Naratriptan hydrochloride (GR-85548A hydroc...
T23405 Sumatriptan Others
Sumatriptan succinate is a selective 5-HT1 receptor agonist with specificity towards 5-HT1D, 5-HT1B, and 5-HT1A.
T68176 Isamoltane
Isamoltane is a serotonin 5-HT1 Receptor Antagonist
T4375 Methiothepin maleate Metitepine 5-HT Receptor
Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.

Compounds

FAUC 213
T24055
Synonym: FAUC213,FAUC-213
Target: Dopamine Receptor
Nitisinone
T1684
Synonym: NTBC,SC0735,Nitisone
Target: Others, Reactive Oxygen Species
5-HT1A modulator 2 hydrochloride
T37197
Synonym:
Target: 5-HT Receptor
5-HT1A modulator 1
T10168
Synonym: 5-HT1Amodulator1
Target: Phospholipase, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
5-HT1A antagonist 1
T62843
Synonym:
Target:
HT1042
T27558
Synonym: HT 1042,HT-1042
Target:
Sumatriptan succinate
T0203
Synonym: GR 43175
Target: 5-HT Receptor
Naratriptan
T8666
Synonym:
Target: 5-HT Receptor
NEO 376
T12207
Synonym: SPI-376
Target: Dopamine Receptor, 5-HT Receptor, GABA Receptor
CP 96021
T10872L
Synonym:
Target: 5-HT Receptor
8-Hydroxy-DPAT hydrobromide
T22534
Synonym: 8-OH-DPAT hydrobromide
Target: 5-HT Receptor
Spiroxatrine
T23382
Synonym: R 5188
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Cinitapride
T21385
Synonym: Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove
Target: 5-HT Receptor
Sarpogrelate hydrochloride
T4978
Synonym: MCI-9042
Target: 5-HT Receptor
Rizatriptan benzoate
T1512
Synonym: MK-462 Benzoate
Target: 5-HT Receptor
Quetiapine
T0162
Synonym: ICI204636,Quetiapin
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor
Naratriptan hydrochloride
T6602
Synonym: Naratriptan HCl,Amerge,Naramig,GR-85548A hydrochloride
Target: 5-HT Receptor
Sumatriptan
T23405
Synonym:
Target: Others
Isamoltane
T68176
Synonym:
Target:
Methiothepin maleate
T4375
Synonym: Metitepine
Target: 5-HT Receptor
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TargetMol